Compile Data Set for Download or QSAR
Report error Found 102 of affinity data for UniProtKB/TrEMBL: P42568
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459744(CHEMBL4204744)
Affinity DataKd:  15nMAssay Description:Binding affinity to MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) by Bio-layer interferometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50576674(CHEMBL4850575)
Affinity DataKd:  370nMAssay Description:Binding affinity to AF9 YEATS domain (1 to 138 residues) (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50576675(CHEMBL4848627)
Affinity DataKd:  800nMAssay Description:Binding affinity to AF9 YEATS domain (1 to 138 residues) (unknown origin) by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625619(CHEMBL4752253)
Affinity DataKd:  110nMAssay Description:Binding affinity to MLLT3 YD domain (unknown origin) assessed as dissociation constant by biolayer interferometry assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625619(CHEMBL4752253)
Affinity DataKd:  76nMAssay Description:Binding affinity to MLLT3 YD domain (unknown origin) assessed as dissociation constant by isothermal calorimetry assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633970(CHEMBL5430585)
Affinity DataKd:  7.80E+3nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human AF9 YEATS domain (1 to 138 residues) expressed in Escherichia coli 2(DE3)pLysS cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633971(CHEMBL5409871)
Affinity DataKd:  1.37E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human AF9 YEATS domain (1 to 138 residues) expressed in Escherichia coli 2(DE3)pLysS cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633972(CHEMBL5409621)
Affinity DataKd:  1.36E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human AF9 YEATS domain (1 to 138 residues) expressed in Escherichia coli 2(DE3)pLysS cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633973(CHEMBL5434543)
Affinity DataKd:  5.10E+3nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human AF9 YEATS domain (1 to 138 residues) expressed in Escherichia coli 2(DE3)pLysS cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633974(CHEMBL5399658)
Affinity DataKd:  4.65E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human AF9 YEATS domain (1 to 138 residues) expressed in Escherichia coli 2(DE3)pLysS cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633975(CHEMBL5398587)
Affinity DataKd:  1.59E+5nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human AF9 YEATS domain (1 to 138 residues) expressed in Escherichia coli 2(DE3)pLysS cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633976(CHEMBL5415562)
Affinity DataKd:  2.05E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human AF9 YEATS domain (1 to 138 residues) expressed in Escherichia coli 2(DE3)pLysS cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50633977(CHEMBL5398289)
Affinity DataKd:  4.85E+4nMAssay Description:Binding affinity to N-terminal His-tagged recombinant human AF9 YEATS domain (1 to 138 residues) expressed in Escherichia coli 2(DE3)pLysS cells asse...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459727(CHEMBL4206834)
Affinity DataIC50: 57nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459737(CHEMBL4211204)
Affinity DataIC50: 82nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459731(CHEMBL4216416)
Affinity DataIC50: 120nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625618(CHEMBL5429859)
Affinity DataIC50: 120nMAssay Description:Inhibition of MLLT3 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459738(CHEMBL4209820)
Affinity DataIC50: 140nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459730(CHEMBL4211714)
Affinity DataIC50: 149nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625619(CHEMBL4752253)
Affinity DataIC50: 160nMAssay Description:Inhibition of MLLT3 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625617(CHEMBL5421606)
Affinity DataIC50: 200nMAssay Description:Inhibition of MLLT3 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459747(CHEMBL4216933)
Affinity DataIC50: 341nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459735(CHEMBL4216170)
Affinity DataIC50: 369nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459726(CHEMBL4211962)
Affinity DataIC50: 372nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50576674(CHEMBL4850575)
Affinity DataIC50: 410nMAssay Description:Inhibition of AF9 YEATS domain (1 to 138 residues) (unknown origin) assessed as inhibition of probe-1 induced AF9 YEATS domain labelling incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625612(CHEMBL5416331)
Affinity DataIC50: 500nMAssay Description:Inhibition of MLLT3 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625616(CHEMBL5398308)
Affinity DataIC50: 500nMAssay Description:Inhibition of MLLT3 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50529556(CHEMBL4552313)
Affinity DataIC50: 600nMAssay Description:Binding affinity to MLLT3 in human HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625604(CHEMBL5439680)
Affinity DataIC50: 630nMAssay Description:Inhibition of MLLT3 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50566890(CHEMBL4865432)
Affinity DataIC50: 729nMAssay Description:Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625619(CHEMBL4752253)
Affinity DataIC50: 760nMAssay Description:Binding affinity to MLLT3 in human HEK293 cells by NanoBRET assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459733(CHEMBL4209508)
Affinity DataIC50: 850nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50566877(CHEMBL4863719)
Affinity DataIC50: 984nMAssay Description:Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459722(CHEMBL4204545)
Affinity DataIC50: 1.02E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459739(CHEMBL4204942)
Affinity DataIC50: 1.04E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459745(CHEMBL4210431)
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459742(CHEMBL4204647)
Affinity DataIC50: 1.14E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459743(CHEMBL4209087)
Affinity DataIC50: 1.20E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459748(CHEMBL4213382)
Affinity DataIC50: 1.49E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459746(CHEMBL4212941)
Affinity DataIC50: 1.66E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50576675(CHEMBL4848627)
Affinity DataIC50: 1.74E+3nMAssay Description:Inhibition of AF9 YEATS domain (1 to 138 residues) (unknown origin) assessed as inhibition of probe-1 induced AF9 YEATS domain labelling incubated fo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2022
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459736(CHEMBL4216206)
Affinity DataIC50: 1.78E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50566867(CHEMBL4855926)
Affinity DataIC50: 1.85E+3nMAssay Description:Inhibition of human His-AF9 YEATS domain and biotinylated H3K9ac peptide interaction by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2022
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459729(CHEMBL4217882)
Affinity DataIC50: 2.37E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625613(CHEMBL5394670)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of MLLT3 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50616142(CHEMBL5428051)
Affinity DataIC50: 2.98E+3nMAssay Description:Inhibition of N-terminal nanoLuc-tagged YEATS3 in HEK293T cells co-transfected with C-terminal halo-tagged histone 3.3 incubated for 24 hrs in presen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50625614(CHEMBL5427853)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of MLLT3 YD domain (unknown origin) assessed as disruption of histone peptide binding using histone peptide as substrate by HTRF assayMore data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/18/2024
Entry Details
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459732(CHEMBL4206070)
Affinity DataIC50: 3.49E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459734(CHEMBL4208554)
Affinity DataIC50: 4.11E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
TargetProtein AF-9(Human)
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50459740(CHEMBL4214833)
Affinity DataIC50: 4.29E+3nMAssay Description:Displacement of N-Flu-DOT1L from MBP-tagged AF9 (unknown origin) (487 to 568 residues) expressed in Escherichia coli BL21(DE3) measured after 3 hrs b...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/16/2020
Entry Details Article
PubMed
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