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Report error Found 7 of affinity data for UniProtKB/TrEMBL: Q11128
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101904(GDP-Azasugar analogue | CHEMBL52741)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 1 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM92459(Guanosine Diphosphate | CHEMBL384759 | GDP)
Affinity DataIC50: 6.70E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101904(GDP-Azasugar analogue | CHEMBL52741)
Affinity DataIC50: 8.20E+4nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101907(({[(2R,3S,4R,5R)-5-(2-azaniumyl-6-hydroxy-9H-purin...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50101906(GDP-Azasugar analogue | CHEMBL53188)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against fucosyltransferase (FucT V) in the presence of 10 mM fucosyl acceptor N-acetyllactosamineMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/3/2012
Entry Details Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50366926(CHEMBL609638)
Affinity DataKi:  6.71E+4nMAssay Description:Inhibition of Fucosyltransferase 5 by the compound was evaluated; Weak competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
Target4-galactosyl-N-acetylglucosaminide 3-alpha-L-fucosyltransferase FUT5(Human)
Technische Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50366925(CHEMBL610712)
Affinity DataKi:  8.89E+5nMAssay Description:Inhibition of Fucosyltransferase 5 by the compound was evaluated; Weak competitive inhibitionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed