Compile Data Set for Download or QSAR
Report error Found 129 of affinity data for UniProtKB/TrEMBL: P15085
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50478894(Anabaenopeptin G)
Affinity DataIC50: 2nMAssay Description:Inhibition of carboxypeptidase A (unknown origin) assessed as reduction in hydrolysis of hippuryl-L-phenylalanine using hippuryl-L-phenylalanine as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50478891(Anabaenopeptin I)
Affinity DataIC50: 6.84nMAssay Description:Inhibition of carboxypeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50478894(Anabaenopeptin G)
Affinity DataIC50: 7nMAssay Description:Inhibition of carboxypeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50478895(Anabaenopeptin J)
Affinity DataIC50: 9.57nMAssay Description:Inhibition of carboxypeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50478892(Anabaenopeptin T)
Affinity DataIC50: 25.4nMAssay Description:Inhibition of carboxypeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50480481(Anabaenopeptin 915)
Affinity DataIC50: 130nMAssay Description:Inhibition of carboxypeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50121929(2-benzylbutanedioic acid | 2-benzylsuccinic acid |...)
Affinity DataIC50: 400nMAssay Description:In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50089687(Anabaenopeptin F)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of CPA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2016
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50135934(3-(6-Amino-pyridin-3-yl)-2-[1-(3-methyl-butyl)-1H-...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50135934(3-(6-Amino-pyridin-3-yl)-2-[1-(3-methyl-butyl)-1H-...)
Affinity DataIC50: 1.40E+3nMAssay Description:In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50100009(2-(1H-Imidazol-4-yl)-3-phenyl-propionic acid | 2-(...)
Affinity DataIC50: 1.70E+3nMAssay Description:In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50478893(Anabaenopeptin H)
Affinity DataIC50: 3.68E+3nMAssay Description:Inhibition of carboxypeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50478893(Anabaenopeptin H)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of carboxypeptidase A (unknown origin) assessed as reduction in hydrolysis of hippuryl-L-phenylalanine using hippuryl-L-phenylalanine as s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50089688(ANABAENOPEPTIN B)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of CPA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2016
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50135938(3-(6-Amino-pyridin-3-yl)-2-(1-isopropyl-1H-imidazo...)
Affinity DataIC50: 6.40E+3nMAssay Description:In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50558425(CHEMBL4746522)
Affinity DataIC50: 6.74E+3nMAssay Description:Inhibition of carboxypeptidase A (unknown origin) assessed as reduction in degradation of N-(4-methoxyphenylazoformyl)-Phe-OH using N-(4-methoxypheny...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50478893(Anabaenopeptin H)
Affinity DataIC50: 1.02E+4nMAssay Description:Inhibition of carboxypeptidase A (unknown origin) assessed as reduction in degradation of N-(4-methoxyphenylazoformyl)-Phe-OH using N-(4-methoxypheny...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50558424(Anabaenopeptin 908)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of carboxypeptidase A (unknown origin) assessed as reduction in degradation of N-(4-methoxyphenylazoformyl)-Phe-OH using N-(4-methoxypheny...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50558424(Anabaenopeptin 908)
Affinity DataIC50: 2.20E+4nMAssay Description:Inhibition of carboxypeptidase A (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50089687(Anabaenopeptin F)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of carboxypeptidase A (unknown origin) assessed as reduction in degradation of N-(4-methoxyphenylazoformyl)-Phe-OH using N-(4-methoxypheny...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50089688(ANABAENOPEPTIN B)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of carboxypeptidase A (unknown origin) assessed as reduction in degradation of N-(4-methoxyphenylazoformyl)-Phe-OH using N-(4-methoxypheny...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50135933(3-(6-Amino-pyridin-3-yl)-2-(1H-imidazol-4-yl)-prop...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50135933(3-(6-Amino-pyridin-3-yl)-2-(1H-imidazol-4-yl)-prop...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50135939(3-(4,4-Diamino-but-3-enylsulfanyl)-2-mercaptomethy...)
Affinity DataIC50: 5.00E+4nMAssay Description:In vitro inhibition of Carboxypeptidase A (CPA) was determined by clot lysis assay using human plasmaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50089686(CHEMBL3577334)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of CPA (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/9/2016
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530229(CHEMBL4460840)
Affinity DataKi:  0.0400nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530229(CHEMBL4460840)
Affinity DataKi:  0.0400nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530230(CHEMBL4445882)
Affinity DataKi:  0.0700nMAssay Description:Inhibition of human CPA1 using AAFP as substrate measured at pre-steady state by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530230(CHEMBL4445882)
Affinity DataKi:  0.0700nMAssay Description:Inhibition of human CPA1 using AAFP as substrate measured at pre-steady state by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530235(CHEMBL4436298)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530235(CHEMBL4436298)
Affinity DataKi:  0.0800nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530231(CHEMBL4528407)
Affinity DataKi:  0.0870nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530231(CHEMBL4528407)
Affinity DataKi:  0.0870nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530230(CHEMBL4445882)
Affinity DataKi:  0.0890nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530230(CHEMBL4445882)
Affinity DataKi:  0.0890nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530228(CHEMBL4483485)
Affinity DataKi:  0.107nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530228(CHEMBL4483485)
Affinity DataKi:  0.107nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530227(CHEMBL4454162)
Affinity DataKi:  0.129nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530227(CHEMBL4454162)
Affinity DataKi:  0.129nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530231(CHEMBL4528407)
Affinity DataKi:  0.140nMAssay Description:Inhibition of human CPA1 using AAFP as substrate measured at pre-steady state by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530231(CHEMBL4528407)
Affinity DataKi:  0.140nMAssay Description:Inhibition of human CPA1 using AAFP as substrate measured at pre-steady state by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530227(CHEMBL4454162)
Affinity DataKi:  0.160nMAssay Description:Inhibition of human CPA1 using AAFP as substrate measured at pre-steady state by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530228(CHEMBL4483485)
Affinity DataKi:  0.160nMAssay Description:Inhibition of human CPA1 using AAFP as substrate measured at pre-steady state by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530228(CHEMBL4483485)
Affinity DataKi:  0.160nMAssay Description:Inhibition of human CPA1 using AAFP as substrate measured at pre-steady state by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530227(CHEMBL4454162)
Affinity DataKi:  0.160nMAssay Description:Inhibition of human CPA1 using AAFP as substrate measured at pre-steady state by spectrophotometryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530230(CHEMBL4445882)
Affinity DataKi:  0.240nMAssay Description:Inhibition of human CPA1 using AAFP as substrate assessed as apparent first-order rate constant measured at pre-steady state by measuring Koff/Kon ra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530230(CHEMBL4445882)
Affinity DataKi:  0.240nMAssay Description:Inhibition of human CPA1 using AAFP as substrate assessed as apparent first-order rate constant measured at pre-steady state by measuring Koff/Kon ra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530237(CHEMBL4513310)
Affinity DataKi:  0.300nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530237(CHEMBL4513310)
Affinity DataKi:  0.300nMAssay Description:Inhibition of human CPA1 using AAFP as substrate preincubated for 45 mins to 2 hrs measured at 30 sec intervals for 15 mins by UV/vis-spectrophotomet...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Human)
University of California Santa Cruz

Curated by ChEMBL
LigandPNGBDBM50530231(CHEMBL4528407)
Affinity DataKi:  0.470nMAssay Description:Inhibition of human CPA1 using AAFP as substrate assessed as apparent first-order rate constant measured at pre-steady state by measuring Koff/Kon ra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
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