Affinity DataKd: 39nMAssay Description:Displacement of [3H]kainate from rat GLUK6 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR6 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR6 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR6 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: 6.60E+4nMAssay Description:Activity at rat cloned iGluR6 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR6 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: 8.20E+4nMAssay Description:Activity at rat cloned iGluR6 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat recombinant GluR6(Q) RNA-edited isoform expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo...More data for this Ligand-Target Pair
Affinity DataEC50: 7.30E+4nMAssay Description:Agonist activity at rat recombinant GluR6(Q) RNA-edited isoform expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo...More data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat recombinant GluR6(Q) RNA-edited isoform expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo...More data for this Ligand-Target Pair
Affinity DataEC50: 1.80E+3nMAssay Description:Agonist activity at rat recombinant GluR6(Q) RNA-edited isoform expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at recombinant rat full length GluK2 receptor expressed in HEK293T cells assessed as inhibition of glutamate induced increase in ...More data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.10nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.70nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 2.80nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.60nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 3.90nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 6.04nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 9.10nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 9.5nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 11.9nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 12.7nMAssay Description:Displacement of [3H]kainic acid from rat recombinant iGluR6(V,C,R) receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 12.7nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
Affinity DataKi: 18.5nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23.3nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: >100nMAssay Description:Displacement of [3H]KA from rat recombinant GluR6 expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 123nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 134nMAssay Description:Displacement of [3H]SYM2081 from rat recombinant iGluR6More data for this Ligand-Target Pair
Affinity DataKi: 210nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
Affinity DataKi: 230nMAssay Description:Inhibition of [3H]kainate binding at rat forebrain ionotropic glutamate receptor kainate 2More data for this Ligand-Target Pair
