Affinity DataKd: 500nMAssay Description:Binding affinity to human SULT1A1 expressed in Escherichia coli assessed as change in intrinsic fluorescenceMore data for this Ligand-Target Pair
Affinity DataKd: 2.30E+3nMAssay Description:Binding affinity to human SULT1A1 expressed in Escherichia coli assessed as change in intrinsic fluorescenceMore data for this Ligand-Target Pair
Affinity DataKd: 4.30nMAssay Description:Binding affinity to human SULT1A1 expressed in Escherichia coli assessed as change in intrinsic fluorescence in presence of 3',5'-phosphoadenosineMore data for this Ligand-Target Pair
Affinity DataKd: 1.20E+3nMAssay Description:Binding affinity to human SULT1A1 expressed in Escherichia coli assessed as change in intrinsic fluorescence in presence of 3',5'-phosphoadenosineMore data for this Ligand-Target Pair
Affinity DataIC50: 20nMAssay Description:Inhibition of SULT1A1 in human MCF7 cells assessed as 17beta-estradiol sulfationMore data for this Ligand-Target Pair
Affinity DataKi: 8.90nMAssay Description:Inhibition of human SULT1A1 expressed in Escherichia coli assessed as p-nitrophenol sulfation at 100 nM by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 15nMAssay Description:Inhibition of human SULT1A1 expressed in Escherichia coli assessed as 17beta-estradiol sulfation at 100 nM by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Inhibition of human SULT1A1 expressed in Escherichia coli assessed as beta-naphthol sulfation at 100 nM by Michaelis-Menten equation analysisMore data for this Ligand-Target Pair
Affinity DataKi: 3.50E+4nM ΔG°: -23.5kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
Affinity DataKi: 5.50E+4nM ΔG°: -22.4kJ/molepH: 7.5 T: 2°CAssay Description:Reaction conditions were as follows: SULT1A1 or 2A1 (50 nM), PnP (3.0 or 100 uM, respectively; 2 x Km PnP), amoxipine or protriptyline (0, 50, 100, o...More data for this Ligand-Target Pair
