Compile Data Set for Download or QSAR
Report error Found 85 of affinity data for UniProtKB/TrEMBL: P34971
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50225516(CHEMBL156326)
Affinity DataEC50:  1.60E+5nMAssay Description:Effective concentration against 125I]iodocyanopindolol(ICYP) binding to beta adrenergic receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  980nMAssay Description:Effective concentration against 125I]iodocyanopindolol(ICYP) binding to beta adrenergic receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50225515(CHEMBL345618)
Affinity DataEC50:  49nMAssay Description:Effective concentration against 125I]iodocyanopindolol(ICYP) binding to beta adrenergic receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50225514(CHEMBL160277)
Affinity DataKd:  1.00E+4nMAssay Description:KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50225513(CHEMBL423055)
Affinity DataKd:  470nMAssay Description:KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) binding in SF-49 lymphoma cellMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50225512(CHEMBL157187)
Affinity DataKd:  320nMAssay Description:KD constant value was evaluated for the displacement of ICYP (iodocyanopindolol) bindingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50225511(CHEMBL160788)
Affinity DataEC50:  8.70nMAssay Description:Effective concentration against 125I]iodocyanopindolol(ICYP) binding to beta adrenergic receptor was determinedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2018
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50027663(Carazolol | 1-(9H-carbazol-4-yloxy)-3-(isopropylam...)
Affinity DataKi:  0.0900nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50167072(CHEMBL3799125)
Affinity DataKi:  0.210nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526681(CHEMBL4537221)
Affinity DataKi:  0.490nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526679(CHEMBL4456301)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM25746(cid_2685 | 2-hydroxy-5-{2-[(2-hydroxy-3-{4-[1-meth...)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM25761(Propanolol,(+/-) | PROPRANOLOL, l- | PROPRANOLOL,(...)
Affinity DataKi:  2.40nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526684(CHEMBL4437569)
Affinity DataKi:  2.60nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50167073(CHEMBL3798017)
Affinity DataKi:  3.40nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50166979(CHEMBL3798748)
Affinity DataKi:  5.10nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM25751(Bisoprolol fumarate | Concor | [2-hydroxy-3-(4-{[2...)
Affinity DataKi:  5.30nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50167066(CHEMBL3800400)
Affinity DataKi:  5.80nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525097(CHEMBL4593181)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525100(CHEMBL4451135)
Affinity DataKi:  6.60nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525095(CHEMBL4435895)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525098(CHEMBL1160694)
Affinity DataKi:  14nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526685(CHEMBL4566666)
Affinity DataKi:  22nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525101(CHEMBL4513932)
Affinity DataKi:  24nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526690(CHEMBL4553747)
Affinity DataKi:  27nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526686(CHEMBL4463246)
Affinity DataKi:  29nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526680(CHEMBL4463925)
Affinity DataKi:  33nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526682(CHEMBL4443911)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM25756(Betalok | Spesikor | {2-hydroxy-3-[4-(2-methoxyeth...)
Affinity DataKi:  49nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526687(CHEMBL4576034)
Affinity DataKi:  71nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50167063(CHEMBL3800341)
Affinity DataKi:  79nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50166977(CHEMBL3800303)
Affinity DataKi:  85nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50166976(CHEMBL3799455)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526683(CHEMBL4450085)
Affinity DataKi:  150nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50167064(CHEMBL3797876)
Affinity DataKi:  160nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50166980(CHEMBL3797205)
Affinity DataKi:  180nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50407517(CHEMBL1160723 | (-)ISOPROTERENOL | US9492405, 27)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526688(CHEMBL4473272)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataKi:  220nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50167067(CHEMBL3800468)
Affinity DataKi:  300nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525106(CHEMBL4470694)
Affinity DataKi:  310nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525105(CHEMBL4436343)
Affinity DataKi:  330nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525096(CHEMBL4450756)
Affinity DataKi:  340nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50167068(CHEMBL3799427)
Affinity DataKi:  530nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2017
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM25771(salmeterol xinafoate | 4-(1-hydroxy-2-{[6-(4-pheny...)
Affinity DataKi:  550nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50526689(CHEMBL4456505)
Affinity DataKi:  740nMAssay Description:Displacement of [3H]CGP12177 from mouse beta1 adrenoceptor expressed in HEK293T cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525107(CHEMBL4439238)
Affinity DataKi:  860nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Mouse)
TBA

Curated by ChEMBL
LigandPNGBDBM50525093(CHEMBL4437939)
Affinity DataKi:  1.20E+3nMAssay Description:Displacement of [3H]-CGP-12177 from murine beta1-adrenergic receptor expressed in HEK293T cells after 60 mins by radioligand competition binding assa...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
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