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Report error Found 13 of affinity data for UniProtKB/TrEMBL: P49407
TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM86253(CAS_100929-53-1 | NSC_104742 | DAMGO | US10836728,...)
Affinity DataEC50:  60nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
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TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM224017((+)-Morphine | US10752592, Compound morphine | US1...)
Affinity DataEC50:  310nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472704(3-(1-(2-Chloro-4-fluorobenzyl)-3-((dimethylamino)m...)
Affinity DataEC50:  2.56E+3nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472714(US10836728, Compound Ent-A-syn-(6))
Affinity DataEC50:  3.17E+3nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472715(US10836728, Compound Ent-B-syn-(6))
Affinity DataEC50:  3.67E+3nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472721(3-(3-((Dimethylamino)methyl)-4-hydroxy-1-phenethyl...)
Affinity DataEC50:  830nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472831(US10836728, Compound (11))
Affinity DataEC50:  1.07E+4nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472832(US10836728, Compound (15))
Affinity DataEC50: >1.00E+5nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472834(US10836728, Compound (17))
Affinity DataEC50: >1.00E+5nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472835(3-(3-((Dimethylamino)methyl)-4-hydroxy-1-(4-hydrox...)
Affinity DataEC50:  3.10E+3nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM472836(3-[3-Dimethylaminomethyl-4-hydroxy-1-(3-phenyl-pro...)
Affinity DataEC50:  270nMAssay Description:The DISCOVERX PATHHUNTER β-Arrestin assay is used to measure β-arrestin-2 activity. The technology is based on Enzyme Fragment Complementat...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/30/2021
Entry Details
Go to US Patent

TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM50652793(CHEMBL5653589)
Affinity DataKd:  45nMMore data for this Ligand-Target Pair
Ligand Info
In Depth
Date in BDB:
10/13/2025
Entry Details
PubMed
TargetBeta-arrestin-1(Human)
Mebias Discovery

US Patent
LigandPNGBDBM34233(EBSELEN | 2-Phenyl-benzo[d]isoselenazol-3-one(Ebse...)
Affinity DataIC50: 1.52E+3nMAssay Description:University of New Mexico Assay Overview: Assay Support: 1 R03 DA031665-01A1 Project Title: MLP Assay for Arrestin-AP2 Inhibitors Assay Provider: Er...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/6/2012
Entry Details
PCBioAssay