Compile Data Set for Download or QSAR
Report error Found 149 of affinity data for UniProtKB/TrEMBL: P49881
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128299(4-Methyl-benzo[1,3]dioxole-5-carboxylic acid [1-(3...)
Affinity DataEC50:  3.68E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128300(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-3-methoxy-...)
Affinity DataEC50:  1.41E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128301(N-[1-(3,5-Dimethyl-benzoyl)-cyclobutyl]-3-methoxy-...)
Affinity DataEC50:  8.52E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128302(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-2-ethyl-3-...)
Affinity DataEC50:  1.81E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128305(N'-tert-butyl-N'-(3,5-dimethylbenzoyl)-3-methoxy-2...)
Affinity DataEC50:  100nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128306(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cycloheptyl]-2-...)
Affinity DataEC50:  1.94E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128297(5-Ethyl-2,3-dihydro-benzo[1,4]dioxine-6-carboxylic...)
Affinity DataEC50:  740nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128307(N-[4-(3,5-Dimethyl-benzoyl)-tetrahydro-pyran-4-yl]...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128298(N-[1-(3,5-Dimethyl-benzoyl)-1-ethyl-propyl]-3-meth...)
Affinity DataEC50:  4.53E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128308(N-[4-(3,5-Dimethyl-benzoyl)-1,1-dioxo-hexahydro-1l...)
Affinity DataEC50:  1.50E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128309(3,5-Dimethyl-benzoic acid N-tert-butyl-N'-(2-ethyl...)
Affinity DataEC50:  250nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128310(N-[1-(3,5-Dimethyl-benzoyl)-cyclopropyl]-3-methoxy...)
Affinity DataEC50:  2.04E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128303(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cyclopentyl]-2-...)
Affinity DataEC50:  5.16E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128312(3-Methoxy-N-[1-(2-methoxy-benzoyl)-cyclohexyl]-2-m...)
Affinity DataEC50:  980nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128304(N-[4-(3,5-Dimethyl-benzoyl)-tetrahydro-thiopyran-4...)
Affinity DataEC50:  1.60E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128313(N-[1-(3,5-Dimethyl-benzoyl)-cyclopentyl]-3-methoxy...)
Affinity DataEC50:  1.87E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50:  1.51E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128311(N-[2-(3,5-Dimethyl-phenyl)-1,1-dimethyl-2-oxo-ethy...)
Affinity DataEC50:  1.00E+4nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128315(N-[1-(3,5-Dimethyl-benzoyl)-cycloheptyl]-3-methoxy...)
Affinity DataEC50:  1.61E+3nMAssay Description:Dose affording 50% of maximum transactivation for ecdysone receptor from Bombyx mori (BmEcR) and a beta-galactosidase reporter gene in HEK293 cell-li...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488441(CHEMBL2286428)
Affinity DataEC50:  6.60nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488442(CHEMBL2286438)
Affinity DataEC50:  115nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488443(CHEMBL2286420)
Affinity DataEC50:  871nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488445(CHEMBL2286440)
Affinity DataEC50:  1.23E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50178988(CHEBI:38452 | Tebufenozide)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488447(CHEMBL2286412)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488444(CHEMBL2286409)
Affinity DataEC50:  191nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488468(CHEMBL2286448)
Affinity DataEC50:  4.40nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488449(CHEMBL2286446)
Affinity DataEC50:  427nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488469(CHEMBL2286410)
Affinity DataEC50:  1.26E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488453(CHEMBL2286439)
Affinity DataEC50:  1.15E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50178990(CHEMBL2286425)
Affinity DataEC50:  309nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488470(CHEMBL2286444)
Affinity DataEC50:  33nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488451(CHEMBL2286443)
Affinity DataEC50:  447nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488452(CHEMBL2286442)
Affinity DataEC50:  1.78E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488471(CHEMBL2286437)
Affinity DataEC50:  1.18E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488454(CHEMBL2286436)
Affinity DataEC50:  2.88E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488472(CHEMBL2286435)
Affinity DataEC50:  7.76E+3nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488440(CHEMBL2228849)
Affinity DataEC50:  11nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488457(CHEMBL2286430)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488458(CHEMBL2286427)
Affinity DataEC50:  31nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488473(CHEMBL2286426)
Affinity DataEC50:  151nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488474(CHEMBL2286423)
Affinity DataEC50:  129nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488475(CHEMBL2286422)
Affinity DataEC50:  145nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50178982(CHEMBL2228438)
Affinity DataEC50:  200nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488460(CHEBI:38450 | Chromafenozide)
Affinity DataEC50:  1nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488461(CHEBI:38451 | Halofenozide)
Affinity DataEC50:  78nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50128314(N-[1-(3,5-Dimethyl-benzoyl)-cyclohexyl]-4-ethyl-be...)
Affinity DataEC50:  78nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488450(CHEMBL2286445)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488439(CHEMBL2286441)
Affinity DataEC50:  302nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetEcdysone receptor(Silk moth)
Rheogene

Curated by ChEMBL
LigandPNGBDBM50488455(CHEMBL2286434)
Affinity DataEC50:  1.91E+4nMAssay Description:Agonist activity at ecdysone receptor in Bombyx mori Bm5 cells after 24 hr by luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
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