Compile Data Set for Download or QSAR
Report error Found 27 for UniProtKB: P97717
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50060964(5-[(2R)-2-{[2-(2-ethoxyphenoxy)ethyl]amino}propyl]...)
Affinity DataIC50: 1.80nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM39687(cid_5717105 | MLS000532635 | SMR000137574 | CHEMBL...)
Affinity DataIC50: 60nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280829(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280821(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280832(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280818(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280823(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280828(3-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280822(4-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280825(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280831(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280819(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280817(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280827(1'-{2-[4-(5-fluoro-1H-3-indolylmethyl)hexahydro-1-...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280820(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280830(3-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280815(N-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280826(2-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280816(N-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50280824(1-{2-[4-(5-Fluoro-1H-indol-3-ylmethyl)-piperidin-1...)
Affinity DataIC50: 100nMAssay Description:Tested for its binding affinity against Alpha-1 adrenergic receptor; showed no appreciable affinity at concentration specifiedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50270777(CHEMBL4126353)
Affinity DataIC50: 348nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50270778(CHEMBL4126498)
Affinity DataIC50: 577nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50270779(CHEMBL4129778)
Affinity DataIC50: 711nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50270772(CHEMBL4128701)
Affinity DataIC50: 1.07E+3nMAssay Description:Displacement of [3H]prazosin from alpha1 adrenoceptor in C57BL/6 mouse hippocampal homogenates after 40 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2020
Entry Details Article
PubMed
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Mouse)
The Australian Nuclear Science and Technology Organisation

Curated by ChEMBL
LigandPNGBDBM50078561(CHEMBL416266 | CHEMBL1204203 | Ethanesulfonic acid...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAlpha-1B adrenergic receptor(Mouse)
University of Dundee

US Patent
LigandPNGBDBM186935(US9079895, 23s)
Affinity DataKi:  6.64E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
Go to US Patent

TargetAlpha-1B adrenergic receptor(Mouse)
University of Dundee

US Patent
LigandPNGBDBM186927(US9079895, 19s)
Affinity DataKi:  7.21E+3nMpH: 7.4Assay Description:The detailed experimental protocols for the radioligand and functional receptor assays are available on the NIMH PDSP website at http://pdsp.med.unc....More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2016
Entry Details
Go to US Patent