Compile Data Set for Download or QSAR
Report error Found 62 of affinity data for UniProtKB/TrEMBL: P11416
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526314(CHEMBL4459692 | US10752616, Code No. BHBA-001)
Affinity DataEC50:  26nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  1.5nMAssay Description:Transactivation of mouse Gal4-fused RARalpha-LBD expressed in COS-7 cells after 1 day by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526312(CHEMBL4449668 | US10752616, Code No. BHBA-007)
Affinity DataEC50:  16nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526311(CHEMBL4588745)
Affinity DataEC50:  18nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526316(CHEMBL4531897)
Affinity DataEC50:  61nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526317(CHEMBL4437942)
Affinity DataEC50:  18nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526318(CHEMBL4215742)
Affinity DataEC50:  46nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50048292(6-[4-Methoxy-3-(1-methyl-cyclohexyl)-phenyl]-napht...)
Affinity DataEC50:  9.20nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526320(CHEMBL4448702)
Affinity DataEC50:  600nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526313(CHEMBL4469143 | US10752616, Code No. BHBA-006)
Affinity DataEC50:  89nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526315(CHEMBL4439399 | US10752616, Code No. BHBA-019)
Affinity DataEC50:  19nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064255((2E,4Z,6Z)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataEC50: >1.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526321(CHEMBL4572914)
Affinity DataEC50:  4nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526322(CHEMBL4442948)
Affinity DataEC50:  31nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526319(CHEMBL4517145)
Affinity DataEC50:  60nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526323(CHEMBL4539676)
Affinity DataEC50:  240nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  1.20nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526325(CHEMBL4438880 | US10752616, Code No. BHBA-021)
Affinity DataEC50:  30nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50413272(AC-261066 | CHEMBL198997)
Affinity DataEC50:  70nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526327(CHEMBL4562084 | US10752616, Code No. BHBA-023)
Affinity DataEC50:  114nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526324(CHEMBL4439947)
Affinity DataEC50:  58nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50526326(CHEMBL4590840)
Affinity DataEC50:  594nMAssay Description:Transactivation of GAL4-fused mouse RARalpha-LBD expressed in COS-7 cells after 24 hrs by bright-Glo reagent based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/25/2021
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064250(3,7-dimethyl-8-(1,2,3,4-tetrahydro-1-naphthalenyli...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50052958(4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd:  1.00E+4nMAssay Description:Dissociation constant for binding to Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50052961(4-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-naphthal...)
Affinity DataKd:  4.08E+3nMAssay Description:Dissociation constant for binding to Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50052957(4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd:  1.00E+4nMAssay Description:Dissociation constant for binding to Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  15nMAssay Description:Dissociation constant for binding to Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataKd:  7nMAssay Description:Dissociation constant for binding to Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50052959(4-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd:  1.00E+4nMAssay Description:Dissociation constant for binding to Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50052960(2-(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-naphth...)
Affinity DataKd:  1.00E+3nMAssay Description:Dissociation constant for binding to Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064252((2Z,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataEC50:  51nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064254((2E,4E,6E,8Z)-3,7-Dimethyl-9-(2,6,6-trimethyl-cycl...)
Affinity DataEC50:  18nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  22nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064251((2Z,4E,6E)-8-[3,4-Dihydro-2H-naphthalen-(1E)-ylide...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064253((2E,4Z,6Z)-8-[3,4-Dihydro-2H-naphthalen-(1E)-ylide...)
Affinity DataEC50: >2.00E+3nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataEC50:  33nMAssay Description:Transcriptional activation in CV-1 cells expressing retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataIC50: 5nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataIC50: 6nMAssay Description:Inhibition of binding to retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataIC50: 6nMAssay Description:Inhibition of [3H]ATRA binding to mouse Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50035477((2E,4E,6E)-8-[2-Isopropyl-3-methyl-cyclohex-2-en-(...)
Affinity DataIC50: 8nMAssay Description:Inhibition of [3H]ATRA binding to mouse Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataIC50: 11nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataIC50: 11nMAssay Description:Inhibition of [3H]ATRA binding to mouse Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50031460((2E,4E,6E)-8-[3-Ethyl-2-isopropyl-cyclohex-2-en-(E...)
Affinity DataIC50: 14nMAssay Description:Inhibition of binding to retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataIC50: 31nMAssay Description:Inhibition of [3H]ATRA binding to mouse Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064254((2E,4E,6E,8Z)-3,7-Dimethyl-9-(2,6,6-trimethyl-cycl...)
Affinity DataIC50: 31nMAssay Description:Inhibition of binding to retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50031458((2Z,5E)-7-Methyl-3-[(E)-2-(2,6,6-trimethyl-cyclohe...)
Affinity DataIC50: 31nMAssay Description:Inhibition of murine Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50064250(3,7-dimethyl-8-(1,2,3,4-tetrahydro-1-naphthalenyli...)
Affinity DataIC50: 35nMAssay Description:Inhibition of binding to retinoid A receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50053094((2E,4E,6E)-8-[2,3-Dimethyl-cyclohex-2-en-(E)-ylide...)
Affinity DataIC50: 55nMAssay Description:Inhibition of [3H]ATRA binding to mouse Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50346143(rac-4-[(1E)-3-(7,8-Dihydro-8,8-dimethyl-5-p-tolyln...)
Affinity DataIC50: 400nMAssay Description:Antagonist activity at yeast GAL4 fused mouse RARalpha ligand binding domain expressed in HeLa cells assessed as inhibition of TTNPB-induced receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2011
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Mouse)
King'S College

Curated by ChEMBL
LigandPNGBDBM50053093((2E,4E,6E)-8-Cyclohex-2-en-(E)-ylidene-3,7-dimethy...)
Affinity DataIC50: 600nMAssay Description:Inhibition of [3H]ATRA binding to mouse Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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