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TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326010(Dehydromutactin | CHEMBL1242196)
Affinity DataKd:  9nMAssay Description:Inhibition of recombinant full length HuR assessed as protein interaction with TMR-labeled A/U-rich element of COX2 by confocal fluctuation spectrosc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326009(5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...)
Affinity DataKd:  0.100nMAssay Description:Inhibition of recombinant HuR RRM1/RRM2 domain assessed as protein dimerization with TMR-labeled A/U-rich element of TNFalpha by confocal fluctuation...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50270003(CHEMBL4075458)
Affinity DataKd:  4.50E+3nMAssay Description:Binding affinity to human full length recombinant HuR expressed in Escherichia coli Rosetta DH5alpha measured for 30 mins by DMR analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2020
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326011(Okicenone | CHEMBL1240971)
Affinity DataKd:  85nMAssay Description:Binding affinity to recombinant full length HuR assessed as protein dimerization with TMR-labeled A/U-rich element of IL-2 by confocal fluctuation sp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326009(5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...)
Affinity DataKd:  420nMAssay Description:Binding affinity recombinant HuR RRM1/RRM2 domain by confocal fluctuation spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326009(5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...)
Affinity DataKd:  230nMAssay Description:Inhibition of recombinant HuR RRM1/RRM2 domain assessed as protein interaction with TMR-labeled A/U-rich element of IL-2 by confocal fluctuation spec...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326010(Dehydromutactin | CHEMBL1242196)
Affinity DataKd:  6nMAssay Description:Binding affinity to recombinant full length HuR assessed as protein dimerization with TMR-labeled A/U-rich element of COX2 by confocal fluctuation sp...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326010(Dehydromutactin | CHEMBL1242196)
Affinity DataKd:  9nMAssay Description:Inhibition of recombinant full length HuR assessed as protein interaction with TMR-labeled A/U-rich element of IL-2 by confocal fluctuation spectrosc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326010(Dehydromutactin | CHEMBL1242196)
Affinity DataKd:  0.100nMAssay Description:Inhibition of recombinant full length HuR assessed as protein dimerization with TMR-labeled A/U-rich element of IL-2 by confocal fluctuation spectros...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326009(5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...)
Affinity DataKd:  0.100nMAssay Description:Inhibition of recombinant HuR RRM1/RRM2 domain assessed as protein dimerization with TMR-labeled A/U-rich element of IL-2 by confocal fluctuation spe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326010(Dehydromutactin | CHEMBL1242196)
Affinity DataKd:  0.0100nMAssay Description:Inhibition of recombinant full length HuR assessed as protein dimerization with TMR-labeled A/U-rich element of COX2 by confocal fluctuation spectros...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326011(Okicenone | CHEMBL1240971)
Affinity DataKd:  90nMAssay Description:Binding affinity to HuR after 24 hrs by microdialysis methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50326009(5,8-dihydroxy-3-methylnaphtho[2,3-c]furan-4(9H)-on...)
Affinity DataKd:  14nMAssay Description:Inhibition of recombinant HuR RRM1/RRM2 domain assessed as protein interaction with TMR-labeled A/U-rich element of TNFalpha by confocal fluctuation ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/10/2011
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423877(Dihydrotanshinone I | DIHYDROTANSHINONE | acs.jmed...)
Affinity DataIC50: 68nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE TNFalpha complex formation after 90 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50423877(Dihydrotanshinone I | DIHYDROTANSHINONE | acs.jmed...)
Affinity DataIC50: 149nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE TNFalpha complex formation after 3 hrs by REMSA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50240691(CHEMBL4061748)
Affinity DataIC50: 380nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE TNFalpha complex formation after 20 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM7460(2-(3,4-dihydroxyphenyl)-3,5,7-trihydroxy-chromone;...)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE TNFalpha complex formation after 20 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50746(5,7-dimethoxy-8-[1-(4-methoxyphenyl)-3-oxidanylide...)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of Mushashi1 transcript complex formation after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM200225(cid_5992379)
Affinity DataIC50: 2.70E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50240685(CHEMBL1522581)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of Mushashi1 transcript complex formation after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50745(MLS000879482 | 3-(5,7-dimethoxy-2-oxidanylidene-4-...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of Mushashi1 transcript complex formation after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM83193(cid_260346 | MLS002695075 | ethyl 2-oxidanylidene-...)
Affinity DataIC50: 4.60E+3nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM51309(MLS000879474 | 5,7-dimethoxy-8-[1-(4-methoxyphenyl...)
Affinity DataIC50: 5.10E+3nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of Mushashi1 transcript complex formation after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50240686(CHEMBL4095140)
Affinity DataIC50: 6.21E+3nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE TNFalpha complex formation after 20 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50240684(CHEMBL1309685)
Affinity DataIC50: 6.60E+3nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of Mushashi1 transcript complex formation after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM61111(5,7-dimethoxy-8-[3-oxo-3-pyrrolidin-1-yl-1-(3,4,5-...)
Affinity DataIC50: 6.70E+3nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of Mushashi1 transcript complex formation after 2 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50746(5,7-dimethoxy-8-[1-(4-methoxyphenyl)-3-oxidanylide...)
Affinity DataIC50: 8.20E+3nMAssay Description:Inhibition of ELAV1 RRM1/RRM2 domains (unknown origin) interaction with ARE sequence of Mushashi1 transcript after 2 hrs by AlphaLISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50240685(CHEMBL1522581)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of ELAV1 RRM1/RRM2 domains (unknown origin) interaction with ARE sequence of Mushashi1 transcript after 2 hrs by AlphaLISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50745(MLS000879482 | 3-(5,7-dimethoxy-2-oxidanylidene-4-...)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of ELAV1 RRM1/RRM2 domains (unknown origin) interaction with ARE sequence of Mushashi1 transcript after 2 hrs by AlphaLISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM200223(cid_3034178)
Affinity DataIC50: 1.47E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM51309(MLS000879474 | 5,7-dimethoxy-8-[1-(4-methoxyphenyl...)
Affinity DataIC50: 1.57E+4nMAssay Description:Inhibition of ELAV1 RRM1/RRM2 domains (unknown origin) interaction with ARE sequence of Mushashi1 transcript after 2 hrs by AlphaLISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50240684(CHEMBL1309685)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibition of ELAV1 RRM1/RRM2 domains (unknown origin) interaction with ARE sequence of Mushashi1 transcript after 2 hrs by AlphaLISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM200224(cid_247668)
Affinity DataIC50: 1.67E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM200227(cid_374010)
Affinity DataIC50: 1.74E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM61111(5,7-dimethoxy-8-[3-oxo-3-pyrrolidin-1-yl-1-(3,4,5-...)
Affinity DataIC50: 1.76E+4nMAssay Description:Inhibition of ELAV1 RRM1/RRM2 domains (unknown origin) interaction with ARE sequence of Mushashi1 transcript after 2 hrs by AlphaLISA methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM200226(cid_83851)
Affinity DataIC50: 2.17E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM128146(SMR001527404 | cid_239577 | 3,5-bis(2,5-dioxopyrro...)
Affinity DataIC50: 2.69E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM94953(SMR000528071 | 5-amino-2-(4-methylanilino)benzenes...)
Affinity DataIC50: 4.10E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50240687(CHEMBL4066821)
Affinity DataIC50: 4.19E+4nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of c-fos complex formation by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM283(Coumarin-Based, DNA Gyrase Inhibitor | cid_5467792...)
Affinity DataIC50: 4.19E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM82867(6-penta-1,3-diynyl-2-pyranone | MLS000737691 | SMR...)
Affinity DataIC50: 4.44E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM94953(SMR000528071 | 5-amino-2-(4-methylanilino)benzenes...)
Affinity DataIC50: 4.44E+4nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of c-fos complex formation by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50240688(CHEMBL4077803)
Affinity DataIC50: 6.96E+4nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of c-fos complex formation by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM89219(SMR001574695 | MLS002707303 | cid_276150)
Affinity DataIC50: 6.96E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM82867(6-penta-1,3-diynyl-2-pyranone | MLS000737691 | SMR...)
Affinity DataIC50: 9.74E+4nMAssay Description:Inhibition of ELAV1 (unknown origin)-ARE sequence of c-fos complex formation by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2019
Entry Details Article
PubMed
TargetELAV-like protein 1 [I180A](Human)
University of Texas Health Science Center

Curated by PubChem BioAssay
LigandPNGBDBM54386(cid_242249 | MLS000736670 | N-(3-nitrophenyl)-1-ox...)
Affinity DataIC50: 9.74E+4nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2016
Entry Details
PCBioAssay
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50270003(CHEMBL4075458)
Affinity DataKi:  13nMAssay Description:Binding affinity to human full length recombinant His-tagged HuR expressed in Escherichia coli Rosetta DH5alpha assessed as inhibition of interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2020
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50269995(CHEMBL4064932)
Affinity DataKi:  15nMAssay Description:Binding affinity to human full length recombinant His-tagged HuR expressed in Escherichia coli Rosetta DH5alpha assessed as inhibition of interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2020
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50269992(CHEMBL4095060)
Affinity DataKi:  41nMAssay Description:Binding affinity to human full length recombinant His-tagged HuR expressed in Escherichia coli Rosetta DH5alpha assessed as inhibition of interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2020
Entry Details Article
PubMed
TargetELAV-like protein 1(Human)
Novartis Institutes For Biomedical Research

Curated by ChEMBL
LigandPNGBDBM50269999(CHEMBL4100171)
Affinity DataKi:  48nMAssay Description:Binding affinity to human full length recombinant His-tagged HuR expressed in Escherichia coli Rosetta DH5alpha assessed as inhibition of interaction...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/22/2020
Entry Details Article
PubMed
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