Compile Data Set for Download or QSAR
Report error Found 1512 for UniProtKB: P21396
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19164(cid_379337 | CHEMBL421088 | 3-phenyl-5H-indeno[1,2...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19166(3-phenyl-5H-pyridazino[4,3-b]indole | Aza-heterocy...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19167(3-(phenoxymethyl)-5H-indeno[1,2-c]pyridazin-5-one ...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19168(3-(4-fluorophenoxymethyl)-5H-indeno[1,2-c]pyridazi...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19169(3-[4-(trifluoromethyl)phenoxymethyl]-5H-indeno[1,2...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19173(2-phenyl-2H,3H,5H-indeno[1,2-c]pyridazine-3,5-dion...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19177(2-(3-nitrophenyl)-9H-indeno[2,1-d]pyrimidin-9-one ...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19181(3-phenyl-4aH,9H,9aH-indeno[1,2-e][1,2,4]triazin-9-...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19182(3-(3-aminophenyl)-4aH,9H,9aH-indeno[1,2-e][1,2,4]t...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19183(3-(3-nitrophenyl)-4aH,9H,9aH-indeno[1,2-e][1,2,4]t...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM19184(3-(3-nitrophenyl)-4aH,5H,9bH-indeno[2,1-e][1,2,4]t...)
Affinity DatapH: 7.4 T: 2°CAssay Description:A continuous spectrophotometric assay that monitors the rate of oxidation of the nonselective MAO substrate kynuramine into 4-hydroxyquinoline was us...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/24/2007
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50516235(CHEMBL4563408)
Affinity DataEC50: >1.00E+4nMAssay Description:Displacement of [3H]Ro41-1049 from rat brain MAOA after 60 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/22/2021
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM174835(US9114126, 2027BA1)
Affinity DataIC50: 0.220nMAssay Description:Inhibition of rat MAO-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/21/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 0.420nMAssay Description:Inhibition of MAO-A in Sprague-Dawley rat brain homogenate using kynuramine as substrate preincubated for 10 mins measured by fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 0.700nMAssay Description:In vitro Inhibitory activity of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT (serotonin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50381960(CHEMBL2022927)
Affinity DataIC50: 0.790nMAssay Description:Inhibition of mitochondrial MAO-A in rat liver homogenates using [14C]-(5-hydroxy-triptamine) as substrate preincubated for 30 mins by liquid scintil...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50049682(2-Methoxy-6-(5-methyl-[1,3,4]oxadiazol-2-yl)-10,10...)
Affinity DataIC50: 1nMAssay Description:Inhibitory concentration against rat brain mitochondrial monoamine oxidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM10989((1R)-N-(prop-2-yn-1-yl)-2,3-dihydro-1H-inden-1-ami...)
Affinity DataIC50: 1nMAssay Description:Inhibition of rat brain MAO-A in nuclei-free homogenates using [14C]hydroxytryptamine substrate after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50367064(CHEMBL1204338)
Affinity DataIC50: 1nMAssay Description:Compound was tested in vitro for inhibition of rat brain mitochondrial monoamine oxidase A.More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/12/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50179019(3-benzyl-N-(2-morpholinoethyl)quinoxalin-2-amine |...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50075965(CHEMBL3415613)
Affinity DataIC50: 1.5nMAssay Description:Inhibition of rat brain MAO-A in nuclei-free homogenates using [14C]hydroxytryptamine substrate after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50179021(3-(4-chlorobenzyl)-N-(2-morpholinoethyl)quinoxalin...)
Affinity DataIC50: 1.70nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50049666(5-(10,10-Dioxo-10H-10lambda*6*-phenoxathiin-2-yl)-...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against rat brain mitochondrial monoamine oxidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50049671(2-Methyl-6-(5-methyl-[1,3,4]oxadiazol-2-yl)-10,10-...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against rat brain mitochondrial monoamine oxidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50049701(3-(5-Methyl-[1,3,4]oxadiazol-2-yl)-10,10-dioxo-10H...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against rat brain mitochondrial monoamine oxidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50049704(2-(5-Methyl-[1,3,4]oxadiazol-2-yl)-10,11-dioxa-dib...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against Monoamine oxidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50049703(6-(2-Methyl-2H-tetrazol-5-yl)-10,10-dioxo-2-propox...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against rat brain mitochondrial monoamine oxidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50049686(2-Methoxy-6-(2-methyl-2H-tetrazol-5-yl)-10,10-diox...)
Affinity DataIC50: 2nMAssay Description:Inhibitory concentration against rat brain mitochondrial monoamine oxidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50075969(CHEMBL3415617)
Affinity DataIC50: 2nMAssay Description:Inhibition of rat brain MAO-A in nuclei-free homogenates using [14C]hydroxytryptamine substrate after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50059304(9,10,10-Trioxo-7-propoxy-9,10-dihydro-10lambda*6*-...)
Affinity DataIC50: 2nMAssay Description:Inhibition of Monoamine oxidase A (MAO A) in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50179017(1-(3-(4-chlorobenzyl)quinoxalin-2-yl)hydrazine | C...)
Affinity DataIC50: 2.10nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50608295(CHEMBL5271774)
Affinity DataIC50: 2.30nMAssay Description:Inhibition of rat brain synaptosome MAO-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50088564(CHEMBL3577041)
Affinity DataIC50: 2.80nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 2.90nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using serotonin as substrate preincubated with enzyme for 60 mins prior to substrate additionMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/7/2016
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50179020(2-(3-benzylquinoxalin-2-ylamino)ethanol | CHEMBL20...)
Affinity DataIC50: 3.70nMAssay Description:Inhibition of rat liver mitochondria MAOAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM15579(US8633208, Deprenyl | CHEMBL972 | L-Deprenyl | SLG...)
Affinity DataIC50: 3.90nMAssay Description:Inhibition of rat brain synaptosome MAO-AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/19/2024
Entry Details
PubMed
LigandPNGBDBM50224952(CHEMBL441014)
Affinity DataIC50: 4nMAssay Description:In vitro inhibition of Monoamine oxidase at rat hyphalamic mitochondrial 5-HT by displacing 2.5 uM of [14C]5-HT.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/8/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM15581(US8633208, Clorgyline | [3-(2,4-dichlorophenoxy)pr...)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of MAO-A in rat liver mitochondria using p-tyramine as substrate preincubated for 10 mins followed by substrate addition measured after 30...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/8/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50049687(2-Isopropyl-6-(2-methyl-2H-tetrazol-5-yl)-10,10-di...)
Affinity DataIC50: 5nMAssay Description:Inhibitory concentration against rat brain mitochondrial monoamine oxidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50282522(4-Chloro-benzenesulfonic acid 3,4-dimethyl-2-oxo-2...)
Affinity DataIC50: 5nMAssay Description:In vitro inhibitory against monoamine oxidase A (MAO-A) in rat brain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50288969(Brofaromine | 4-(7-Bromo-5-methoxy-benzofuran-2-yl...)
Affinity DataIC50: 5nMAssay Description:In vitro inhibitory against monoamine oxidase A (MAO-A) in rat brain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

LigandPNGBDBM50225462(CHEMBL554775)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against rat brain mitochondrial Monoamine oxidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/14/2018
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of rat liver mitochondrial MAO-A using [14C]-5-hydroxytryptamine after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of rat liver mitochondrial MAOA using [14C]-5-HT as substrate preincubated for 30 mins followed by substrate addition measured after 10 mi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50359391(CHEMBL1929421)
Affinity DataIC50: 5.20nMAssay Description:Inhibition of rat liver mitochondrial MAOA [14C]-5-HT as substrate preincubated for 30 mins followed by substrate addition by liquid scintillation co...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/21/2021
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50064684(3-Ethyl-phenoxathiine 10,10-dioxide | CHEMBL67629)
Affinity DataIC50: 6nMAssay Description:Inhibitory concentration against monoamine oxidase A.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50075994(CHEMBL3415785)
Affinity DataIC50: 6nMAssay Description:Inhibition of rat brain MAO-A in nuclei-free homogenates using [14C]hydroxytryptamine substrate after 20 mins by liquid scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/24/2016
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50282520(4-Bromo-benzenesulfonic acid 3,4-dimethyl-2-oxo-2H...)
Affinity DataIC50: 6nMAssay Description:In vitro inhibitory against monoamine oxidase A (MAO-A) in rat brain homogenate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2012
Entry Details Article

TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50059303(7-Isopropyl-9,10,10-trioxo-9,10-dihydro-10lambda*6...)
Affinity DataIC50: 6nMAssay Description:Inhibition of Monoamine oxidase A (MAO A) in rat brain.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/4/2012
Entry Details Article
PubMed
TargetAmine oxidase [flavin-containing] A(Rat)
University of Bari

LigandPNGBDBM50359396(CHEMBL1929420 | US8999994, 5)
Affinity DataIC50: 6.70nMAssay Description:Inhibition of rat liver mitochondrial MAO-A using [14C]-5-hydroxytryptamine after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
Displayed 1 to 50 (of 1512 total ) | Next | Last >>
Jump to: