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Report error Found 75 for UniProtKB: P63319
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 2.70nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
LigandPNGBDBM50108296(Indolocarbazole analogue | CHEMBL289772)
Affinity DataIC50: 3nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C gamma type(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282632(Ro-32-0557 | 3-((3aR,10aR)-2-Methyl-2,3,3a,4,10,10...)
Affinity DataIC50: 5.40nMAssay Description:Inhibition of Protein kinase C gamma (PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 9nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM3033(Indolocarbazole deriv. | 3-{23-methyl-14-oxo-3,13,...)
Affinity DataIC50: 20nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280871(12-(3-azidopropyl)-13-methyl-6,7,12,13-tetrahydro-...)
Affinity DataIC50: 25nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280873(2-(13-ethyl-5-oxo-6,7,12,13-tetrahydro-5H-indolo[2...)
Affinity DataIC50: 27nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280870(12-(2,2-difluoroethyl)-13-methyl-6,7,12,13-tetrahy...)
Affinity DataIC50: 32nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProtein kinase C gamma type(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282633((S)-3-(8-((dimethylamino)methyl)-6,7,8,9-tetrahydr...)
Affinity DataIC50: 36.5nMAssay Description:Inhibition of Protein kinase C gamma (PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

LigandPNGBDBM50280877(2-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 75nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280868(12-(2,3-dihydroxypropyl)-6,7,12,13-tetrahydro-5H-i...)
Affinity DataIC50: 99nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280869(13-methyl-12-propyl-6,7,12,13-tetrahydro-5H-indolo...)
Affinity DataIC50: 100nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280875(3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 110nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM2579(CHEMBL388978 | Staurosporine, 8 | Staurosporin, 4 ...)
Affinity DataIC50: 190nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50280879(12,13-diethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a...)
Affinity DataIC50: 200nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50128280(3-[1-(1-Ethyl-piperidin-4-yl)-1H-indol-3-yl]-4-(1-...)
Affinity DataIC50: 200nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50128282(3-(1H-Indol-3-yl)-4-[1-(1-methyl-piperidin-4-yl)-1...)
Affinity DataIC50: 200nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50128287(3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-methyl-piperidi...)
Affinity DataIC50: 200nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50108291(Indolocarbazole analogue | CHEMBL36891)
Affinity DataIC50: 222nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50128286(3-[1-(1-Isopropyl-piperidin-4-yl)-1H-indol-3-yl]-4...)
Affinity DataIC50: 250nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50128290(3-[1-(1-Cyclopropylmethyl-piperidin-4-yl)-1H-indol...)
Affinity DataIC50: 300nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50128281(18-dimethylaminomethyl-(18S)-17-oxa-4,14,21-triaza...)
Affinity DataIC50: 320nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50108299(Indolocarbazole analogue | CHEMBL288229)
Affinity DataIC50: 400nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50128288(3-(1-methyl-1H-indol-3-yl)-4-(1-(piperidin-4-yl)-1...)
Affinity DataIC50: 400nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50108295(Indolocarbazole analogue | CHEMBL288817)
Affinity DataIC50: 450nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50280878(12,13-dimethyl-6,7,12,13-tetrahydro-5H-indolo[2,3-...)
Affinity DataIC50: 450nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280876(12-methyl-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyr...)
Affinity DataIC50: 520nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50052039(18-hydroxymethyl-(18S)-17-oxa-4,14,21-triazahexacy...)
Affinity DataIC50: 550nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50280874(3-(5-oxo-6,7,12,13-tetrahydro-5H-indolo[2,3-a]pyrr...)
Affinity DataIC50: 590nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM2581(CHEMBL16958 | 3,13,23-triazahexacyclo[14.7.0.0^{2,...)
Affinity DataIC50: 680nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50128285(3-(1-Methyl-1H-indol-3-yl)-4-[1-(1-pyridin-2-ylmet...)
Affinity DataIC50: 700nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50108297(Indolocarbazole analogue | CHEMBL288816)
Affinity DataIC50: 980nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C gamma type(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50213062(CHEMBL342866)
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to rat brain protein kinase C gamma regulatory domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50108300(Indolocarbazole analogue | CHEMBL38338)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50108293(Indolocarbazole analogue | CHEMBL277817)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C gamma type(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50057511(CHEMBL27266 | 13-Hydroxymethyl-10-isopropyl-9-meth...)
Affinity DataIC50: 2.75E+3nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to rat brain protein kinase C gamma regulatory domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50128283(3-[1-(1-Benzyl-pyrrolidin-3-yl)-1H-indol-3-yl]-4-(...)
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50212623(CHEMBL299248)
Affinity DataIC50: 3.50E+3nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50128284(3-[1-(1-Benzyl-piperidin-4-yl)-1H-indol-3-yl]-4-(1...)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of purified rat brain protein kinase C (RB-PKC)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50285193(17-hydroxymethyl-18-oxa-4,14,22-triazahexacyclo[20...)
Affinity DataIC50: 6.40E+3nMAssay Description:Inhibition of rat brain PKCMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

LigandPNGBDBM50108298(Indolocarbazole analogue | CHEMBL29709)
Affinity DataIC50: 7.60E+3nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50212624(CHEMBL294684)
Affinity DataIC50: 8.10E+3nMAssay Description:In vitro for inhibitory activity against protein kinase C from rat brainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50136008(12-(3-hydroxypropyl)-9-isopropoxymethyl-6,7,12,13-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat brain Protein kinase CMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C gamma type(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50213063(CHEMBL342131)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to rat brain protein kinase C gamma regulatory domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50108294(Indolocarbazole analogue | CHEMBL288818)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50108292(Indolocarbazole analogue | CHEMBL37529)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM24942(methyl (15S,16R,18R)-10,23-bis[(ethylsulfanyl)meth...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of protein kinase C (PKC) from rat brain homogenateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50009723(CHEMBL329705 | 2,6-Diamino-hexanoic acid (1-tridec...)
Affinity DataIC50: 2.00E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetProtein kinase C alpha/beta/gamma type(Rat)
Nova Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50229926(CHEMBL319584)
Affinity DataIC50: 2.30E+4nMAssay Description:In vitro inhibition of [32P] incorporation into histones by rat brain partially purified Protein kinase C in the presence of PMA, [Ca2+] and phosphat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/22/2012
Entry Details Article
PubMed
TargetProtein kinase C gamma type(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50213064(CHEMBL342147)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of [3H]phorbol-12,13-dibutyrate (PDBu) binding to rat brain protein kinase C gamma regulatory domainMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

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