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Report error Found 67 of affinity data for UniProtKB/TrEMBL: P25023
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408055(CHEMBL3038102)
Affinity DataKd:  50.1nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408053(CHEMBL3038094)
Affinity DataKd:  3.16nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408047(CHEMBL3038096)
Affinity DataKd:  18.6nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408045(CHEMBL2372278)
Affinity DataKd:  0.490nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408044(CHEMBL3038104)
Affinity DataKd:  174nMAssay Description:In vitro Bradykinin receptor B2 antagonist activity by using rat uterus functional assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50409528(CHEMBL2112220)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of Bradykinin receptor B2-mediated contractions of rat uterus smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50409527(CHEMBL2112283)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of Bradykinin receptor B2-mediated contractions of rat uterus smooth muscleMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50409527(CHEMBL2112283)
Affinity DataIC50: 105nMAssay Description:Inhibition of increase in [Ca2+] efflux from NG108-15 cells caused by activation of rat Bradykinin receptor B2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50409528(CHEMBL2112220)
Affinity DataIC50: 141nMAssay Description:Inhibition of increase in [Ca2+] efflux from NG108-15 cells caused by activation of rat Bradykinin receptor B2More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097740(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 410nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097734(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097736(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097723(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097730(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097737(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097732(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097727(CHEMBL351059 | CHEMBL163510 | (S)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097742(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097726(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097738(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097731(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097743(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097724(CHEMBL162787 | CHEMBL159456 | (R)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097733(CHEMBL351387 | CHEMBL164361 | (S)-1-[N'-(2-Nitro-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097727(CHEMBL351059 | CHEMBL163510 | (S)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097728(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097729(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097725(1-(2-nitrophenyl)thiosemicarbazide analogue | CHEM...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097724(CHEMBL162787 | CHEMBL159456 | (R)-1-{N'-[4-(2-Meth...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50097733(CHEMBL351387 | CHEMBL164361 | (S)-1-[N'-(2-Nitro-p...)
Affinity DataIC50: 1.00E+5nMAssay Description:In vitro binding affinity against Bradykinin receptor B2 in rat NG 108-15 neuroblastoma-glioma hybrid cell membranes using [3H]BK binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/5/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50370083(CHEMBL1907651)
Affinity DataKi:  0.0230nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50403371(Firazyr | HOE-140 | ICATIBANT)
Affinity DataKi:  0.0770nMAssay Description:Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50370077(CHEMBL1907652)
Affinity DataKi:  0.310nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50049949(2-(2-{[1-(2-{2-[2-({1-[1-(2-Amino-5-guanidino-pent...)
Affinity DataKi:  0.460nMAssay Description:Binding affinity against rat Bradykinin receptor B2 expressed in CHO cells using [3H]-bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50409120(CHEMBL2112044 | CHEMBL2112937)
Affinity DataKi:  0.5nMAssay Description:Inhibition of binding of [3H]BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50113263(CHEMBL308468 | CHEMBL431562 | (S)-1-[4-(4-benzhydr...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50113263(CHEMBL308468 | CHEMBL431562 | (S)-1-[4-(4-benzhydr...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50409120(CHEMBL2112044 | CHEMBL2112937)
Affinity DataKi:  0.600nMAssay Description:Inhibition of binding of [3H]BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50085685(4-benzhydrylamino(thioxo)methylhydrazine-3-nitrobe...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of binding of [3H]BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50085684(4-benzhydrylamino(thioxo)methylhydrazine-3-nitro-1...)
Affinity DataKi:  4nMAssay Description:Inhibition of binding of [3H]BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50370081(CHEMBL1907654)
Affinity DataKi:  5.46nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50408748(CHEMBL2112698)
Affinity DataKi:  6nMAssay Description:Binding affinity against rat bradykinin B2 receptors expressed in CHO cells using [3H]bradykinin as radioligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/12/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50370078(CHEMBL1907653)
Affinity DataKi:  7.30nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50409527(CHEMBL2112283)
Affinity DataKi:  10.7nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50370080(CHEMBL1907656)
Affinity DataKi:  14.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50085698(benzhydrylamino-2-nitrobenzylhydrazinemethanethion...)
Affinity DataKi:  38nMAssay Description:Inhibition of binding of [3H]BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50409529(CHEMBL2112221)
Affinity DataKi:  64.5nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50085696(1N,1N-di(3-dimethylaminopropyl)-4-benzhydrylamino(...)
Affinity DataKi:  148nMAssay Description:Inhibition of binding of [3H]BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50409528(CHEMBL2112220)
Affinity DataKi:  176nMAssay Description:Inhibition of specific binding of [3H]-BK (1 nM) to rat Bradykinin receptor B2 by 50% in NG108-15 cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/26/2012
Entry Details Article
PubMed
TargetB2 bradykinin receptor(Rat)
Cortech

Curated by ChEMBL
LigandPNGBDBM50085689(1N-benzyl-4-benzylamino(thioxo)methylhydrazine-3-n...)
Affinity DataKi:  310nMAssay Description:Inhibition of binding of [3H]BK to rat bradykinin B2 receptor expressed in NG108-15 neuroblastoma-glioma hybrid cell membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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