Compile Data Set for Download or QSAR
Report error Found 345 of affinity data for UniProtKB/TrEMBL: P97639
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193694(N-(2-(diethylamino)quinolin-6-yl)-3-(4-(trifluorom...)
Affinity DataEC50:  830nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193690(N-(2-(2,5-diazabicyclo[2.2.1]heptan-2-yl)quinolin-...)
Affinity DataEC50:  490nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193697(N-(2-aminoquinolin-6-yl)-3-(4-(trifluoromethyl)phe...)
Affinity DataEC50:  720nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193701(N-(2-(cyclopentyl(methyl)amino)quinolin-6-yl)-3-(4...)
Affinity DataEC50:  350nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193682(N-(2-(cyclohexyl(methyl)amino)quinolin-6-yl)-3-(4-...)
Affinity DataEC50:  1.20E+3nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193695(N-(2-(methylamino)quinolin-6-yl)-3-(4-(trifluorome...)
Affinity DataEC50:  330nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50241102(N-(2-(azepan-1-yl)quinolin-6-yl)-3-(4-(trifluorome...)
Affinity DataEC50:  1.80E+3nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193675(N-(2-(3-(3-methylureido)pyrrolidin-1-yl)quinolin-6...)
Affinity DataEC50:  30nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193687(N-(2-(3-acetamidopyrrolidin-1-yl)quinolin-6-yl)-3-...)
Affinity DataEC50:  440nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193699(N-(2-(piperidin-1-yl)quinolin-6-yl)-3-(4-(trifluor...)
Affinity DataEC50:  110nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193703(N-(2-(3-aminopyrrolidin-1-yl)quinolin-6-yl)-3-(4-(...)
Affinity DataEC50:  200nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193677(N-(2-(methyl(propyl)amino)quinolin-6-yl)-3-(4-(tri...)
Affinity DataEC50:  140nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193681(N-(2-(isopropyl(methyl)amino)quinolin-6-yl)-3-(4-(...)
Affinity DataEC50:  140nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193676(N-(2-(dimethylamino)quinolin-6-yl)-3-(4-(trifluoro...)
Affinity DataEC50:  320nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193684(N-(2-(2-oxa-5-azabicyclo[2.2.1]heptan-5-yl)quinoli...)
Affinity DataEC50:  70nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193678(1-(6-{13-[4-(trifluoromethyl)phenyl]tridecanamido}...)
Affinity DataEC50:  25nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193692(1-(6-(3-(4-(trifluoromethyl)phenyl)propanamido)qui...)
Affinity DataEC50:  50nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193702(N-(2-(2-azabicyclo[2.2.1]heptan-2-yl)quinolin-6-yl...)
Affinity DataEC50:  150nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193686(1-{6-[6-(trifluoromethyl)pyridine-3-amido]quinolin...)
Affinity DataEC50: >1.00E+4nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193674(N-(2-(2-methylpyrrolidin-1-yl)quinolin-6-yl)-3-(4-...)
Affinity DataEC50:  270nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193688(N-(2-(azetidin-1-yl)quinolin-6-yl)-3-(4-(trifluoro...)
Affinity DataEC50:  56nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193680(N-(2-(2-azabicyclo[2.2.2]octan-2-yl)quinolin-6-yl)...)
Affinity DataEC50:  190nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193679(N-(2-(3-methylpyrrolidin-1-yl)quinolin-6-yl)-3-(4-...)
Affinity DataEC50:  400nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193696(N-(2-(3-isobutyramidopyrrolidin-1-yl)quinolin-6-yl...)
Affinity DataEC50:  90nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193691(N-(2-(3-phenylpyrrolidin-1-yl)quinolin-6-yl)-3-(4-...)
Affinity DataEC50:  1.77E+3nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193683(methyl 1-(6-(3-(4-(trifluoromethyl)phenyl)propanam...)
Affinity DataEC50:  580nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193685(N-(1-(6-(3-(4-(trifluoromethyl)phenyl)propanamido)...)
Affinity DataEC50:  110nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193689(N-(2-(dimethylamino)quinolin-6-yl)-3-(4-(trifluoro...)
Affinity DataEC50:  110nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50193700(N-(2-(2,7-diazaspiro[4.4]nonan-2-yl)quinolin-6-yl)...)
Affinity DataEC50:  140nMAssay Description:Stimulation of IP3-coupled mobilization of calcium in HEK293 cells expressing rat MCH-R1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50383522(CHEMBL2032049)
Affinity DataIC50: 0.800nMAssay Description:Antagonist activity at rat MCHR1 assessed inhibition of MCH-mediated intracellular Ca2+ calcium mobilizationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50383112(CHEMBL2029372)
Affinity DataIC50: 1nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50388442(CHEMBL2059408)
Affinity DataIC50: 1.20nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50388443(CHEMBL2059409)
Affinity DataIC50: 1.60nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50383112(CHEMBL2029372)
Affinity DataIC50: 1.70nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 1 hr by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50219047(N-(3-{1-[4-(3,4-difluorophenoxy)benzyl]-4-piperidi...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of rat MCH1R receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50388452(CHEMBL2059420)
Affinity DataIC50: 1.90nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50388444(CHEMBL2059410)
Affinity DataIC50: 2nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50351312(CHEMBL1818800)
Affinity DataIC50: 2.20nMAssay Description:Displacement of [125I]-MCH from rat MCHR1 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50351322(CHEMBL1818810)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]-MCH from rat MCHR1 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50388460(CHEMBL2059513)
Affinity DataIC50: 2.40nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50351313(CHEMBL1818801)
Affinity DataIC50: 2.5nMAssay Description:Displacement of [125I]-MCH from rat MCHR1 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50351308(CHEMBL1818795)
Affinity DataIC50: 2.70nMAssay Description:Displacement of [125I]-MCH from rat MCHR1 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50388457(CHEMBL2059426)
Affinity DataIC50: 2.70nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50388458(CHEMBL2059511)
Affinity DataIC50: 3.40nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50351323(CHEMBL1818811)
Affinity DataIC50: 3.70nMAssay Description:Displacement of [125I]-MCH from rat MCHR1 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50358743(CHEMBL1922270)
Affinity DataIC50: 4nMAssay Description:Antagonist activity at rat MCHR1 expressed in HEK293 cells by aequorin bioluminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50351324(CHEMBL1818901)
Affinity DataIC50: 4.10nMAssay Description:Displacement of [125I]-MCH from rat MCHR1 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50388450(CHEMBL2059418)
Affinity DataIC50: 4.20nMAssay Description:Displacement of [125I]MCH from rat MCHR1 expressed in CHO cells after 60 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50351314(CHEMBL1818802)
Affinity DataIC50: 5.30nMAssay Description:Displacement of [125I]-MCH from rat MCHR1 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetMelanin-concentrating hormone receptor 1(Rat)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50351297(CHEMBL1818783)
Affinity DataIC50: 5.30nMAssay Description:Displacement of [125I]-MCH from rat MCHR1 expressed in CHO cells after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
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