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TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065450(2-Amino-3-phenyl-N-{4-[(2S,5S,8S,14S,17R)-8,10,14-...)
Affinity DataKd:  69nMAssay Description:In vitro inhibition of radioligand binding to human Somatostatin receptor type 5 expressed in CCL-39 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataEC50:  0.190nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50169467(4-{3-[2-(5-Chloro-1H-indol-3-yl)-ethylsulfanyl]-5-...)
Affinity DataEC50:  52nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50169465(3-[4-(4-Amino-butyl)-5-quinolin-2-yl-4H-[1,2,4]tri...)
Affinity DataEC50:  2.30nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50169462(4-{3-[2-(7-Methyl-1H-indol-3-yl)-ethylsulfanyl]-5-...)
Affinity DataEC50:  34nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50169468(4-{3-[2-(6-Fluoro-1H-indol-3-yl)-ethylsulfanyl]-5-...)
Affinity DataEC50:  44nMAssay Description:Inhibition of forskolin-induced cAMP accumulation in CHO-K1 cells expressing human sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/2/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065451(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  407nMAssay Description:In vitro inhibition of radioligand binding to human Somatostatin receptor type 5 expressed in CCL-39 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065453(CHEMBL421362 | L-361,301 | L-363,301 | L-363301 | ...)
Affinity DataKd:  7.60nMAssay Description:In vitro inhibition of radioligand binding to human Somatostatin receptor type 5 expressed in CCL-39 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065452(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  6.17nMAssay Description:In vitro inhibition of radioligand binding to human Somatostatin receptor type 5 expressed in CCL-39 cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM81767(15-28-Somatostatin-28 | CB6417646 | CAS_38916-34-6...)
Affinity DataEC50:  0.0650nMAssay Description:Effective concentration on human somatostatin receptor 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098604(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  114nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098607(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  629nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098617(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  71.8nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098608(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  83.2nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098616(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  8.41nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098614(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  28.4nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098619(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  8.35nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098613(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  27nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098618(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  33.0nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098612(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  4.89nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098611(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  50.4nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098609(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  313nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098610(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  16.9nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098602(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098606(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  95.0nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098605(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  92.8nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098615(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  0.610nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098603(10-(4-Amino-butyl)-19-[(2-amino-3-phenyl-propionyl...)
Affinity DataKd:  23.7nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50215029((2S)-6-amino-N-benzyl-2-[(4R)-3-oxo-4-[(phenylacet...)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human SST5 receptor expressed in CHOK1 cells assessed as effect on forskolin-induced cAMP productionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322980(N-(1-((2,6-diethoxybiphenyl-4-yl)methyl)piperidin-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322979(N-(1-((2,6-diethoxy-4'-fluorobiphenyl-4-yl)methyl)...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322978(6-amino-N-(1-((2-(benzyloxy)-6-ethoxy-4'-fluorobip...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322977(N-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-yl)-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322973(N-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-yl)-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322971(rac-N-(1-((2,6-diethoxy-4'-fluorobiphenyl-4-yl)met...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322983(N-(1-((2,6-diethoxybiphenyl-4-yl)methyl)piperidin-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322982(6-chloro-N-(1-((2,6-diethoxy-4'-fluorobiphenyl-4-y...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322981(N-(1-((2,6-diethoxy-4'-fluorobiphenyl-4-yl)methyl)...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322993(6-amino-N-(1-(3-ethoxy-4-methylbenzyl)piperidin-4-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322992(N-(1-((2-ethoxy-4'-fluorobiphenyl-4-yl)methyl)pipe...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322990(rac-6-amino-N-(1-(3-ethoxy-4,5-difluorobenzyl)azep...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322989(N-(1-(3,5-diethoxy-4-(1H-imidazol-1-yl)benzyl)pipe...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322987(N-(1-(4-chloro-3,5-diethoxybenzyl)piperidin-4-yl)-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322986(N-(1-((2,6-diethoxy-4'-(trifluoromethoxy)biphenyl-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322985(6-amino-N-(1-((2,6-diethoxy-4'-fluorobiphenyl-4-yl...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50322984(N-(1-(3,5-diethoxy-4-fluorobenzyl)piperidin-4-yl)-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Antagonist activity at human SST5 receptor expressed in CHO cells assessed as inhibition of forskolin-induced cAMP accumulation by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/19/2011
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50097789(2-[8-(3-Amino-propyl)-6-benzo[b]thiophen-3-yl-imid...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity on human somatostatin receptor 5More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423297(Obelin | CHEMBL251541)
Affinity DataKd:  1.78E+3nMAssay Description:Binding affinity to human recombinant sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423462(CHEMBL251835)
Affinity DataKd:  6.46E+3nMAssay Description:Binding affinity to human recombinant sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 5(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50423465(ERGOLINE)
Affinity DataKd:  5.62E+4nMAssay Description:Binding affinity to human recombinant sst5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
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