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Report error Found 2235 for UniProtKB: P08912
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  210nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  0.512nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50305818(cid_45281794 | CHEMBL593506 | 1-(biphenyl-4-ylmeth...)
Affinity DataEC50: >442nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50305819(cid_45281797 | CHEMBL603445 | 1-(4-(thiophen-3-yl)...)
Affinity DataEC50: >442nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  1.71E+3nMAssay Description:Assay Provider: P. Jeffrey Conn Assay Provider Affiliation: Vanderbilt University Muscarinic acetylcholine receptors are family A GPCRs comprised of...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/5/2011
Entry Details
PCBioAssay
LigandPNGBDBM50229048(CHEMBL349844)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229049(CHEMBL351934)
Affinity DataEC50:  100nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229050(CHEMBL422710)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229054(CHEMBL161748)
Affinity DataEC50:  1.28E+3nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229057(CHEMBL161419)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229059(CHEMBL159708)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229053(CHEMBL161364)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229052(CHEMBL159651)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229051(CHEMBL159935)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229064(CHEMBL159839)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229055(CHEMBL161670)
Affinity DataEC50:  1.46E+3nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50046728(1-Methyl-5-(3-methyl-[1,2,4]oxadiazol-5-yl)-1,2,3,...)
Affinity DataEC50:  32nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229058(CHEMBL161088)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50228565(CHEMBL108557)
Affinity DataKd:  7.00E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228566(CHEMBL2092932)
Affinity DataKd:  3.23E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228567(CHEMBL2092931)
Affinity DataKd:  7.85E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228568(CHEMBL322126)
Affinity DataKd:  1.60E+4nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228569(CHEMBL1788225)
Affinity DataKd:  161nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228570(CHEMBL1788202)
Affinity DataKd:  200nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228571(CHEMBL107456)
Affinity DataKd:  97nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228572(CHEMBL432629)
Affinity DataKd:  110nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228573(CHEMBL106056)
Affinity DataKd:  3.55E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228071(CHEMBL110892)
Affinity DataKd:  1.40E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228574(CHEMBL108582)
Affinity DataKd:  8.30E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228087(CHEMBL323032)
Affinity DataKd:  1.25E+5nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228575(CHEMBL108140)
Affinity DataEC50:  2.80E+3nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228576(CHEMBL2092930)
Affinity DataKd:  80nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228577(CHEMBL1788224)
Affinity DataKd:  1.16E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataEC50:  100nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228578(CHEMBL111327)
Affinity DataKd:  4.95E+4nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228579(CHEMBL1788219)
Affinity DataKd:  6.32E+3nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228578(CHEMBL111327)
Affinity DataEC50:  7.50E+3nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50228570(CHEMBL1788202)
Affinity DataEC50:  94nMAssay Description:Compound was tested for its potency against Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50403547(ATROPEN | ATROPINE)
Affinity DataKd:  0.900nMAssay Description:Dissociation constant towards Muscarinic acetylcholine receptor in guinea pig ileumMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/15/2019
Entry Details Article
PubMed
LigandPNGBDBM50229065(CHEMBL262517)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229067(CHEMBL355824)
Affinity DataEC50:  320nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
LigandPNGBDBM50229047(CHEMBL159628)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at muscarinic acetylcholine receptor in isolated guinea pig ileum.More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/29/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50035277(3-Prop-2-ynyloxy-5,6,7,8-tetrahydro-4H-isoxazolo[4...)
Affinity DataEC50:  950nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50004656((2-Hydroxyethyl)trimethyl ammonium chloride carbam...)
Affinity DataEC50:  360nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50035279(3-Methoxy-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-c]az...)
Affinity DataEC50:  4.70E+3nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50004665(1-[4-(2-oxo-pyrrolidin-1-yl)-but-2-ynyl]-pyrrolidi...)
Affinity DataEC50:  55nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM46858(cid_9301 | ARECOLINE HYDROBROMIDE | SMR000058258 |...)
Affinity DataEC50:  600nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50035278(3-Ethoxy-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-c]aze...)
Affinity DataEC50:  2.10E+3nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50035280(3-Isopropoxy-5,6,7,8-tetrahydro-4H-isoxazolo[4,5-c...)
Affinity DataEC50:  110nMAssay Description:In Vitro activity at the cloned Human Muscarinic acetylcholine receptor M5 determined by receptor selection and amplification technology (R-SAT)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Human)
Vanderbilt Screening Center For Gpcrs, Ion Channels and Transporters

Curated by PubChem BioAssay
LigandPNGBDBM50263887(1-(1'-2-methylbenzyl)-1,4'-bipiperidin-4-yl)-1H-be...)
Affinity DataEC50: >3.00E+4nMAssay Description:Partial agonist activity at human muscarinic M5 receptor expressed in CHO cells calcium responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
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