Compile Data Set for Download or QSAR
Report error Found 105 of affinity data for UniProtKB/TrEMBL: P50129
LigandPNGBDBM30704(METERGOLINE | (phenylmethyl) N-[[(6aR,9S,10aR)-4,7...)
Affinity DataKi:  0.370nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM84933(LY-193525 | 6-Methyl-N-cyclohexylergoline-8-beta-c...)
Affinity DataKi:  3.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM81446(CAS_60-79-7 | NSC_104873 | ERGONOVINE)
Affinity DataKi:  3.80nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM84935(LY86057 | LY 86057)
Affinity DataKi:  4.60nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM50328443(1-(4-Fluorophenyl)-4-[4-([2.2]paracyclophan-4-yl)-...)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM21398(4-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-1...)
Affinity DataKi:  30nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM82516(NSC_60740 | CAS_121588-75-8 | AMESERGIDE)
Affinity DataKi:  30.7nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM84930(CAS_60634-51-7 | NSC_107989 | LY 53857)
Affinity DataKi:  40nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM50024204(MESULERGINE | CHEMBL12314 | 4,7-dimethyl-(6aR,9S,1...)
Affinity DataKi:  54.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM84939(1,6-Dimethylergoline-8 -carboxylic acid 2-hydroxy-...)
Affinity DataKi:  57.2nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM50401953(CHEMBL2207643)
Affinity DataKi:  92nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50373711(CHEMBL256637)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]ketanserin from pig cortical membrane 5HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50328444(4-[4-(2,5-Dimethylphenyl)-4-hydroxypiperidin-1-yl]...)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM84938(LY-197541 | (6aR)-7-Methyl-4-isobutyl-4,6,6a ,7,8,...)
Affinity DataKi:  148nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM50342706(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50328452(4-[4-(4-Chlorophenyl)piperazin-1-yl]-1-(2,5-dimeth...)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM50342704(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  190nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50331549([11C]-3-(2-oxo-3-(2-(4-(trifluoromethyl)piperidin-...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50342714(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  230nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50373714(CHEMBL270406)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]ketanserin from pig cortical membrane 5HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50328453(4-[4-([2.2]Paracyclophan-4-yl)piperazin-1-yl]-1-([...)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM50132069(3-(4-Fluoro-phenyl)-N-{4-[4-(2-methoxy-phenyl)-pip...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/14/2011
Entry Details Article
PubMed
LigandPNGBDBM50342713(3,4-Dihydro-2-[4-(4-(2-methoxyphenyl)piperazin-1-y...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50342715(3,4-Dihydro-6-(2-furyl)-2-[4-(4-(2-methoxyphenyl)p...)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50119386(Benzo[b]thiophene-2-carboxylic acid {4-[4-(2-metho...)
Affinity DataKi:  350nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM50115717(1-(4-Ethynyl-1H-pyrrol-2-ylmethyl)-4-phenyl-pipera...)
Affinity DataKi:  380nMAssay Description:Ability to displace [3H]-Ketanserin radioligand from porcine 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
LigandPNGBDBM50073805(FAUC 113 | 3-[4-(4-Chloro-phenyl)-piperazin-1-ylme...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in porcine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
LigandPNGBDBM50073805(FAUC 113 | 3-[4-(4-Chloro-phenyl)-piperazin-1-ylme...)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50401954(CHEMBL2207636)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50342707(2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-1-o...)
Affinity DataKi:  430nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50155520(CHEMBL558392 | CHEMBL476935 | 4-[4-(4-Chloro-pheny...)
Affinity DataKi:  440nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM50328449(4-[4-([2.2]Paracyclophan-4-yl)piperazin-1-yl]-1-(4...)
Affinity DataKi:  450nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM50342705(2-[4-(4-(2-Methoxyphenyl)piperazin-1-yl)butyl]-2,3...)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50401944(CHEMBL2207641)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
LigandPNGBDBM50115715(5-(4-Phenyl-piperazin-1-ylmethyl)-1H-pyrrole-3-car...)
Affinity DataKi:  610nMAssay Description:Ability to displace [3H]-Ketanserin radioligand from porcine 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
LigandPNGBDBM50328447(4-[4-(4-Chlorophenyl)-4-hydroxypiperidin-1-yl]-1-(...)
Affinity DataKi:  690nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM50342711(7-methoxy-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)...)
Affinity DataKi:  810nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50342712(6-fluoro-2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)b...)
Affinity DataKi:  840nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50403915(CHEMBL2113718)
Affinity DataKi:  850nMAssay Description:Ability to displace [3H]-Ketanserin radioligand from porcine 5-hydroxytryptamine 2A receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
LigandPNGBDBM50328450(4-[4-(2,5-Dimethylphenyl)piperazin-1-yl]-1-(4-fluo...)
Affinity DataKi:  850nMAssay Description:Displacement of [3H]Ketanserin from 5-HT2 receptor in pig cortex membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2011
Entry Details Article
PubMed
LigandPNGBDBM50373713(CHEMBL404888)
Affinity DataKi:  850nMAssay Description:Displacement of [3H]ketanserin from pig cortical membrane 5HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50189837(2-[4-(4-fluorophenyl)piperazin-1-ylmethyl]imidazo[...)
Affinity DataKi:  860nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in porcine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
LigandPNGBDBM50102712(4-(4-Chloro-phenyl)-1-pyrazolo[1,5-a]pyridin-2-ylm...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in pig cortical membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50102712(4-(4-Chloro-phenyl)-1-pyrazolo[1,5-a]pyridin-2-ylm...)
Affinity DataKi:  900nMAssay Description:Displacement of [3H]ketanserin from pig cortical membrane 5HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50189849(6-chloro-2-[4-(4-chlorophenyl)piperazin-1-ylmethyl...)
Affinity DataKi:  910nMAssay Description:Displacement of [3H]ketanserin from 5HT2 receptor in porcine cortical membraneMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
LigandPNGBDBM50342708(3,4-Dihydro-6-ethynyl-2-[4-(4-(2-methoxyphenyl)pip...)
Affinity DataKi:  920nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM82087(tryptamine, 5-Methoxy | 5-Methoxytryptamine hydroc...)
Affinity DataKi:  923nMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2012
Entry Details
PubMed
LigandPNGBDBM50373712(CHEMBL255163)
Affinity DataKi:  980nMAssay Description:Displacement of [3H]ketanserin from pig cortical membrane 5HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2012
Entry Details Article
PubMed
LigandPNGBDBM50342709(2-(4-(4-(2-methoxyphenyl)piperazin-1-yl)butyl)-3,4...)
Affinity DataKi:  990nMAssay Description:Displacement of [3H]Ketanserin from pig 5-HT2 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/3/2011
Entry Details Article
PubMed
LigandPNGBDBM50401949(CHEMBL2207635)
Affinity DataKi:  990nMAssay Description:Displacement of [3H]ketanserin from 5-HT2 receptor in porcine cerebral cortex homogenate after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/17/2013
Entry Details Article
PubMed
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