Compile Data Set for Download or QSAR
Report error Found 584 for UniProtKB: P10276
LigandPNGBDBM31882(CHEMBL80992 | BMS184394-R)
Affinity DataKd:  1.60E+4nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31884(CHEMBL81273 | BMS184394-S)
Affinity DataKd:  7.50E+3nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31885(CHEMBL82089 | BMS184394)
Affinity DataKd:  7.50E+3nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31886(CHEMBL309282 | CD564)
Affinity DataKd:  118nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31887(Ch 80 | BMS181156)
Affinity DataKd:  0.400nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31888(CD666)
Affinity DataKd:  2.24E+3nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31889(BMS 961 | BMS961 | BMS270394)
Affinity DatapH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31890(BMS270395)
Affinity DatapH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  0.400nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMed
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataKd:  0.300nMpH: 7.9 T: 2°CAssay Description:Recombinant RAR protein expressed in E. coli was used in the direct binding assay. The apparent dissociation constants (Kd) were determined by the ch...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/28/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataKd:  15nMAssay Description:Binding affinity for Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290184(4-(1-Isopropyl-4,4-dimethyl-1,2,3,4-tetrahydro-qui...)
Affinity DataKd:  52nMAssay Description:Binding affinity for Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290177(4-(4,4-Dimethyl-1,2,3,4-tetrahydro-quinolin-6-ylet...)
Affinity DataKd:  5.20E+3nMAssay Description:Binding affinity for Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50032219(4-[(E)-2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2...)
Affinity DataKd:  36nMAssay Description:Binding affinity for Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article
PDB3D3D Structure (crystal)
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290184(4-(1-Isopropyl-4,4-dimethyl-1,2,3,4-tetrahydro-qui...)
Affinity DataEC50:  17nMAssay Description:Transactivation potency for Retinoic acid receptor alpha; Not activeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  350nMAssay Description:Transactivation potency for Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50032219(4-[(E)-2-(5,6,7,8-tetrahydro-5,5,8,8-tetramethyl-2...)
Affinity DataEC50:  30nMAssay Description:Transactivation potency for Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article
PDB3D3D Structure (crystal)
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50290177(4-(4,4-Dimethyl-1,2,3,4-tetrahydro-quinolin-6-ylet...)
Affinity DataEC50:  2.30E+3nMAssay Description:Transactivation potency for Retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50287964((E)-3-Methyl-5-[2-methyl-2-(3,5,5,8,8-pentamethyl-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Compound was tested for binding affinity against retinoic acid receptor using 5 nM of [3H]RA as a radioligand in baculovirus expressed receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075877(4-[5,5-Dimethyl-8-(5-methyl-thiophen-2-yl)-5,6-dih...)
Affinity DataKd:  15nMAssay Description:Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075879(4-(2,2-Dimethyl-4-p-tolyl-2H-1-thia-anthracen-6-yl...)
Affinity DataKd:  5.5nMAssay Description:Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50075878(4-(2,2-Dimethyl-4-p-tolyl-2H-benzo[g]chromen-7-yl)...)
Affinity DataKd:  14nMAssay Description:Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPBMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50052412(4-[(4-Bromo-3-hydroxy-5,5,8,8-tetramethyl-5,6,7,8-...)
Affinity DataKd:  4nMAssay Description:Binding affinity fo retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50120063(2,6-Difluoro-4-[(3-hydroxy-5,5,8,8-tetramethyl-5,6...)
Affinity DataEC50:  112nMAssay Description:Effective concentration for retinoic acid receptor RAR alpha transcriptional activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50052414(4-(1,1,4,4-tetramethyl-1,2,3,4-tetrahydronaphthale...)
Affinity DataKd:  36nMAssay Description:Binding affinity fo retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  240nMAssay Description:Effective concentration for retinoic acid receptor RAR alpha transcriptional activationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50097822(4-{(E)-4-[2-(4-tert-Butyl-phenyl)-6,6-dimethyl-cyc...)
Affinity DataKd:  350nMAssay Description:Ability to inhibit TTNPB-induced transactivation at retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50097823(4-[(E)-4-(6,6-Dimethyl-2-p-tolyl-cyclohex-1-enyl)-...)
Affinity DataKd:  148nMAssay Description:Ability to inhibit TTNPB-induced transactivation at retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  240nMAssay Description:Ability to inhibit TTNPB-induced transactivation at retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50097824(4-[(E)-4-(2,6,6-Trimethyl-cyclohex-1-enyl)-but-3-e...)
Affinity DataKd:  135nMAssay Description:Ability to inhibit TTNPB-induced transactivation at retinoic acid receptor alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50122348((2E,4E)-6-[1-(3,5-Di-tert-butyl-phenyl)-cyclopropy...)
Affinity DataEC50:  733nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50122351((2E,4E)-3-Methyl-6-[1-(5,5,8,8-tetramethyl-5,6,7,8...)
Affinity DataEC50:  59nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31892(CHEMBL705 | 9-cis retinoic acid | alitretinoin | P...)
Affinity DataEC50:  220nMAssay Description:Transcriptional activation in CV-1 cells expressing human Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50029774(4-(5,5-Dimethyl-8-p-tolyl-5,6-dihydro-naphthalen-2...)
Affinity DataKd:  2nMAssay Description:Binding constant for baculovirus-expressed Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM31883(ALL-TRANS-RETINOIC ACID | SMR000058245 | cid_44479...)
Affinity DataEC50:  7nMAssay Description:Transcriptional activation in CV-1 cells expressing Retinoic acid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040010(4-(3-Ethyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro-...)
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040017(4-[1-(3-Ethyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahyd...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration against retinoid receptor isoform (RAR alpha) expressed in CV-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040021(4-[1-(3-Isopropyl-5,5,8,8-tetramethyl-5,6,7,8-tetr...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration against retinoid receptor isoform (RAR alpha) expressed in CV-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50032675(4-[1-(3,5,5,8,8-pentamethyl-5,6,7,8-tetrahydronaph...)
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50032667(4-[(3,5,5,8,8-Pentamethyl-5,6,7,8-tetrahydro-2-nap...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration against retinoid receptor isoform (RAR alpha) expressed in CV-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040015(4-[1-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrah...)
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of [3H]ATRA binding to baculovirus expressed retinoid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040016(4-[1-(3-Chloro-5,5,8,8-tetramethyl-5,6,7,8-tetrahy...)
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040012(4-[1-(3-Bromo-5,5,8,8-tetramethyl-5,6,7,8-tetrahyd...)
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040014(4-[1-(3-Fluoro-5,5,8,8-tetramethyl-5,6,7,8-tetrahy...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration against retinoid receptor isoform (RAR alpha) expressed in CV-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040025(4-(3-Methoxy-5,5,8,8-tetramethyl-5,6,7,8-tetrahydr...)
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040019(4-(5,5,8,8-Tetramethyl-3-propyl-5,6,7,8-tetrahydro...)
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50033079(4-[1-(5,5,8,8-Tetramethyl-5,6,7,8-tetrahydro-napht...)
Affinity DataKd:  944nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040013(4-(3-Chloro-5,5,8,8-tetramethyl-5,6,7,8-tetrahydro...)
Affinity DataKd: >1.00E+3nMAssay Description:Inhibition of [3H]-ATRA binding to baculovirus expressed retinoid receptor RAR alphaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040024(4-[1-(3-Hydroxy-5,5,8,8-tetramethyl-5,6,7,8-tetrah...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration against retinoid receptor isoform (RAR alpha) expressed in CV-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetRetinoic acid receptor alpha(Human)
TBA

Curated by ChEMBL
LigandPNGBDBM50040018(4-(3-Isopropyl-5,5,8,8-tetramethyl-5,6,7,8-tetrahy...)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration against retinoid receptor isoform (RAR alpha) expressed in CV-1 cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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