Compile Data Set for Download or QSAR
Report error Found 19 of affinity data for UniProtKB/TrEMBL: P33436
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199123(N-(4-(1-(4,6-bis((4-hydroxyphenyl)amino)-1,3,5-tri...)
Affinity DataIC50: 8.12nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199124(N-(4-(1-(4,6-bis((4-methoxyphenyl)amino)-1,3,5-tri...)
Affinity DataIC50: 18.6nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199128(N-(4-(1-(4,6-dimorpholino-1,3,5-triazin-2-yl)-5-(4...)
Affinity DataIC50: 42.3nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199127(N-(4-(1-(4,6-di(piperazin-1-yl)-1,3,5-triazin-2-yl...)
Affinity DataIC50: 55.3nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199125(N-(4-(1-(4,6-bis(o-tolylamino)-1,3,5-triazin-2-yl)...)
Affinity DataIC50: 67.1nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199126(N-(4-(1-(4,6-bis((4-nitrophenyl)amino)-1,3,5-triaz...)
Affinity DataIC50: 76.6nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199122(N-(4-(1-(4,6-bis(phenylamino)-1,3,5-triazin-2-yl)-...)
Affinity DataIC50: 123nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199121(N-(4-(1-(4,6-bis((3-aminopropyl)amino)-1,3,5-triaz...)
Affinity DataIC50: 189nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199120(N-(4-(1-(4,6-bis(ethylamino)-1,3,5-triazin-2-yl)-5...)
Affinity DataIC50: 332nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM199119(N-(4-(1-(4,6-bis(methylamino)-1,3,5-triazin-2-yl)-...)
Affinity DataIC50: 666nMpH: 7.5 T: 2°CAssay Description:For this assay, the reagents used as follows. The substrate corresponds to Mca-Pro-Leu-Gly-Leu-Dpa-Ala-Arg 25 mm in assay buffer. This low-fluorescen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2016
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM50310832(Clinopodic acid C | CHEMBL1080779)
Affinity DataIC50: 3.26E+3nMAssay Description:Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM50250808(lithospermic acid | CHEMBL518243)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM50133496(Rosmarinic acid, 2 | cid_5281792 | CHEMBL324842 | ...)
Affinity DataIC50: 2.72E+4nMAssay Description:Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM50310827(clinopodic acid H | CHEMBL1079357)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM50310828(clinopodic acid F | CHEMBL1079356)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM50310829(clinopodic acid E | CHEMBL1081512)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM50310830(Clinopodic acid B | CHEMBL1080778)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM50310831(Clinopodic acid A | CHEMBL1079231)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
Target72 kDa type IV collagenase(Rat)
Zhejiang Hospital

LigandPNGBDBM50210054(3-(3,4-dihydroxy-phenyl)-acrylic acid 2-(3,4-dihyd...)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of gelatinolytic activity of MMP2 in rat lung homogenate after 40 mins by SDS-PAGE preincubated for 30 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed