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Report error Found 202 for UniProtKB: Q28838
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM85099(SDZ SER 082 FUMARATE | CAS_141474-54-6 | SDZ SER-0...)
Affinity DataKd:  999nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor of calf brain cortex using [3H]clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM85099(SDZ SER 082 FUMARATE | CAS_141474-54-6 | SDZ SER-0...)
Affinity DataKd:  1.00E+3nMAssay Description:Binding affinity towards Alpha-2 adrenergic receptor of calf brain cortex using [3H]clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2020
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016897(2-(2,6-dichloroanilino)-2-imidazoline | 2-(2,6-dic...)
Affinity DataIC50: 2nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50027226(3-Methyl-1,2,3,4,4a,8-hexahydro-7-thia-3,12b-diaza...)
Affinity DataIC50: 2nMAssay Description:In vitro binding affinity towards alpha-adrenoceptor of calf cortex membrane Site A using [3H]clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50027227(3-Methyl-1,2,3,4,4a,8-hexahydro-5-thia-3,12b-diaza...)
Affinity DataIC50: 3nMAssay Description:In vitro binding affinity towards alpha-adrenoceptor of calf cortex membrane Site B using [3H]-clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50027227(3-Methyl-1,2,3,4,4a,8-hexahydro-5-thia-3,12b-diaza...)
Affinity DataIC50: 3nMAssay Description:In vitro binding affinity towards alpha-adrenoceptor of calf cortex membrane Site A using [3H]clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50027226(3-Methyl-1,2,3,4,4a,8-hexahydro-7-thia-3,12b-diaza...)
Affinity DataIC50: 3nMAssay Description:In vitro binding affinity towards alpha-adrenoceptor of calf cortex membrane Site B using [3H]-clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM31005(MIANSERIN HYDROCHLORIDE | SMR000058472 | MLS000069...)
Affinity DataIC50: 6nMAssay Description:In vitro binding affinity towards alpha-adrenoceptor of calf cortex membrane Site B using [3H]-clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50224790(CHEMBL333794)
Affinity DataIC50: 7nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
LigandPNGBDBM31005(MIANSERIN HYDROCHLORIDE | SMR000058472 | MLS000069...)
Affinity DataIC50: 20nMAssay Description:In vitro binding affinity towards alpha-adrenoceptor of calf cortex membrane Site A using [3H]clonidineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50224793(CHEMBL330997)
Affinity DataIC50: 27nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
LigandPNGBDBM50224791(RU-29717 | CHEMBL333795)
Affinity DataIC50: 31nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
LigandPNGBDBM50224790(CHEMBL333794)
Affinity DataIC50: 34nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016882(CHEMBL263574 | 1-Butyl-2,3,4,4a,10,10a-hexahydro-1...)
Affinity DataIC50: 39nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50017543(9-Methylsulfanylmethyl-7-propyl-4,6,6a,7,8,9,10,10...)
Affinity DataIC50: 41nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
LigandPNGBDBM50224795(CHEMBL332337)
Affinity DataIC50: 46nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
LigandPNGBDBM50224794(CHEMBL121653)
Affinity DataIC50: 55nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016890(CHEMBL163281 | 5-Methoxy-1-propyl-2,3,4,4a,10,10a-...)
Affinity DataIC50: 71nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016884(CHEMBL162170 | 1-Propyl-2,3,4,4a,10,10a-hexahydro-...)
Affinity DataIC50: 77nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016898(CHEMBL163532 | 1-Propyl-2,3,4,4a,10,10a-hexahydro-...)
Affinity DataIC50: 88nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036857(2-Methoxy-N-{4-[(5-methoxy-chroman-3-yl)-propyl-am...)
Affinity DataIC50: 100nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036873(8-{5-[(5-Methoxy-chroman-3-yl)-propyl-amino]-penty...)
Affinity DataIC50: 100nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
LigandPNGBDBM50027226(3-Methyl-1,2,3,4,4a,8-hexahydro-7-thia-3,12b-diaza...)
Affinity DataIC50: 100nMAssay Description:In vitro binding affinity of alpha-adrenoceptor by interacting with high affinity, [3H]serotonin from calf caudate nucleusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016895(CHEMBL349824 | 5-Methoxy-1-propyl-2,3,10,10a-tetra...)
Affinity DataIC50: 151nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50224792(CHEMBL332546)
Affinity DataIC50: 206nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016881(CHEMBL163803 | 1-Propyl-2,3,10,10a-tetrahydro-1H-9...)
Affinity DataIC50: 208nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016885(CHEMBL162282 | 1-Propyl-2,3,4,4a,10,10a-hexahydro-...)
Affinity DataIC50: 249nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM31005(MIANSERIN HYDROCHLORIDE | SMR000058472 | MLS000069...)
Affinity DataIC50: 300nMAssay Description:In vitro binding affinity of alpha-adrenoceptor by interacting with high affinity [3H]5-HT from calf caudate nucleusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016883(CHEMBL161947 | 1-Propyl-2,3,4,4a,10,10a-hexahydro-...)
Affinity DataIC50: 362nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036849(1-{4-[(5-Methoxy-chroman-3-yl)-propyl-amino]-butyl...)
Affinity DataIC50: 400nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036847(N-{3-[(5-Methoxy-chroman-3-yl)-propyl-amino]-propy...)
Affinity DataIC50: 500nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
LigandPNGBDBM50027227(3-Methyl-1,2,3,4,4a,8-hexahydro-5-thia-3,12b-diaza...)
Affinity DataIC50: 500nMAssay Description:In vitro binding affinity of alpha-adrenoceptor by interacting with high affinity [3H]5-HT from calf caudate nucleusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016891(CHEMBL162510 | 5-Methoxy-7-methyl-1-propyl-2,3,4,4...)
Affinity DataIC50: 504nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM81993(Bromocriptine+ (GTP+) | BROMOCRIPTINE | Bromocript...)
Affinity DataIC50: 514nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016888(CHEMBL162955 | 1-Propyl-2,3,4,4a,10,10a-hexahydro-...)
Affinity DataIC50: 559nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016894(CHEMBL163061 | 1-Propyl-2,3,10,10a-tetrahydro-1H-9...)
Affinity DataIC50: 634nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016892(CHEMBL162449 | 5-Methoxy-1,7-dimethyl-2,3,4,4a,10,...)
Affinity DataIC50: 946nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036861(2-{3-[(5-Methoxy-chroman-3-yl)-propyl-amino]-propy...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM21393(cid_1220 | CHEMBL56 | 7-(dipropylamino)-5,6,7,8-te...)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50016886(CHEMBL422024 | 1,5-Dimethyl-2,3,4,4a,10,10a-hexahy...)
Affinity DataIC50: 1.02E+3nMAssay Description:Concentration necessary to achieve half maximal inhibition of [3H]clonidine binding to Alpha-2 adrenergic receptor at 1 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50224790(CHEMBL333794)
Affinity DataIC50: 1.35E+3nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
LigandPNGBDBM50224790(CHEMBL333794)
Affinity DataIC50: 1.35E+3nMAssay Description:In vitro affinity for alpha adrenergic receptor by displacement of 3[H]clonidine in calf cerebral cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2018
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036859(N-{4-[(5-Methoxy-chroman-3-yl)-propyl-amino]-butyl...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036844(2-{4-[(5-Methoxy-chroman-3-yl)-propyl-amino]-butyl...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036865(8-{3-[(5-Methoxy-chroman-3-yl)-propyl-amino]-propo...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036859(N-{4-[(5-Methoxy-chroman-3-yl)-propyl-amino]-butyl...)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036864(3-Dipropylamino-chroman-5-ol | CHEMBL27995)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50005127(1,1-Dioxo-2-[4-(4-pyrimidin-2-yl-piperazin-1-yl)-b...)
Affinity DataIC50: 2.80E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036854(1-(5-Methoxy-chroman-3-yl)-pyrrolidine | CHEMBL285...)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
TargetAlpha-2A adrenergic receptor(Bovine)
Sandoz Pharma

Curated by ChEMBL
LigandPNGBDBM50036867(2-[4-(5-Methoxy-chroman-3-ylamino)-butyl]-isoindol...)
Affinity DataIC50: 4.00E+3nMAssay Description:Binding affinity against alpha-2 adrenergic receptor in calf frontal cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/27/2012
Entry Details Article
PubMed
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