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Report error Found 74 of affinity data for UniProtKB/TrEMBL: P52500
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112639(pQ-Q-R-Y-G-N-Q-W-A-V-G-H-L-M-NH2 | CHEMBL402688)
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112626(Carbocyanine derivative | CHEMBL442514)
Affinity DataIC50: 1.80nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112623((FITC-Q-W-A-V-G-H-L-M-NH2) | CHEMBL274327)
Affinity DataIC50: 3.20nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112643((DTPA-P-Q-R-Y-G-N-Q-W-A-V-G-H-L-M-NH2) | CHEMBL442...)
Affinity DataIC50: 4.70nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112611((K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL405669)
Affinity DataIC50: 4.80nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112640((epsilon-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL21696...)
Affinity DataIC50: 4.80nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112629((epsilon-FITC-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL38528...)
Affinity DataIC50: 5.70nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112632((alpha-FITC-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL428280)
Affinity DataIC50: 5.80nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112619((G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL408739)
Affinity DataIC50: 7.60nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112633((FITC-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL385928)
Affinity DataIC50: 9.20nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112635((alpha,epsilon-(-FITC)2-K-Q-W-A-V-G-H-L-M-NH2) | C...)
Affinity DataIC50: 9.5nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112620((epsilon-FITC-K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMB...)
Affinity DataIC50: 9.60nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112625((K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL269310)
Affinity DataIC50: 10.5nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112627((alpha-FITC-epsilon-DOTA-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50: 15nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112646((alpha-FITC-K-G-S-G-Q-W-A-V-G-H-L-M-NH2) | CHEMBL4...)
Affinity DataIC50: 15.6nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112614((alpha-FITC-epsilon-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50: 20nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112616((alpha,epsilon-(FITC)2-K-G-S-G-Q-W-A-V-G-H-L-M-NH2...)
Affinity DataIC50: 20.5nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112642((Q-W-A-V-G-H-L-M-NH2) | CHEMBL300318)
Affinity DataIC50: 28.3nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112630((alpha,epsilon-(DTPA)2-K-Q-W-A-V-G-H-L-M-NH2) | CH...)
Affinity DataIC50: 240nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112621((alpha-DTPA-epsilon-FITC-K-Q-W-A-V-G-H-L-M-NH2) | ...)
Affinity DataIC50: 276nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50112622((alpha-DTPA-K-Q-W-A-V-G-H-L-M-NH2) | CHEMBL440609)
Affinity DataIC50: 410nMAssay Description:In vitro binding affinity of [111In]DTPA-[Y4]-bombesin to bombesin receptor in the rat pancreatic acinar cell line, AR42JMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50280412(CP-70030 | 2-{3-[1-(3,5-Di-tert-butyl-4-hydroxy-ph...)
Affinity DataIC50: 1.50E+3nMAssay Description:Compound was evaluated for displacement of radiolabeled [I-125]GRP from rat brain receptor; 1.5-3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

LigandPNGBDBM50280413(CP-75998 | 5'-bromo-1'-(3,4-dichlorobenzyl)spiro[t...)
Affinity DataIC50: 1.50E+3nMAssay Description:Compound was evaluated for displacement of radiolabeled [I-125]GRP from rat brain receptor; 1.5-3 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50005601(CHEMBL2369819)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50408923(CHEMBL2114155)
Affinity DataKi: >0nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85480(CAS_l | (3-Ph-Pr6)His7,DAla11,DPro13,Psi13-14,Phe1...)
Affinity DataKi:  0.740nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85500(Bombesin,Phe13)
Affinity DataKi:  0.770nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85488(DPhe6,BetaAla11,Phe13,Nle14-Bn(6-14))
Affinity DataKi:  0.990nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50089280(JMV 1535 | CHEMBL437655)
Affinity DataKi:  1.70nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50089284(JMV 1803 | CHEMBL265856)
Affinity DataKi:  1.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85499(CAS_29451-71-6 | NSC_5489061 | Ranatensin)
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85486(DPhe6-Bn[6-14))
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85502(PG-L)
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50089285(JMV 1799 | CHEMBL415110)
Affinity DataKi:  3.10nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50089282((D)Phe-Gln-Trp-Ala-Val-Gly-His-Leu-Leu-NH2 | CHEMB...)
Affinity DataKi:  3.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50089281(JMV 1802 | CHEMBL386480)
Affinity DataKi:  3.80nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85484(Bombesin)
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50089291(JMV 1813 | CHEMBL415021)
Affinity DataKi:  5.20nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85498(CAS_5486808 | NSC_5486808 | Litorin)
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85493(DTyr6,DAla11-Bn(6-13)butylamide)
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85495(DPhe6-Bn(6-13)propylamide)
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50089278(JMV 1801 | CHEMBL411016)
Affinity DataKi:  9nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85496(DPhe6-Bn(6-13)methylester)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM50089279(JMV 1719 | CHEMBL406013)
Affinity DataKi:  13nMAssay Description:In vitro binding affinity against bombesin / GRP receptors on rat pancreatic acini.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85481(CAS_93755-85-2 | GRP)
Affinity DataKi:  18nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM81964(NSC_5486814 | CAS_5486814 | Neuromedin C | Gastrin)
Affinity DataKi:  20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85494(DPhe6-Bn(6-13)NH2)
Affinity DataKi:  27nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85506(CAS_125988 | NSC_125988 | Rhodei-Litorin)
Affinity DataKi:  31nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85490(DPhe6,Leu13,Psi(CH2NH),Cpa14-Bn(6-14))
Affinity DataKi:  42nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
TargetGastrin-releasing peptide receptor(Rat)
Washington University

Curated by ChEMBL
LigandPNGBDBM85497(CAS_31078-12-3 | Alytesin)
Affinity DataKi:  62nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/12/2012
Entry Details Article
PubMed
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