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TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176672(US9115122, 76)
Affinity DataKd:  5.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176673(US9115122, 76.2)
Affinity DataKd:  3.30E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176674(US9115122, 76.3)
Affinity DataKd:  1.50E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176675(US9115122, 76.4)
Affinity DataKd:  2.40E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [T157A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176672(US9115122, 76)
Affinity DataKd:  6.10E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [T157A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176673(US9115122, 76.2)
Affinity DataKd:  2.40E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [T157A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176674(US9115122, 76.3)
Affinity DataKd:  8.10E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [T157A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176675(US9115122, 76.4)
Affinity DataKd:  3.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176672(US9115122, 76)
Affinity DataKd:  7.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176673(US9115122, 76.2)
Affinity DataKd:  1.90E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176674(US9115122, 76.3)
Affinity DataKd:  1.34E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176675(US9115122, 76.4)
Affinity DataKd:  1.80E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [T157A,D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176672(US9115122, 76)
Affinity DataKd:  6.40E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [T157A,D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176673(US9115122, 76.2)
Affinity DataKd:  4.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [T157A,D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176674(US9115122, 76.3)
Affinity DataKd: >2.00E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [T157A,D319N](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176675(US9115122, 76.4)
Affinity DataKd: >2.00E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  130nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [L114A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  27nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [Y191A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  130nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [R275A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  240nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [L265A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  280nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [L232A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  130nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [L235A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  90nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [L198A,L232A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd:  140nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1 [L198A,L235A](Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176676(US9115122, 2.3.2)
Affinity DataKd: >2.00E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176677(US9115122, SF-2-062)
Affinity DataKd:  1.30E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176678(US9115122, SF-2-054)
Affinity DataKd:  170nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176679(US9115122, SS-1-019)
Affinity DataKd:  9.30E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176677(US9115122, SF-2-062)
Affinity DataKd:  6.00E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176678(US9115122, SF-2-054)
Affinity DataKd:  1.02E+4nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176677(US9115122, SF-2-062)
Affinity DataKd:  3.70E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176678(US9115122, SF-2-054)
Affinity DataKd:  400nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176677(US9115122, SF-2-062)
Affinity DataKd:  6.80E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM176678(US9115122, SF-2-054)
Affinity DataKd:  1.40E+3nMAssay Description:CADD and biological testing to identify compounds that interact with novel ERK substrate docking sites. The known ERK2 docking sites include the DRS ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203308(US9242981, 37)
Affinity DataKd:  6nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203317(US9242981, 46)
Affinity DataKd:  0.700nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203319(US9242981, 48)
Affinity DataKd:  0.370nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203321(US9242981, 53)
Affinity DataKd:  0.150nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203322(US9242981, 54)
Affinity DataKd:  0.510nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203325(US9242981, 57)
Affinity DataKd:  0.300nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203326(US9242981, 58)
Affinity DataKd:  0.25nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203327(US9242981, 59)
Affinity DataKd:  1.51nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203328(US9242981, 60)
Affinity DataKd:  1.12nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203329(US9242981, 61)
Affinity DataKd:  0.470nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203330(US9242981, 62)
Affinity DataKd:  2.10nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203337(US9242981, 69)
Affinity DataKd:  0.310nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203339(US9242981, 71)
Affinity DataKd:  0.150nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203343(US9242981, 75)
Affinity DataKd:  1.36nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203344(US9242981, 76)
Affinity DataKd:  1.55nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

TargetMitogen-activated protein kinase 1(Mouse)
University of Maryland, Baltimore

US Patent
LigandPNGBDBM203349(US9242981, 84)
Affinity DataKd:  0.130nMT: 2°CAssay Description:The SAR (Structure Activity Relationship) for ERK ligands covered by this invention was interrogated using the TdF (Temperature Dependence Fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/28/2016
Entry Details
Go to US Patent

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