Compile Data Set for Download or QSAR
Report error Found 71 of affinity data for UniProtKB/TrEMBL: P34978
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391305(CHEMBL433884)
Affinity DataKd:  39.8nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391303(CHEMBL158576)
Affinity DataKd:  10nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391309(GR-83783 | CHEMBL159517)
Affinity DataKd:  31.6nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391310(CHEMBL158875)
Affinity DataKd:  25.1nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391307(CHEMBL162133)
Affinity DataKd:  15.8nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391313(CHEMBL159787)
Affinity DataKd:  12.6nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391301(CHEMBL162409)
Affinity DataKd:  3.16nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391312(CHEMBL345876)
Affinity DataKd:  3.16nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391311(CHEMBL352040)
Affinity DataKd:  10nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391308(CHEMBL159860)
Affinity DataKd:  19.9nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391306(CHEMBL161532)
Affinity DataKd:  3.16nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50010960((E)-7-Phenyl-7-pyridin-3-yl-hept-6-enoic acid | CV...)
Affinity DataKd:  6.31E+3nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391304(CHEMBL350292)
Affinity DataKd:  15.8nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283057((1R,5S,6R,7R)-6-((Z)-7-Hydroxy-hept-2-enyl)-7-((E)...)
Affinity DataEC50:  1nMAssay Description:Activity against thromboxane A2 receptor evaluated by contraction of isolated rat thoracic aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283058((Z)-7-[(1R,5S,6R,7R)-7-((E)-3-Hydroxy-oct-1-enyl)-...)
Affinity DataEC50:  324nMAssay Description:Activity against thromboxane A2 receptor evaluated by contraction of isolated rat thoracic aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283059((Z)-7-[(1R,5S,6R,7R)-7-((E)-3-Hydroxy-oct-1-enyl)-...)
Affinity DataEC50:  0.230nMAssay Description:Activity against thromboxane A2 receptor evaluated by contraction of isolated rat thoracic aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50283060((Z)-7-[(1R,5S,6R,7R)-7-((E)-3-Hydroxy-oct-1-enyl)-...)
Affinity DataEC50:  58nMAssay Description:Activity against thromboxane A2 receptor evaluated by contraction of isolated rat thoracic aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50212318(BMS-180291 | Ifetroban)
Affinity DataKd:  4nMAssay Description:Inhibition of [3H]-SQ 29,548 radioligand binding to thromboxane A2 (TXA2) receptor of human platelet membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391300(CHEMBL162691)
Affinity DataKd:  79.4nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50003795(5-[Pyridin-3-yl-(3-trifluoromethyl-phenyl)-methyle...)
Affinity DataKd:  1.26E+3nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50391302(CHEMBL349625)
Affinity DataKd:  31.6nMAssay Description:In vitro thromboxane A2 receptor antagonism through inhibition of U-46619-induced contraction of rat isolated thoracic aortic stripMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/19/2013
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50013027(CHEMBL262655 | Sodium; 3-[4-(4-chloro-benzenesulfo...)
Affinity DataIC50: 0.900nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075089(Sodium; [2-(4-chloro-benzenesulfonylamino)-indan-5...)
Affinity DataIC50: 2.20nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075088(Sodium; {2-[(4-chloro-benzenesulfonylamino)-methyl...)
Affinity DataIC50: 3nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075086(Sodium; [2-(benzenesulfonylamino-methyl)-indan-5-y...)
Affinity DataIC50: 13nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075091(Sodium; 3-{2-[(4-chloro-benzenesulfonylamino)-meth...)
Affinity DataIC50: 15nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075077(Sodium; {2-[(naphthalene-2-sulfonylamino)-methyl]-...)
Affinity DataIC50: 22nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075082(Sodium; 2-[(4-chloro-benzenesulfonylamino)-methyl]...)
Affinity DataIC50: 26nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075094(Sodium; {2-[2-(4-chloro-benzenesulfonylamino)-ethy...)
Affinity DataIC50: 32nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075093(Sodium; 5-{2-[(4-chloro-benzenesulfonylamino)-meth...)
Affinity DataIC50: 36nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50002805(CHEMBL71685 | (daltroban){4-[2-(4-Chloro-benzenesu...)
Affinity DataIC50: 37nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075079(Sodium; 4-{2-[(4-chloro-benzenesulfonylamino)-meth...)
Affinity DataIC50: 39nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075096(Sodium; 2-[2-(4-chloro-benzenesulfonylamino)-ethyl...)
Affinity DataIC50: 66nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075092(Sodium; 2-[3-(4-chloro-benzenesulfonylamino)-propy...)
Affinity DataIC50: 85nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075076(Sodium; {2-[(thiophene-2-sulfonylamino)-methyl]-in...)
Affinity DataIC50: 85nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075085(Sodium; {2-[(4-chloro-benzenesulfonylamino)-methyl...)
Affinity DataIC50: 141nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282138(Sodium; 3-[4-(4-chloro-phenylsulfamoyl)-butyl]-6-i...)
Affinity DataIC50: 220nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075090(Sodium; {2-[(naphthalene-1-sulfonylamino)-methyl]-...)
Affinity DataIC50: 295nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075081(Sodium; 2-[4-(4-chloro-benzenesulfonylamino)-butyl...)
Affinity DataIC50: 479nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075084(Sodium; {2-[3-(4-chloro-benzenesulfonylamino)-prop...)
Affinity DataIC50: 513nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282141(Sodium; 3-[5-(4-chloro-phenylsulfamoyl)-pentyl]-6-...)
Affinity DataIC50: 860nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282135(Sodium; 3-[3-(4-chloro-phenylsulfamoyl)-propyl]-6-...)
Affinity DataIC50: 860nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075095(Sodium; {2-[4-(4-chloro-benzenesulfonylamino)-buty...)
Affinity DataIC50: 977nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075080(Sodium; [2-(cyclohexanesulfonylamino-methyl)-indan...)
Affinity DataIC50: 1.20E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50075083(Sodium; {2-[(pentane-1-sulfonylamino)-methyl]-inda...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro thromboxane A2 antagonistic activity on U-46619 (0.1 uM) induced contraction of rat aortaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282152(Sodium; 6-isopropyl-3-(5-phenylsulfamoyl-pentyl)-a...)
Affinity DataIC50: 1.40E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50002765(BM 13177 | CHEMBL8273 | [4-(2-Benzenesulfonylamino...)
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282146(Sodium; 6-isopropyl-3-(4-phenylsulfamoyl-butyl)-az...)
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282136(6-Isopropyl-3-(5-phenylsulfamoyl-pentyl)-azulene-1...)
Affinity DataIC50: 1.50E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

TargetThromboxane A2 receptor(Rat)
TBA

Curated by ChEMBL
LigandPNGBDBM50282156(3-[5-(4-Chloro-phenylsulfamoyl)-pentyl]-6-isopropy...)
Affinity DataIC50: 1.70E+3nMAssay Description:Tested for antagonistic activity on isolated rat thoracic aorta (thromboxane A2 receptor) precontracted by U-46619 (3 x 10 e-8 M)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2010
Entry Details Article

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