Compile Data Set for Download or QSAR
Report error Found 16 of affinity data for UniProtKB/TrEMBL: P35813
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50061067(8-[3-amino(imino)methylaminopropyl]-15-isobutyl-5-...)
Affinity DataIC50: 3nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50090297(Hexadecanoic acid (R)-2-hydroxy-2-((5S,8R)-2-isopr...)
Affinity DataIC50: 3.00E+3nMAssay Description:Compound was evaluated for inhibitory effect against protein phosphatase I (PP-I)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50090298(Hexadecanoic acid (R)-2-((4aS,7R,7aR)-2,4a-dihydro...)
Affinity DataIC50: 1.10E+4nMAssay Description:Compound was evaluated for inhibitory effect against protein phosphatase I (PP-I)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50183456(N-methyl-N'-9-phenanthrylimidodicarbonimidic diami...)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of PP2C alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50343530(5,7-dichloro-4-((3-(4-methoxyphenylthio)benzyl)(me...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of PPM1A (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50031908(CHEMBL3360906)
Affinity DataIC50: 3.18E+4nMAssay Description:Inhibition of PPM1A (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50031910(CHEMBL3360908)
Affinity DataIC50: 4.25E+4nMAssay Description:Inhibition of PPM1A (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135681((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Amino-9-methoxy-2,6...)
Affinity DataIC50: 4.50E+4nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50031906(CHEMBL3360905)
Affinity DataIC50: 6.78E+4nMAssay Description:Inhibition of PPM1A (unknown origin) assessed as reduction in pNPP hydrolysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/12/2016
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135676((S)-2-[(R)-2-(2-{[(R)-4-((4E,6E)-(2S,3S,8S,9S)-3-A...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135677((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135680((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135675((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135679((S)-2-[(R)-2-(2-{[(R)-4-((4E,6E)-(2S,3S,8S,9S)-3-A...)
Affinity DataIC50: 2.30E+5nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135678((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Amino-9-methoxy-2,6...)
Affinity DataIC50: 2.80E+5nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetProtein phosphatase 1A(Human)
University of California Irvine

Curated by ChEMBL
LigandPNGBDBM50135674((R)-2-((4E,6E)-(2S,3S,8S,9S)-3-Acetylamino-9-metho...)
Affinity DataIC50: 4.00E+5nMAssay Description:Inhibitory concentration required against protein phosphatase 1 using pNPP assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed