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Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50085554(Oligoadenylate analogue | 5'-O-MONOPHOSPHORYLADENY...)
Affinity DataEC50:  0.150nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of poly (U) 3'[32P]p5'C3'pMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388147(CHEMBL2058765)
Affinity DataEC50:  6.5nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388146(CHEMBL2058766)
Affinity DataEC50:  4.20nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388145(CHEMBL2057900)
Affinity DataEC50:  53nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50085557(Oligoadenylate analogue | CHEMBL407239)
Affinity DataEC50:  30nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50085557(Oligoadenylate analogue | CHEMBL407239)
Affinity DataEC50:  16nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of poly (U) 3'[32P]p5'C3'pMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50085556(Oligoadenylate analogue | CHEMBL405496)
Affinity DataEC50:  0.680nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of poly (U) 3'[32P]p5'C3'pMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50085559(Oligoadenylate analogue | CHEMBL410213)
Affinity DataEC50:  4.60nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of poly (U) 3'[32P]p5'C3'pMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50085556(Oligoadenylate analogue | CHEMBL405496)
Affinity DataEC50:  0.800nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50085559(Oligoadenylate analogue | CHEMBL410213)
Affinity DataEC50:  4nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388148(CHEMBL2058764)
Affinity DataEC50:  15nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataKd:  0.220nMAssay Description:Displacement of 5'-phosphorylated, 2',5'-oligoadenylate from human recombinant RNase L assessed as decrease in resonance by surface plasma resonanceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataEC50:  0.5nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373177(CHEMBL404038)
Affinity DataKd:  0.0400nMAssay Description:Binding affinity to human recombinant RNase LMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373176(C-5950331 | CHEMBL259633)
Affinity DataKd:  1.20E+4nMAssay Description:Displacement of 5'-phosphorylated, 2',5'-oligoadenylate from human recombinant RNase L assessed as decrease in resonance by surface plasma resonanceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373166(CHEMBL259819)
Affinity DataKd:  1.80E+4nMAssay Description:Displacement of 5'-phosphorylated, 2',5'-oligoadenylate from human recombinant RNase L assessed as decrease in resonance by surface plasma resonanceMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373176(C-5950331 | CHEMBL259633)
Affinity DataEC50:  2.20E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373175(C-5972155 | CHEMBL411931)
Affinity DataEC50:  4.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373174(C-6131864 | CHEMBL265469)
Affinity DataEC50:  7.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373173(CHEMBL410485)
Affinity DataEC50:  4.90E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388157(CHEMBL2057899)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388165(CHEMBL2058185)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388164(CHEMBL2058184)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388163(CHEMBL2058183)
Affinity DataEC50:  300nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388162(CHEMBL2058182)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388161(CHEMBL2057897)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50152834([(2R,3R,4R,5R)-5-(6-amino-9H-purin-9-yl)-4-[({[(2R...)
Affinity DataEC50:  17nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388160(CHEMBL2058186)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388159(CHEMBL2058187)
Affinity DataEC50:  200nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388158(CHEMBL2057898)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50438547(CHEMBL2414866)
Affinity DataEC50:  19nMAssay Description:Activation of human recombinant RNase L endonuclease activity using 6-FAM-UUA UCA AAU UCU UAU UUG CCC CAU UUU UUU GGU UUA-BHQ-1 as substrate assessed...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388156(CHEMBL2057901)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388155(CHEMBL2057902)
Affinity DataEC50:  300nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388154(CHEMBL2058188)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388153(CHEMBL2058189)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388152(CHEMBL2058190)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388151(CHEMBL2058191)
Affinity DataEC50:  300nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388150(CHEMBL2058192)
Affinity DataEC50: >1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50388149(CHEMBL2058763)
Affinity DataEC50:  1.00E+3nMAssay Description:Activation of human RNase L expressed in Escherichia coli BL21 (DE3) cells assessed as RNA cleavage using Cy5-rC11-UU-C7-BHQ2 as substrate by FRET as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50085555(Oligoadenylate analogue | CHEMBL384725)
Affinity DataEC50:  0.700nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50183322(CHEMBL601940)
Affinity DataEC50:  13nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2017
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50309129({[(2R,3R,4R,5R)-4-[({[(2R,3R,4R,5R)-4-[({[(2R,3S,4...)
Affinity DataEC50:  2.30nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2017
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50183278(CHEMBL3819262)
Affinity DataEC50:  84nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2017
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50183271(CHEMBL3819183)
Affinity DataEC50:  2.70nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2017
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50183270(CHEMBL3818262)
Affinity DataEC50:  2.40nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2017
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50183269(CHEMBL3818726)
Affinity DataEC50:  20nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2017
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50183268(CHEMBL3818137)
Affinity DataEC50:  134nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2017
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50183267(CHEMBL3817920)
Affinity DataEC50:  0.450nMAssay Description:Induction of recombinant human RNase L activity expressed in Escherichia coli using F-5'-r(C11U2C7)-3' as substrate by polyacrylamide gel electrophor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2017
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50373171(CHEMBL260229)
Affinity DataEC50:  5.00E+4nMAssay Description:Activation of human recombinant Rnase L assessed as cleavage of FRET RNA probeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target2-5A-dependent ribonuclease(Human)
Gifu University

Curated by ChEMBL
LigandPNGBDBM50085558(Oligoadenylate analogue | CHEMBL402676)
Affinity DataEC50:  0.200nMAssay Description:Activation of purified recombinant human Ribonuclease L by the compound was measured as degradation of [32P]-pC11U2C7More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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