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Report error Found 97 for UniProtKB: P17538
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50133629(2,3-Dioxo-2,3-dihydro-indole-1-carboxylic acid ben...)
Affinity DataKoff:  253s-1Assay Description:Rate constant against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50133629(2,3-Dioxo-2,3-dihydro-indole-1-carboxylic acid ben...)
Affinity DataKon:  0.0000400M-1s-1Assay Description:Rate constant against alpha-chymotrypsin from time dependent inhibition and reactivation dataMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50133629(2,3-Dioxo-2,3-dihydro-indole-1-carboxylic acid ben...)
Affinity DataKoff:  7.60s-1Assay Description:Rate constant against Alpha-chymotrypsin from time dependent inhibition and reactivation dataMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50133629(2,3-Dioxo-2,3-dihydro-indole-1-carboxylic acid ben...)
Affinity DataKon:  0.000948M-1s-1Assay Description:Rate constant against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/19/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50073139([2,2-dimethyl-3-(N-(4-cyanobenzoyl)aminoi)-5-pheny...)
Affinity DataIC50: 2.10nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075109(1,1-dimethyl-2-phenylcarboxamidoheptanoic anhydrid...)
Affinity DataIC50: 5.30nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50142284(2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-...)
Affinity DataIC50: 10nMAssay Description:Inhibitory activity against chymotrypsinogen; Range 1-10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075107(1,1-dimethyl-4-phenyl-2-propylcarboxamidopentanoic...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075107(1,1-dimethyl-4-phenyl-2-propylcarboxamidopentanoic...)
Affinity DataIC50: 12nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075110(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-phenyl...)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075106(1,1-dimethyl-4-phenyl-2-phenylcarboxamidopentanoic...)
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075106(1,1-dimethyl-4-phenyl-2-phenylcarboxamidopentanoic...)
Affinity DataIC50: 18nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075114(1,1-dimethyl-2-phenylcarboxamidooctanoic anhydride...)
Affinity DataIC50: 31nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075104(1,1-dimethyl-2-phenylcarboxamidononanoic anhydride...)
Affinity DataIC50: 44nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075118(1,1-dimethyl-2-phenylcarboxamidohexanoic anhydride...)
Affinity DataIC50: 49nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289952(6-Dimethylamino-5-methyl-2-(1-phenyl-ethylamino)-b...)
Affinity DataIC50: 65nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075105(1,1-dimethyl-2-phenylcarboxamidopentanoic anhydrid...)
Affinity DataIC50: 72nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289954(5-Methyl-2-(1-phenyl-ethylamino)-benzo[d][1,3]oxaz...)
Affinity DataIC50: 88nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289953(2-[1-(4-Bromo-phenyl)-ethylamino]-5-methyl-benzo[d...)
Affinity DataIC50: 140nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075113(1,1-dimethyl-2-phenylcarboxamidopropanoic anhydrid...)
Affinity DataIC50: 140nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289955(5-Methyl-2-(1-phenyl-ethylamino)-benzo[d][1,3]oxaz...)
Affinity DataIC50: 180nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075116(2-(4-cyanophenylcarboxamido)-1,1-dimethyl-2-(2-met...)
Affinity DataIC50: 190nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075111(2-(4-cyanophenylcarboxamido)-2-cyclohex-3-enyl-1,1...)
Affinity DataIC50: 220nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075108(2-(2-chlorophenyl)-2-(4-cyanophenylcarboxamido)-1,...)
Affinity DataIC50: 250nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070440({(S)-1-[(S)-1-(1-Benzylcarbamoyl-4-oxo-azetidin-2-...)
Affinity DataIC50: 800nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075112(1,1-dimethyl-2-propylcarboxamidooctanoic anhydride...)
Affinity DataIC50: 810nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070444((3R,4S)-3-Methyl-2-oxo-4-(pyridin-2-ylmethylsulfan...)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50063719(2-Isopropylamino-5-methyl-benzo[d][1,3]oxazin-4-on...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289948(2-Dimethylamino-N-[5-methyl-4-oxo-2-(1-phenyl-ethy...)
Affinity DataIC50: 2.60E+3nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289950(4-Methoxy-N-[5-methyl-4-oxo-2-(1-phenyl-ethylamino...)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50139465(((S)-1-Mercaptomethyl-2-phenyl-ethyl)-carbamic aci...)
Affinity DataIC50: 3.80E+3nMAssay Description:Inhibitory activity against chymotrypsinogen in the presence of Zn(II) (500 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075117(2-phenylcarboxamidopropanoic anhydride | CHEMBL134...)
Affinity DataIC50: 4.60E+3nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50139460(((R)-1-Mercaptomethyl-2-phenyl-ethyl)-carbamic aci...)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibitory activity against chymotrypsinogen in the presence of Zn(II) (500 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50139463((S)-2-((S)-1-Mercaptomethyl-2-phenyl-ethylcarbamoy...)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibitory activity against chymotrypsinogen in the presence of Zn(II) (500 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070442({(S)-1-[(S)-1-(1-Benzylcarbamoyl-4-oxo-azetidin-2-...)
Affinity DataIC50: 8.30E+3nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50142276(2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against chymotrypsinogen; Range 1-10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
LigandPNGBDBM50502656(CHEMBL4455694)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human chymotrypsin using Suc-AAPF-MCA as substrate by fluorescence based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/17/2021
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075115(4-phenyl-2-phenylcarboxamidopentanoic anhydride | ...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against bovine pancreatic alpha-chymotrypsin (alpha-CT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50142275(2-Ethyl-1,1-dioxo-1,2,3,4,6,7-hexahydro-5,8-dioxa-...)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibitory activity against chymotrypsinogen; Range 1-10 uMMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/11/2012
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50139462(N-((S)-1-Mercaptomethyl-2-phenyl-ethyl)-benzamide ...)
Affinity DataIC50: 2.30E+4nMAssay Description:Inhibitory activity against chymotrypsinogen in the presence of Zn(II) (500 uM)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50289951([5-Methyl-4-oxo-2-(1-phenyl-ethylamino)-4H-benzo[d...)
Affinity DataIC50: 4.20E+4nMAssay Description:Inhibitory concentration against human chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070436(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070443(((S)-2,2-Dimethyl-1-{(S)-3-methyl-1-[4-oxo-1-((R)-...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070449(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070441(2-Oxo-4-(pyridin-3-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070448(2-Benzylsulfanyl-4-oxo-azetidine-1-carboxylic acid...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070445(2-Oxo-4-(pyridin-2-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070437(2-Oxo-4-phenethylsulfanyl-azetidine-1-carboxylic a...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070439(2-{(S)-2-[(S)-2-(3,3-Dimethyl-butyrylamino)-3,3-di...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetChymotrypsinogen B(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50070447(2-Oxo-4-(pyridin-4-ylmethylsulfanyl)-azetidine-1-c...)
Affinity DataIC50: 7.50E+4nMAssay Description:Inhibitory activity against alpha-chymotrypsinMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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