Compile Data Set for Download or QSAR
Report error Found 36 of affinity data for UniProtKB/TrEMBL: P31750
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50299148(1-{4-[(3-cyclopropyl-1H-pyrazol-5-yl)amino]pyrrolo...)
Affinity DataIC50: 22nMAssay Description:Inhibition of Akt phosphorylation in mouse Sal cells by Western blottingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338966(Phosphatidylinositol(3,4,5)-trisphosphate | CHEMBL...)
Affinity DataKi:  500nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338967(D-3-deoxyphosphatidylinositol ether lipid | CHEMBL...)
Affinity DataKi:  1.60E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50304369(4-dodecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonam...)
Affinity DataKi:  2.40E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338956(Ethyl 2-(5-(4-Dodecylphenylsulfonamido)-1,3,4-thia...)
Affinity DataKi:  4.30E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338955(2-(5-(4-Dodecylphenylsulfonamido)-1,3,4-thiadiazol...)
Affinity DataKi:  5.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338949(4-Tetradecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfo...)
Affinity DataKi:  5.60E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338959(5-(4-Dodecylphenylsulfonamido)-1,3,4-thiadiazole-2...)
Affinity DataKi:  6.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338953(4-Dodecyl-N-(5-ethyl-1,3,4-thiadiazol-2-yl)benzene...)
Affinity DataKi:  7.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338958(4-Dodecyl-N-(5-(hydroxymethyl)-1,3,4-thiadiazol-2-...)
Affinity DataKi:  7.50E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338950(4-Hexadecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfon...)
Affinity DataKi:  7.60E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338939(N-(4-(N-(5-Ethyl-1,3,4-thiadiazol-2-yl)sulfamoyl)p...)
Affinity DataKi:  8.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338965(3-Dodecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonam...)
Affinity DataKi:  8.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338942(Ethyl 2-(5-(4-Decanamidophenylsulfonamido)-1,3,4-t...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338943(Ethyl 5-(4-Decanamidophenylsulfonamido)-1,3,4-thia...)
Affinity DataKi:  9.00E+3nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338941(2-(5-(4-Decanamidophenylsulfonamido)-1,3,4-thiadia...)
Affinity DataKi:  1.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338944(N-(4-(N-(5-(hydroxymethyl)-1,3,4-thiadiazol-2-yl)s...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338938(N-(4-(N-(5-Methyl-1,3,4-thiadiazol-2-yl)sulfamoyl)...)
Affinity DataKi:  1.10E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338940(N-(4-(N-(5-tert-Butyl-1,3,4-thiadiazol-2-yl)sulfam...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338951(4-Octadecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfon...)
Affinity DataKi:  1.20E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338961(N-(5-Ethyl-1,3,4-thiadiazol-2-yl)biphenyl-4-sulfon...)
Affinity DataKi:  1.70E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338964(ortho-Dodecyl-N-(1,3,4-thiadiazol-2-yl)benzenesulf...)
Affinity DataKi:  1.80E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338957(Ethyl 5-(4-Dodecylphenylsulfonamido)-1,3,4-thiadia...)
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338960(N-(1,3,4-Thiadiazol-2-yl)biphenyl-4-sulfonamide | ...)
Affinity DataKi:  1.90E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50304368(N-(4-(N-1,3,4-thiadiazol-2-ylsulfamoyl)phenyl)deca...)
Affinity DataKi:  2.20E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338962(2-(5-(Biphen-4-ylsulfonamido)-1,3,4-thiadiazol-2-y...)
Affinity DataKi:  4.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50304371(N-(4-(N-1,3,4-thiadiazol-2-ylsulfamoyl)phenyl)-2-(...)
Affinity DataKi:  4.10E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338963(para-Dodecyl-N-phenylbenzenesulfonamide | CHEMBL16...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338952(4-Dodecyl-N-(5-methyl-1,3,4-thiadiazol-2-yl)benzen...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338954(N-(5-tert-Butyl-1,3,4-thiadiazol-2-yl)-4-dodecylbe...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50034417(4-amino-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamid...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338948(4-Octyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamid...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338947(4-Hexyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamid...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338946(4-Butyl-N-(1,3,4-thiadiazol-2-yl)benzenesulfonamid...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50338945(N-(4-(N-(5-Sulfamoyl-1,3,4-thiadiazol-2-yl)sulfamo...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed
TargetRAC-alpha serine/threonine-protein kinase(Mouse)
Bristol-Myers Squibb

Curated by ChEMBL
LigandPNGBDBM50304370(N-(4-(N-1,3,4-thiadiazol-2-ylsulfamoyl)phenyl)acet...)
Affinity DataKi: >5.00E+4nMAssay Description:Displacement of biotinylated phosphatidylinositol-3,4,5-phosphate from mouse AKT1 PH domain by surface plasmon resonance competitive binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/24/2011
Entry Details Article
PubMed