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Report error Found 59 for UniProtKB: P51050
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM29611(CHEMBL289233 | Melatonin,2-Iodo | 2-Iodomelatonin)
Affinity DataKi:  0.130nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231291(CHEMBL421013)
Affinity DataKi:  0.230nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231307(CHEMBL34622)
Affinity DataKi:  0.270nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50043289(CHEMBL34730 | N-[2-(6-Chloro-5-methoxy-1H-indol-3-...)
Affinity DataKi:  0.340nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072660(N-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmet...)
Affinity DataKi:  0.450nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072651(N-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmet...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072651(N-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmet...)
Affinity DataKi:  0.530nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85239(5-MeOT-N-propionyl)
Affinity DataKi:  0.540nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50037220(1-[2-(7-Methoxy-naphthalen-1-yl)-ethyl]-pyrrolidin...)
Affinity DataKi:  0.540nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85239(5-MeOT-N-propionyl)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  0.700nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231304(CHEMBL288084)
Affinity DataKi:  0.730nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072656(N-(3-Methoxy-6,7,8,9-tetrahydro-5H-benzocyclohepte...)
Affinity DataKi:  1nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  1.20nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM9019(CHEMBL45 | N-[2-(5-methoxy-1H-indol-3-yl)ethyl]ace...)
Affinity DataKi:  1.21nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072652(N-(6-Methoxy-indan-1-ylmethyl)-propionamide | CHEM...)
Affinity DataKi:  3nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072652(N-(6-Methoxy-indan-1-ylmethyl)-propionamide | CHEM...)
Affinity DataKi:  3nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231302(CHEMBL99376)
Affinity DataKi:  3.60nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231292(CHEMBL95920)
Affinity DataKi:  3.80nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072654(N-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmet...)
Affinity DataKi:  4nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50045843(CHEMBL99377 | 8-M-PDOT | N-(8-Methoxy-1,2,3,4-tetr...)
Affinity DataKi:  7.40nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072653(N-(6-Methoxy-indan-1-ylmethyl)-butyramide | CHEMBL...)
Affinity DataKi:  7.60nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072652(N-(6-Methoxy-indan-1-ylmethyl)-propionamide | CHEM...)
Affinity DataKi:  16nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85240(5-MeOT-N-pentanyl)
Affinity DataKi:  24.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85240(5-MeOT-N-pentanyl)
Affinity DataKi:  24.5nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072661(N-(3-Methoxy-6,7,8,9-tetrahydro-5H-benzocyclohepte...)
Affinity DataKi:  29nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072657(N-(3-Methoxy-6,7,8,9-tetrahydro-5H-benzocyclohepte...)
Affinity DataKi:  34nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072658(N-(4-Methoxy-bicyclo[4.2.0]octa-1,3,5-trien-7-ylme...)
Affinity DataKi:  40nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231298(CHEMBL330385)
Affinity DataKi:  44nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50035176(CHEMBL53015 | 8-M-ADOT | N-(8-Methoxy-1,2,3,4-tetr...)
Affinity DataKi:  46nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072655(N-(4-Methoxy-bicyclo[4.2.0]octa-1,3,5-trien-7-ylme...)
Affinity DataKi:  49nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072659(N-(6-Methoxy-indan-1-ylmethyl)-acetamide | CHEMBL1...)
Affinity DataKi:  77nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231294(CHEMBL95266)
Affinity DataKi:  95nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231296(CHEMBL316854)
Affinity DataKi:  121nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231303(CHEMBL95364)
Affinity DataKi:  141nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231301(CHEMBL421569)
Affinity DataKi:  145nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50282747(CHEMBL290406 | AANAT Inhibitor, 1 | 2-Bromo-N-[2-(...)
Affinity DataKi:  153nMAssay Description:Binding affinity towards melatonin receptor using 2-[125I]iodomelatonin as radioligand in chick brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/21/2018
Entry Details

TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50035176(CHEMBL53015 | 8-M-ADOT | N-(8-Methoxy-1,2,3,4-tetr...)
Affinity DataKi:  161nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072650(N-(4-Methoxy-bicyclo[4.2.0]octa-1,3,5-trien-7-ylme...)
Affinity DataKi:  224nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231299(CHEMBL95851)
Affinity DataKi:  312nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231305(CHEMBL52801)
Affinity DataKi:  420nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231306(CHEMBL53722)
Affinity DataKi:  581nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231295(CHEMBL322193)
Affinity DataKi:  665nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231308(CHEMBL299966)
Affinity DataKi:  748nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85237(5-MeOT-N-hexanyl)
Affinity DataKi:  773nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85383(Luzindole,5-MeOT-N-hexanyl)
Affinity DataKi:  776nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1A/1B/1C(Chicken)
University of Groningen

Curated by ChEMBL
LigandPNGBDBM50231300(CHEMBL50943)
Affinity DataKi:  789nMAssay Description:Binding affinity to compete for 2-[125I]iodomelatonin binding to chicken retinal membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/7/2019
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM85384(Luzindole,N-pentanoyl)
Affinity DataKi:  933nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2012
Entry Details Article
PubMed
TargetMelatonin receptor type 1B(Chicken)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50072651(N-(7-Methoxy-1,2,3,4-tetrahydro-naphthalen-1-ylmet...)
Affinity DataKi: >1.00E+3nMAssay Description:Binding affinity measured against Chicken brain melatonin receptor by using 2-[125I]iodomelatonin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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