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Report error Found 134 of affinity data for UniProtKB/TrEMBL: P22411
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM11558(CHEMBL381806 | (3S)-2-[(3R)-3-amino-4-(2-fluorophe...)
Affinity DatapH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437403(CHEMBL2408771)
Affinity DataIC50: 0.0500nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437403(CHEMBL2408771)
Affinity DataIC50: 0.270nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50228407(8-((R)-3-amino-piperidin-1-yl)-3-methyl-7-(3-methy...)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437404(CHEMBL2408655)
Affinity DataIC50: 1nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437404(CHEMBL2408655)
Affinity DataIC50: 1.60nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437395(CHEMBL2408638)
Affinity DataIC50: 6.5nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437395(CHEMBL2408638)
Affinity DataIC50: 9nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437396(CHEMBL2408651)
Affinity DataIC50: 16nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437396(CHEMBL2408651)
Affinity DataIC50: 17nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437402(CHEMBL2408774)
Affinity DataIC50: 17nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50228407(8-((R)-3-amino-piperidin-1-yl)-3-methyl-7-(3-methy...)
Affinity DataIC50: 40nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437402(CHEMBL2408774)
Affinity DataIC50: 57nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437398(CHEMBL2408646)
Affinity DataIC50: 84nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310584(CHEMBL1078049 | N-(5-Chloro-pyridin-2-yl)-2-(4-{N-...)
Affinity DataIC50: 88nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310577(CHEMBL1079529 | CHEMBL1077867 | (R)-2-(4-(1-(2-(4-...)
Affinity DataIC50: 90nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310577(CHEMBL1079529 | CHEMBL1077867 | (R)-2-(4-(1-(2-(4-...)
Affinity DataIC50: 98nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310582(CHEMBL1079156 | CHEMBL1079889 | (R)-N-(5-cyanopyri...)
Affinity DataIC50: 110nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310583(CHEMBL1079157 | CHEMBL1079890 | (R)-N-(2-chloropyr...)
Affinity DataIC50: 119nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310584(CHEMBL1078049 | N-(5-Chloro-pyridin-2-yl)-2-(4-{N-...)
Affinity DataIC50: 120nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310583(CHEMBL1079157 | CHEMBL1079890 | (R)-N-(2-chloropyr...)
Affinity DataIC50: 124nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437401(CHEMBL2408642)
Affinity DataIC50: 130nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310582(CHEMBL1079156 | CHEMBL1079889 | (R)-N-(5-cyanopyri...)
Affinity DataIC50: 130nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50150851(2-((R)-2-Amino-3-methyl-pentanoyl)-3,4-dihydro-2H-...)
Affinity DataIC50: 130nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IV of porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310580((R)-N-(benzo[d]thiazol-2-yl)-2-(4-(1-(2-(4-cyanoth...)
Affinity DataIC50: 134nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310581((R)-2-(4-(1-(2-(4-cyanothiazolidin-3-yl)-2-oxoethy...)
Affinity DataIC50: 143nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437399(CHEMBL2408644)
Affinity DataIC50: 145nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437398(CHEMBL2408646)
Affinity DataIC50: 147nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310579((R)-2-(4-(1-(2-(4-cyanothiazolidin-3-yl)-2-oxoethy...)
Affinity DataIC50: 185nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310576((R)-N-(4-cyanophenyl)-2-(4-(1-(2-(4-cyanothiazolid...)
Affinity DataIC50: 200nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437401(CHEMBL2408642)
Affinity DataIC50: 210nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310568(CHEMBL1081168 | CHEMBL1077662 | (R)-2-(4-(1-(2-(4-...)
Affinity DataIC50: 217nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310575((R)-2-(4-(1-(2-(4-cyanothiazolidin-3-yl)-2-oxoethy...)
Affinity DataIC50: 222nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310578((R)-N-(5-bromothiazol-2-yl)-2-(4-(1-(2-(4-cyanothi...)
Affinity DataIC50: 226nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310568(CHEMBL1081168 | CHEMBL1077662 | (R)-2-(4-(1-(2-(4-...)
Affinity DataIC50: 236nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310574((R)-N-(benzo[d][1,3]dioxol-5-yl)-2-(4-(1-(2-(4-cya...)
Affinity DataIC50: 240nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310571((R)-N-(4-chlorophenyl)-2-(4-(1-(2-(4-cyanothiazoli...)
Affinity DataIC50: 258nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437400(CHEMBL2408643)
Affinity DataIC50: 275nMAssay Description:Inhibition of porcine DPP4 using H-Gly-Pro-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310573((R)-2-(4-(1-(2-(4-cyanothiazolidin-3-yl)-2-oxoethy...)
Affinity DataIC50: 308nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50437399(CHEMBL2408644)
Affinity DataIC50: 334nMAssay Description:Inhibition of porcine DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310572((R)-N-(3-chloro-4-fluorophenyl)-2-(4-(1-(2-(4-cyan...)
Affinity DataIC50: 359nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM11559(N-({(2S)-1-[(3R)-3-amino-4-(2-fluorophenyl)butanoy...)
Affinity DataIC50: 410nMpH: 7.4 T: 2°CAssay Description:The DPP4 activity resulted in the formation of the fluorescent product amidomethylcoumarin (AMC), which was monitored by excitation at 370 nm and mea...More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/17/2006
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310569((R)-2-(4-(1-(2-(4-cyanothiazolidin-3-yl)-2-oxoethy...)
Affinity DataIC50: 415nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50049394(cirsimartin | CHEMBL348436 | cid_188323 | 5-Hydrox...)
Affinity DataIC50: 430nMAssay Description:Inhibition of porcine DPP4 after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50150858(6-{2-[2-((S)-5-Cyano-4,5-dihydro-pyrazol-1-yl)-2-o...)
Affinity DataIC50: 440nMAssay Description:Inhibitory concentration against dipeptidyl peptidase IV of porcine kidneyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310565((R)-2-(4-(1-(2-(4-cyanothiazolidin-3-yl)-2-oxoethy...)
Affinity DataIC50: 468nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310589((R)-N-(5-chloropyridin-2-yl)-2-(4-(1-(2-(4-cyanoth...)
Affinity DataIC50: 490nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50150854(6-(2-(2-(5-cyano-4,5-dihydro-1H-pyrazol-1-yl)-2-ox...)
Affinity DataIC50: 490nMAssay Description:Inhibition of pig kidney DPP4More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50049395(5,7-dihydroxy-2-(4-hydroxyphenyl)-6-methoxy-4H-chr...)
Affinity DataIC50: 490nMAssay Description:Inhibition of porcine DPP4 after 30 mins by luminescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Pig)
Santhera Pharmaceuticals

LigandPNGBDBM50310567((R)-2-(4-(1-(2-(4-cyanothiazolidin-3-yl)-2-oxoethy...)
Affinity DataIC50: 506nMAssay Description:Inhibition of pig kidney DPP4 by spectrophotometric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
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