Compile Data Set for Download or QSAR
Report error Found 117 of affinity data for UniProtKB/TrEMBL: P41148
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50087813(CHEMBL3426786)
Affinity DataKd:  520nMAssay Description:Binding affinity to canine full-length His-tagged GRP94 (28 to 754 residues lacking 287 to 327 residues) expressed in Escherichia coli by tryptophan ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/6/2016
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50366480(ATP | ADENOSINE TRIPHOSPHATE)
Affinity DataEC50:  1.90E+4nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50191366(17-((S)-amino-3,2-propanediol)-17-demethoxygeldana...)
Affinity DataEC50:  131nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50191367(17-allylamino-17-demethoxygeldanamycin hydroquinon...)
Affinity DataEC50:  119nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50191368(17-amino-17-demethoxygeldanamycin hydroquinone hyd...)
Affinity DataEC50:  48nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50368125(ADP | ADENOSINE DIPHOSPHATE)
Affinity DataEC50:  2.10E+4nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50191365(Allyl-((12E,16Z,18E)-(7R,9S,10R,11S,14S,15S)-14-ca...)
Affinity DataEC50: >1.00E+4nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM15359(17AAG | Tanespimycin | GLD-36 | (4E,6Z,8S,9S,10E,1...)
Affinity DataEC50:  124nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50030868(17-amino-17-demethoxygeldanamycin | Carbamic acid ...)
Affinity DataEC50:  48nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50191364(17-((S)-amino-3,2-propanediol)-17-demethoxygeldana...)
Affinity DataEC50:  72nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439623(CHEMBL2419342)
Affinity DataKd:  6.60nMAssay Description:Binding affinity to dog Grp94 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439624(CHEMBL1910764)
Affinity DataKd:  31nMAssay Description:Binding affinity to dog Grp94 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50439625(CHEMBL2419341)
Affinity DataKd:  2.5nMAssay Description:Binding affinity to dog Grp94 by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM31996(CHEMBL383824 | 17-(dimethylaminoethylamino)-17-dem...)
Affinity DataEC50:  65nMAssay Description:Inhibition of BODIPY-AG binding to dog Grp94More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50087813(CHEMBL3426786)
Affinity DataKd:  520nMAssay Description:Inhibition of FITC-geldanamycin binding to canine GRP94 incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50087812(CHEMBL3426787)
Affinity DataKd:  1.38E+3nMAssay Description:Inhibition of FITC-geldanamycin binding to canine GRP94 incubated for 5 hrs by fluorescence polarization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279156(CHEMBL4169566)
Affinity DataKd:  31nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279157(CHEMBL4168916)
Affinity DataKd:  9.89E+3nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279158(CHEMBL4175693)
Affinity DataKd:  34nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279170(CHEMBL4162283)
Affinity DataKd:  59nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279171(CHEMBL4170382)
Affinity DataKd:  30nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279160(CHEMBL4176780)
Affinity DataKd:  770nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279161(CHEMBL4168694)
Affinity DataKd: >1.00E+5nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279187(CHEMBL4174059)
Affinity DataKd:  8nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279173(CHEMBL4162694)
Affinity DataKd:  40nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279188(CHEMBL4172951)
Affinity DataKd:  60nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279159(CHEMBL4177418)
Affinity DataKd:  29nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279172(CHEMBL4159747)
Affinity DataKd:  21nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279189(CHEMBL4165074)
Affinity DataKd:  70nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279190(CHEMBL4161657)
Affinity DataKd:  29nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279174(CHEMBL4172281)
Affinity DataKd: >1.00E+4nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279185(CHEMBL4173418)
Affinity DataKd:  15nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279186(CHEMBL4165495)
Affinity DataKd:  17nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279155(CHEMBL4160774)
Affinity DataKd:  13nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM227590(PA1)
Affinity DataKd:  20nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM50279191(CHEMBL4170618)
Affinity DataKd:  13nMAssay Description:Displacement of FITC-GDA from recombinant canine Grp94 expressed in baculovirus infected Sf21 insect cells after 24 hrs by fluorescence polarization ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/13/2020
Entry Details Article
PubMed
TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501623(US11028041, Compound 6)
Affinity DataKd:  630nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501624(US11028041, Compound 7)
Affinity DataKd:  1.04E+4nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501625(US11028041, Compound 16)
Affinity DataKd:  450nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501626(US11028041, Compound 17)
Affinity DataKd:  680nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501627(US11028041, Compound 18)
Affinity DataKd:  730nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501628(US11028041, Compound 19)
Affinity DataKd:  280nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501629(US11028041, Compound 20)
Affinity DataKd:  240nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501630(US11028041, Compound 21)
Affinity DataKd:  180nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501631(US11028041, Compound 22)
Affinity DataKd:  300nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501632(US11028041, Compound 23)
Affinity DataKd:  330nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501633(US11028041, Compound 24)
Affinity DataKd:  540nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501634(US11028041, Compound 25)
Affinity DataKd:  6.10E+3nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501635(US11028041, Compound 26)
Affinity DataKd:  7.80E+3nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

TargetEndoplasmin(Dog)
Sloan-Kettering Institute For Cancer Research

Curated by ChEMBL
LigandPNGBDBM501636(US11028041, Compound 27)
Affinity DataKd:  5.50E+3nMAssay Description:The assay was performed in 96-well black, flat-bottom plates with a final volume of 100 μL. 25 μL of assay buffer (20 mM HEPES, pH 7.3, 50 ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/29/2021
Entry Details
Go to US Patent

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