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Report error Found 1604 for UniProtKB: P32745
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065450(2-Amino-3-phenyl-N-{4-[(2S,5S,8S,14S,17R)-8,10,14-...)
Affinity DataKd:  282nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst3) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065451(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  407nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst3) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065452(2-Amino-N-{4-[(2S,5S,8S,14S,17R)-8,14-dibenzyl-5-(...)
Affinity DataKd:  339nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst3) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50065453(CHEMBL421362 | L-361,301 | L-363,301 | L-363301 | ...)
Affinity DataKd:  525nMAssay Description:In vitro inhibition of radioligand binding to human somatostatin receptor (hsst3) expressed in CHO cells.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021063(CHEMBL3287613)
Affinity DataEC50:  2.90nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021064(CHEMBL3287614)
Affinity DataEC50:  6.10nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021065(CHEMBL3287615)
Affinity DataEC50:  122nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021066(CHEMBL3287616)
Affinity DataEC50:  21nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021067(CHEMBL3287617)
Affinity DataEC50:  13nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021068(CHEMBL3287618)
Affinity DataEC50:  36nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021069(CHEMBL3287619)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021070(CHEMBL3287620)
Affinity DataEC50:  1.52E+4nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021071(CHEMBL3287621)
Affinity DataEC50:  59nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021072(CHEMBL3287622)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021073(CHEMBL3287627)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021074(CHEMBL3287628)
Affinity DataEC50:  0.516nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021075(CHEMBL3287629)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021076(CHEMBL3287630)
Affinity DataEC50:  26nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021089(CHEMBL3287631)
Affinity DataEC50:  22nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021090(CHEMBL3287632)
Affinity DataEC50:  3.70nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021091(CHEMBL3287635)
Affinity DataEC50:  133nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021092(CHEMBL3287639)
Affinity DataEC50:  9.58E+3nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021093(CHEMBL3287643)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021057(CHEMBL3287647)
Affinity DataEC50:  91nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021059(CHEMBL3287648)
Affinity DataEC50:  2.84E+4nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021060(CHEMBL3287649)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021094(CHEMBL3287651)
Affinity DataEC50:  327nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50021061(CHEMBL3287650)
Affinity DataEC50:  348nMAssay Description:Agonist activity at human SST3 expressed in CHO-K1 cells assessed as foreskin-stimulated cAMP accumulation after 45 mins by TR-FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/12/2015
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098605(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  440nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098606(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  94.2nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098609(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  124nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098608(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  830nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098615(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  11.1nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098617(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  535nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098616(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  67.5nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098603(10-(4-Amino-butyl)-19-[(2-amino-3-phenyl-propionyl...)
Affinity DataKd:  13nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098619(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  11.8nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098602(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd: >1.00E+3nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098610(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  17nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098618(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  18.2nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098613(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  3.01nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098612(10-(4-Amino-butyl)-16-benzyl-7-(1-hydroxy-ethyl)-1...)
Affinity DataKd:  17.9nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098614(10-(4-Amino-butyl)-19-(2-amino-3-phenyl-propionyla...)
Affinity DataKd:  44.4nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098607(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  51.0nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098611(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  8nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50098604(10-(4-Amino-butyl)-19-[2-amino-3-(4-hydroxy-phenyl...)
Affinity DataKd:  2.73nMAssay Description:Binding affinity was determined on cloned human somatostatin receptor-1 (hsst3)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50389589(CHEMBL2069501)
Affinity DataKd:  2nMAssay Description:Antagonist activity at human SST3 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/8/2013
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50110439(CHEMBL3605784)
Affinity DataEC50:  160nMAssay Description:Agonist activity at human SSTR3 expressed in CHO cells assessed as intracellular cAMP level after 45 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2016
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50110440(CHEMBL3605785)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human SSTR3 expressed in CHO cells assessed as intracellular cAMP level after 45 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2016
Entry Details Article
PubMed
TargetSomatostatin receptor type 3(Human)
University of California San Diego

Curated by ChEMBL
LigandPNGBDBM50110441(CHEMBL3605786)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human SSTR3 expressed in CHO cells assessed as intracellular cAMP level after 45 mins by time-resolved fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2016
Entry Details Article
PubMed
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