TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 3.43E+4nMAssay Description:Agonist activity at cyclothiazide-desensitized rat recombinant flop iGluR4c expressed in Xenopus laevis oocytes by two electrode voltage-clamp electr...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR4 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR4 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 870nMAssay Description:Inhibition of rat recombinant GluR4 in cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Agonist activity at rat recombinant GluA4i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 1.30E+6nMAssay Description:Agonist activity at rat recombinant GluA4i expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR4 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 3.00E+4nMAssay Description:Activity at rat cloned iGluR4 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 1.70E+4nMAssay Description:Activity at rat cloned iGluR4 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: >1.00E+6nMAssay Description:Activity at rat cloned iGluR4 expressed in human HEK293 cells by calcium imaging assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 2.00E+4nMAssay Description:Agonist activity at rat recombinant GluA4 receptor flip isoform expressed in HEK293 cells assessed as effect on cyclothiazide-induced calcium flux by...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 4.70E+4nMAssay Description:Agonist activity at rat recombinant GluA4 receptor flip isoform expressed in HEK293 cells assessed as effect on cyclothiazide-induced calcium flux by...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 1.60E+4nMAssay Description:Agonist activity at rat recombinant GluA4 receptor flip isoform expressed in HEK293 cells assessed as effect on cyclothiazide-induced calcium flux by...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 1.29E+5nMAssay Description:Agonist activity at recombinant rat GluA4 receptor flip isoform expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 1.96E+4nMAssay Description:Agonist activity at recombinant rat GluA4 receptor flip isoform expressed in Xenopus laevis oocytes by two-electrode voltage clamp assayMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 1.19E+4nMAssay Description:Agonist activity at cyclothiazide-desensitized rat recombinant flip iGluR4 expressed in Xenopus laevis oocytes by two electrode voltage-clamp electro...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 2.42E+4nMAssay Description:Agonist activity at cyclothiazide-desensitized rat recombinant flip iGluR4 expressed in Xenopus laevis oocytes by two electrode voltage-clamp electro...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 3.43E+4nMAssay Description:The potency at recombinant rat AMPA-R was measured on GluR4 receptor expressed in Xenopus Laevis oocytesMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 3.80E+4nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 4 (GluR4) using rat cort...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 1.30E+6nMAssay Description:Effective concentration of compound was determined for electrophysiological properties on Ionotropic glutamate receptor AMPA 4 (GluR4) using rat cort...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 4.70E+4nMAssay Description:Agonist activity at rat recombinant GluR4 flip isomer expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4/AM assa...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 3.50E+4nMAssay Description:Agonist activity at rat recombinant GluR4 flip isomer expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4/AM assa...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 2.00E+4nMAssay Description:Agonist activity at rat recombinant GluR4 flip isomer expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4/AM assa...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 6.70E+3nMAssay Description:Agonist activity at rat recombinant GluR4 flip isomer expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4/AM assa...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataEC50: 9.00E+4nMAssay Description:Agonist activity at cyclothiazide-desensitized rat recombinant flip iGluR4 expressed in Xenopus laevis oocytes by two electrode voltage-clamp electro...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataIC50: 320nMAssay Description:Inhibition of rat recombinant GluA4 receptor expressed in Xenopus oocytes assessed as inhibition of 300 uM kainate-induced currentMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Ligand Info
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat homomeric recombinant GluR4 expressed in HEK293 cells assessed as inhibition of intracellular calcium concentration by FLI...More data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataKi: 0.00270nMAssay Description:Displacement of [3H]AMPA from rat recombinant GluR4 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataKi: 0.0400nMAssay Description:Displacement of [3H]AMPA from rat recombinant GluR4 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataKi: 0.0440nMAssay Description:Displacement of [3H]AMPA from rat recombinant GluR4 expressed in Sf9 cellsMore data for this Ligand-Target Pair
TargetGlutamate receptor 4(Rat)
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
European Research Centre For Drug Discovery and Development (Natsyndrugs)
Curated by ChEMBL
Affinity DataKi: 0.200nMAssay Description:Displacement of [3H]AMPA from rat recombinant GluR4 expressed in Sf9 cellsMore data for this Ligand-Target Pair








































