Compile Data Set for Download or QSAR
Report error Found 494 for UniProtKB: P18090
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337291(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337292(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  550nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337293(1-(4-fluorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy...)
Affinity DataEC50:  6.30E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337294(1-(2,6-dichlorobenzyl)-3-(3-(2-(2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337295(1-benzhydryl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo...)
Affinity DataEC50:  8.89E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337296(1-(biphenyl-2-yl)-3-(3-(2-(2-hydroxy-2-(8-hydroxy-...)
Affinity DataEC50:  5.77E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337297(1-Adamantan-1-ylmethyl-3-(3-{2-[2-hydroxy-2-(8-hyd...)
Affinity DataEC50:  296nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337298(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50:  1.00E+4nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50318159(CHEMBL1095777 | 8-Hydroxy-5-[(R)-1-hydroxy-2-(5,6-...)
Affinity DataEC50:  2.31E+3nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337299(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337300(1-benzyl-3-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50337301(1-(3-(2-(2-hydroxy-2-(8-hydroxy-2-oxo-1,2-dihydroq...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at beta1 adrenoceptor in rat left atria assessed as induction of ionotropic effectMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2011
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.316nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor S190A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat wild type beta-1 adrenergic receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0794nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor Y356F mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
TargetBeta-1 adrenergic receptor(Rat)
RhôNe-Poulenc Rorer

Curated by ChEMBL
LigandPNGBDBM50422862(125I-CYP | CHEMBL210309)
Affinity DataKd:  0.0631nMAssay Description:Antagonist activity at rat beta-1 adrenergic receptor W134A mutant expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/23/2013
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKd:  1nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to membrane preparation from rat lung reticulocyte pretreated with alkylating beta-blocker...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKd:  2nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding sites on beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating be...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating beta-blo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226719(CHEMBL156754)
Affinity DataKd:  1.20nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226717(CHEMBL157881 | (+/-)-Pindobind)
Affinity DataKd:  2.40nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226718(CHEMBL156628)
Affinity DataKd:  1.40nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat lung reticulocytes pretreated with alkylating beta-bloc...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50226716(CHEMBL348176)
Affinity DataKd:  1.60nMAssay Description:Binding affinity against the [3H]dihydroalprenolol binding to beta adrenergic receptor of rat heart reticulocytes pretreated with alkylating beta-blo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2018
Entry Details Article
PubMed
LigandPNGBDBM50029050(4-[(1R)-1-hydroxy-2-(methylamino)ethyl]benzene-1,2...)
Affinity DataEC50:  230nMAssay Description:Agonistic potency at beta adrenergic receptor for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMedPDB3D3D Structure (crystal)
LigandPNGBDBM50019057((+/-)4-Fluoro-5-(1-hydroxy-2-methylamino-ethyl)-be...)
Affinity DataEC50: >1.50E+3nMAssay Description:Agonistic potency at beta adrenergic receptor for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
LigandPNGBDBM50019059(3-Fluoro-4-(1-hydroxy-2-methylamino-ethyl)-benzene...)
Affinity DataEC50:  40nMAssay Description:Agonistic potency at beta adrenergic receptor for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/16/2012
Entry Details Article
PubMed
LigandPNGBDBM50007477(CHEMBL10453 | 4-(3-tert-Butylamino-2-hydroxy-propo...)
Affinity DataEC50:  9.20nMAssay Description:Beta adrenergic receptor agonistic activity for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50007476(CHEMBL266619 | 4-(3-tert-Butylamino-2-hydroxy-prop...)
Affinity DataEC50:  8.20nMAssay Description:Beta adrenergic receptor agonistic activity for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM25392(Isoproterenol,(+) | CHEMBL434 | 4-[1-hydroxy-2-(pr...)
Affinity DataEC50:  7nMAssay Description:Beta adrenergic receptor agonistic activity for the stimulation of accumulation of cyclic AMP in cultured C6 glioma cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  19.8nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat lung tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  391nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat heart tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  42.4nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat heart tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  2.80nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-6 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  125nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat lung tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  4.80nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-5 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  42nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat heart tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  2.10nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]Dihydroalprenolol in rat heart tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  3.20nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]Dihydroalprenolol in rat heart tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  3nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat heart tissue at 1*10e-5 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  20nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat lung tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  1.60nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  2.5nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  2.5nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat lung tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  391nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat heart tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  31.2nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat heart tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  3.20nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]Dihydroalprenolol in rat heart tissue at 1*10e-7 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225368(CHEMBL47370)
Affinity DataKd:  2.80nMAssay Description:Dissociation constant against beta adrenergic receptor using [3H]dihydroalprenolol in rat heart tissue at 1*10e-6 concentrationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
LigandPNGBDBM50225367(Bromoacetyl Alprenolol Menthane)
Affinity DataKd:  29nMAssay Description:Equilibrium dissociation constant (KD) against beta adrenergic receptor of rat lung tissueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/13/2018
Entry Details Article
PubMed
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