Compile Data Set for Download or QSAR
Report error Found 12 of affinity data for UniProtKB/TrEMBL: P09482
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50251867(N-(3-((6-chloropyridin-3-yl)methyl)thiazol-2(3H)-y...)
Affinity DataIC50: 500nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50251868({(2Z)-3-[(6-chloropyridin-3-yl)methyl]-1,3-thiazol...)
Affinity DataIC50: 860nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50252631(N-(3-((6-chloropyridin-3-yl)methyl)thiazol-2(3H)-y...)
Affinity DataIC50: 900nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataIC50: 2.60E+3nMAssay Description:Displacement of [3H]nicotine from chick alpha4beta2 nAChRMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50472282(descyanothiacloprid)
Affinity DataKi:  1.20nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM82070(CAS_29790-52-1 | NICOTINE-L (BASE) | Nicotine-D sa...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50078048(1-(6-Chloro-pyridin-3-ylmethyl)-imidazolidin-(2Z)-...)
Affinity DataKi:  2.20nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50487234(CHEMBL1391421)
Affinity DataKi:  60nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50251868({(2Z)-3-[(6-chloropyridin-3-yl)methyl]-1,3-thiazol...)
Affinity DataKi:  240nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50486223(CHEBI:39164 | acetamiprid)
Affinity DataKi:  680nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Chicken)
University of California

Curated by ChEMBL
LigandPNGBDBM50212288((2E)-1-[(6-chloropyridin-3-yl)methyl]-N-nitroimida...)
Affinity DataKi:  970nMAssay Description:Binding affinity to recombinant Gallus gallus (chicken) alpha4beta2 nicotinic acetylcholine receptor assessed as [3H]NIC binding by radioligand bindi...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/30/2020
Entry Details Article
PubMed