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Report error Found 112 of affinity data for UniProtKB/TrEMBL: P78417
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526135(CHEMBL4593975)
Affinity DataIC50: 0.220nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526136(CHEMBL4513682)
Affinity DataIC50: 0.320nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526140(CHEMBL4463748)
Affinity DataIC50: 5.60nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458512(CHEMBL4215608)
Affinity DataIC50: 21nMAssay Description:Inhibition of human recombinant GSTO1-1 incubated for 30 mins by fluorescence polarization based gel-based competitive ABPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458516(CHEMBL4210652)
Affinity DataIC50: 21nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458512(CHEMBL4215608)
Affinity DataIC50: 21nMAssay Description:Inhibition of SE-Rh binding to human recombinant GSTO1 preincubated with compound for 30 mins followed by SE-Rh addition and measured after 1 hrs by ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM75773(N-[3-(N-(2-chloroacetyl)-4-nitroanilino)propyl]-2,...)
Affinity DataIC50: 23nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526133(CHEMBL4443686)
Affinity DataIC50: 25nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458515(CHEMBL1502738)
Affinity DataIC50: 28nMAssay Description:Inhibition of GSTO1-1 (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526114(CHEMBL4529442)
Affinity DataIC50: 30nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527163(CHEMBL4445050)
Affinity DataIC50: 30nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458516(CHEMBL4210652)
Affinity DataIC50: 31nMAssay Description:Inhibition of GSTO1-1 (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM63200(MLS000583963 | cid_12004949 | SMR000206949 | 2-(3-...)
Affinity DataIC50: 32nMAssay Description:Source (MLPCN Center Name): The Scripps Research Institute Molecular Screening Center (SRIMSC) Center Affiliation: The Scripps Research Institute (TS...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/31/2011
Entry Details
PCBioAssay
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458512(CHEMBL4215608)
Affinity DataIC50: 35nMAssay Description:Inhibition of GSTO1-1 in human MDA-MB-231 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458512(CHEMBL4215608)
Affinity DataIC50: 35nMAssay Description:Inhibition of SE-Rh binding to human recombinant GSTO1 in human MDA-MB-435 cells incubated for 1 hrs by SDS-PAGE based fluorescence analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458522(CHEMBL4203414)
Affinity DataIC50: 40nMAssay Description:Inhibition of GSTO1-1 (unknown origin) by 4-NPG substrate based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526117(CHEMBL4568270)
Affinity DataIC50: 40nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526152(CHEMBL4454963)
Affinity DataIC50: 51nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458520(CHEMBL1486332)
Affinity DataIC50: 54nMAssay Description:Inhibition of GSTO1-1 (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527182(CHEMBL4458115)
Affinity DataIC50: 60nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527184(CHEMBL4454026)
Affinity DataIC50: 70nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526130(CHEMBL4443397)
Affinity DataIC50: 80nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527162(CHEMBL4458365)
Affinity DataIC50: 80nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527169(CHEMBL4437777)
Affinity DataIC50: 110nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM54247(MLS000590567 | cid_3850682 | 2-chloro-N-[(3,4-dime...)
Affinity DataIC50: 120nMAssay Description:Inhibition of GSTO1-1 (unknown origin) by 4-NPG substrate based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458516(CHEMBL4210652)
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527180(CHEMBL4588856)
Affinity DataIC50: 130nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50277889(CHEMBL451887 | CARFILZOMIB)
Affinity DataIC50: 150nMAssay Description:Inhibition of GSTO1-1 (unknown origin) pre-incubated for 1 hr before GSH addition by CDNB-GSH conjugation assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526129(CHEMBL4435063)
Affinity DataIC50: 150nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527179(CHEMBL4475326)
Affinity DataIC50: 150nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527167(CHEMBL4445668)
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527186(CHEMBL4449225)
Affinity DataIC50: 160nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526112(CHEMBL4463910)
Affinity DataIC50: 170nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527188(CHEMBL4465385)
Affinity DataIC50: 180nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526153(CHEMBL4525870)
Affinity DataIC50: 190nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527170(CHEMBL4520358)
Affinity DataIC50: 200nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527191(CHEMBL4544892)
Affinity DataIC50: 210nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526137(CHEMBL4462744)
Affinity DataIC50: 220nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526131(CHEMBL4455136)
Affinity DataIC50: 230nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50155925(CHEMBL3781794)
Affinity DataIC50: 250nMAssay Description:Irreversible inhibition of GSTO 1-1 in LPS activated human monocytes after 30 mins by ELISA analysis in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2017
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527166(CHEMBL4589666)
Affinity DataIC50: 250nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526127(CHEMBL4459484)
Affinity DataIC50: 270nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526119(CHEMBL4473088)
Affinity DataIC50: 300nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50527187(CHEMBL4441594)
Affinity DataIC50: 340nMAssay Description:Inhibition of recombinant GSTO1-1 (unknown origin) expressed in Escherichia coli using S-(4-nitrophenacyl)glutathione as substrate preincubated for 2...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50155924(CHEMBL3780419)
Affinity DataIC50: 350nMAssay Description:Irreversible inhibition of GSTO 1-1 in LPS activated human monocytes after 30 mins by ELISA analysis in presence of ATPMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/11/2017
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526134(CHEMBL4548287)
Affinity DataIC50: 360nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526128(CHEMBL4444587)
Affinity DataIC50: 370nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50458514(CHEMBL4214871)
Affinity DataIC50: 400nMAssay Description:Inhibition of GSTO1-1 (unknown origin) by enzymatic assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526113(CHEMBL4437360)
Affinity DataIC50: 400nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetGlutathione S-transferase omega-1(Human)
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50526150(CHEMBL4464480)
Affinity DataIC50: 470nMAssay Description:Inhibition of CMFDA binding to human N-terminal 6x-His-tagged GSTO1-1 preincubated for 30 mins followed by CMFDA addition and measured after 30 mins ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
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