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Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177407(1-(4-hydroxyphenyl)prop-2-en-1-one | 4-acryloylphe...)
Affinity DataIC50: 5.48E+3nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50561618(CHEMBL4746439)
Affinity DataIC50: 9.69E+3nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50632823(CHEMBL4740703)
Affinity DataIC50: 1.22E+4nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177412(4-(aminomethyl)phenol | 4-hydroxybenzylamine | CHE...)
Affinity DataIC50: 1.54E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177410(4-hydroxy-3-nitrobenzaldehyde | CHEMBL378361)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177411(4-hydroxybenzaldehyde | 4-formylphenol | p-formylp...)
Affinity DataIC50: 1.65E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177405(4-hydroxy-3-methoxybenzaldehyde | vanillin | 3-met...)
Affinity DataIC50: 1.71E+4nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50632821(CHEMBL4750359)
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50632822(CHEMBL5408239)
Affinity DataIC50: 1.92E+4nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50632820(CHEMBL5404015)
Affinity DataIC50: 3.10E+4nMAssay Description:Inhibition of GABA-AT (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177402(1-(4-hydroxyphenyl)propan-1-one | Paroxypropione |...)
Affinity DataIC50: 1.76E+5nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177409(1-(4-hydroxyphenyl)ethanone | 4'-hydroxyacetopheno...)
Affinity DataIC50: 1.88E+5nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50376751(ANTHRANILIC ACID)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of GABA-ATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50376752(CHEMBL535644)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of GABA-ATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50376750(CHEMBL541141)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of GABA-ATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177404(Helicide | 4-((2S,3R,4R,5S,6R)-3,4,5-trihydroxy-6-...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50376753(CHEMBL535415)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of GABA-ATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50145829(4-aminobenzoic acid | 4-Aminobenzoesaeure | PABA |...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50226518(3-aminobenzoic acid | 3-Aminobenzoesaeure | m-Amin...)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of GABA-ATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50376755(CHEMBL535643)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of GABA-ATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50376754(CHEMBL535865)
Affinity DataIC50: 5.00E+6nMAssay Description:Inhibition of GABA-ATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177413(4-hydroxy-3-methoxybenzaldehyde oxime | CHEMBL2024...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50139370(4-Methoxy-benzaldehyde | 4-methoxybenzaldehyde | C...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177408(4-Hydroxybenzyl alcohol | 4-(hydroxymethyl)phenol ...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177406(4-hydroxybenzaldehyde oxime | CHEMBL202611)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50177403((2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-(4-(hydroxyme...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM26194(4-Hydroxybenzoate, III | CHEMBL441343 | p-Hydroxyb...)
Affinity DataIC50: 1.00E+6nMAssay Description:Inhibitory activity against GABATMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50009001(CHEMBL8260 | Baicalein | 5,6,7-Trihydroxyflavone |...)
Affinity DataIC50: 1.28E+7nMAssay Description:Inhibition of GABA transaminase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/26/2016
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50024968((2Z)-4-ammonio-2-(fluoromethyl)but-2-enoate | CHEM...)
Affinity DataKi:  9.00E+3nMAssay Description:Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from bacteriaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50021645(N-Phenylthiohydantoic acid | CHEMBL311337 | (3-Phe...)
Affinity DataKi:  9.10E+4nMAssay Description:Compound was tested for inhibition of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50118885(5-Amino-cyclohex-3-enecarboxylic acid | CHEMBL1379...)
Affinity DataKi:  1.00E+5nMAssay Description:Binding affinity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50118884(2-Amino-cyclohex-3-enecarboxylic acid | CHEMBL1419...)
Affinity DataKi:  1.25E+5nMAssay Description:Binding affinity against Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM323799((2S,4S)-4-Aminotetrahydrothiophene-2-carboxylic ac...)
Affinity DataKi:  1.82E+5nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2019
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM466532(US10800753, Compound 17)
Affinity DataKi:  1.82E+5nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50118886(CHEMBL89598 | 4-Amino-hex-5-enoic acid | VIGABATRI...)
Affinity DataKi:  8.50E+5nMAssay Description:Concentration dependent inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50073151(4-(ammoniomethyl)-2,6-difluorobenzenolate | 4-Amin...)
Affinity DataKi:  1.10E+7nMAssay Description:Competitive inhibition of GABA aminotransferase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50118887(2-Amino-cyclohex-3-enecarboxylic acid | CHEMBL1384...)
Affinity DataKi:  1.30E+7nMAssay Description:Concentration dependent inactivation of Gamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50357219(CHEMBL1361446 | VIGABATRIN | US10800753, Compound ...)
Affinity DataKi:  3.20E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM466539(US10800753, Compound 22)
Affinity DataKi:  7.50E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM466538(US10800753, Compound 21)
Affinity DataKi:  3.30E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM466537(US10800753, Compound 20)
Affinity DataKi:  3.40E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM466536(US10800753, Compound 19)
Affinity DataKi:  3.20E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM323800((2R,4S)-4-Aminotetrahydrothiophene-2-carboxylic ac...)
Affinity DataKi:  2.23E+6nMAssay Description:Inhibition constants were determined by monitoring GABA-AT activity in the presence of 0-50 mM concentrations of synthesized analogues using a couple...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/1/2021
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50118888(5-Amino-cyclohex-3-enecarboxylic acid | CHEMBL3368...)
Affinity DataKi:  2.30E+6nMAssay Description:Concentration dependent inactivation of gGamma-amino-N-butyrate transaminaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50082127(3-Aminomethyl-2,6-difluoro-phenol | 3-(ammoniometh...)
Affinity DataKi:  6.30E+6nMAssay Description:Competitive inhibition of GABA aminotransferase (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM50118886(CHEMBL89598 | 4-Amino-hex-5-enoic acid | VIGABATRI...)
Affinity DataKi:  3.20E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2019
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM323805(US10189807, Compound 22)
Affinity DataKi:  7.50E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2019
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM323803(US10189807, Compound 21)
Affinity DataKi:  3.30E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2019
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM323802(US10189807, Compound 20)
Affinity DataKi:  3.40E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2019
Entry Details
Go to US Patent

Target4-aminobutyrate aminotransferase, mitochondrial(Human)
Huazhong University of Science and Technology

Curated by ChEMBL
LigandPNGBDBM323801((4S)-4-Aminotetrahydrothiophene-2-carboxylic acid ...)
Affinity DataKi:  3.20E+6nMAssay Description:Biochemical assays were performed using a Biotek Synergy H1 microplate reader. Prior to their evaluation, initial experiments were performed to confi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/25/2019
Entry Details
Go to US Patent

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