Compile Data Set for Download or QSAR
Report error Found 4 for UniProtKB: P15389
LigandPNGBDBM50344821(10-hydroxymethyl-5-imino-(2S)-12,13-dioxa-4,6-diaz...)
Affinity DataKd:  1.80nMAssay Description:Displacement of [3H]saxitoxin from NaV in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetSodium channel protein type 5 subunit alpha(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50357365(CHEMBL1917113)
Affinity DataIC50: 2.37E+5nMAssay Description:Inhibition of rat Nav1.5 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50242400(CCNCSSKWCRDHSRCC | CHEMBL525818)
Affinity DataIC50: 2.87E+5nMAssay Description:Inhibition of rat Nav1.5 channel expressed in Xenopus oocytes by whole cell voltage clamp techniqueMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetSodium channel protein type 5 subunit alpha(Rat)
Monash University

Curated by ChEMBL
LigandPNGBDBM50357366(CHEMBL1917112)
Affinity DataIC50: 8.71E+5nMAssay Description:Inhibition of rat Nav1.5 expressed in Xenopus oocytes assessed as blockage of voltage-activated sodium current at holding potential of -100 mV by two...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed