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Report error Found 10 of affinity data for UniProtKB/TrEMBL: P53790
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426887(CHEMBL2323695)
Affinity DataIC50: 22nMAssay Description:Inhibition of rat SGLT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50394534(CHEMBL2159102)
Affinity DataIC50: 67nMAssay Description:Inhibition of rat SGLT1 expressed in COS7 cells assessed as reduction of [14C]-AMG uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50467750(CHEMBL4279519)
Affinity DataIC50: 68nMAssay Description:Inhibition of rat SGLT1 expressed in CHOK1 cells assessed as reduction in Na-dependent [14C]-AMG uptake preincubated for 10 mins followed by [14C]-AM...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50426888(CHEMBL2323694)
Affinity DataIC50: 104nMAssay Description:Inhibition of rat SGLT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50394533(CHEMBL2159101)
Affinity DataIC50: 183nMAssay Description:Inhibition of rat SGLT1 expressed in COS7 cells assessed as reduction of [14C]-AMG uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50394533(CHEMBL2159101)
Affinity DataIC50: 183nMAssay Description:Inhibition of rat SGLT1More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50394532(CHEMBL2159094)
Affinity DataIC50: 227nMAssay Description:Inhibition of rat SGLT1 expressed in COS7 cells assessed as reduction of [14C]-AMG uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50394531(CHEMBL2159091)
Affinity DataIC50: 308nMAssay Description:Inhibition of rat SGLT1 expressed in COS7 cells assessed as reduction of [14C]-AMG uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM20875(CHEMBL245067 | JMC511145 Compound 1 | 1-(2,4-dihyd...)
Affinity DataIC50: 350nMAssay Description:Inhibition of rat SGLT1 expressed in COS7 cells assessed as reduction of [14C]-AMG uptakeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
TargetSodium/glucose cotransporter 1(Rat)
Kissei Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50340014(4-((5-(4-chlorobenzylthio)-4-methyl-4H-1,2,4-triaz...)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of rat SGLT1 expressed in CHO cells assessed as inhibition of [14C]-alpha-methyl-D-glucopyranoside transport after 60 mins by scintillatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2011
Entry Details Article
PubMed