Affinity DataEC50: 1nMAssay Description:Antagonist activity at CRF-R2 beta in rat A7r5 cells assessed as inhibition of rat Ucn1 induced cAMP accumulation after 30 mins by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.630nMAssay Description:Antagonist activity at CRF-R2 beta in rat A7r5 cells assessed as inhibition of rat Ucn1 induced cAMP accumulation after 30 mins by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.910nMAssay Description:Antagonist activity at CRF-R2 beta in rat A7r5 cells assessed as inhibition of rat Ucn1 induced cAMP accumulation after 30 mins by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataEC50: 0.770nMAssay Description:Antagonist activity at CRF-R2 beta in rat A7r5 cells assessed as inhibition of rat Ucn1 induced cAMP accumulation after 30 mins by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Antagonist activity at CRF-R2 beta in rat A7r5 cells assessed as inhibition of rat Ucn1 induced cAMP accumulation after 30 mins by radioimmunoassayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.570nMAssay Description:Compound was evaluated for affinity towards Corticotropin releasing factor receptor 2 expressing tissues such as Choroid plexus, blood vesselsMore data for this Ligand-Target Pair
Affinity DataIC50: 2.10nMAssay Description:Compound was evaluated for affinity towards Corticotropin releasing factor receptor 2 expressing tissues such as Choroid plexus, blood vesselsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:Binding affinity at Corticotropin releasing factor receptor of rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 0.5nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity at Corticotropin releasing factor receptor of rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity at Corticotropin releasing factor receptor of rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:Binding affinity at Corticotropin releasing factor receptor of rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:Binding affinity at Corticotropin releasing factor receptor of rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity at Corticotropin releasing factor receptor of rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Binding affinity at Corticotropin releasing factor receptor of rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Binding affinity at Corticotropin releasing factor receptor of rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 3.30nMAssay Description:Binding affinity at Corticotropin releasing factor receptor of rat cortical homogenates.More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 4.40nMAssay Description:In vitro binding affinity against Corticotropin releasing factor receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:In vitro binding affinity to the CRF receptor in rat cortical homogenatesMore data for this Ligand-Target Pair
