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TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50023229(CHEMBL3329755)
Affinity DataEC50:  610nMAssay Description:Activity at rat muscarinic acetylcholine receptor subtype 5 expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/6/2016
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM43822(ethyl 4-[2-[(2-methylbenzoyl)amino]ethylamino]pipe...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356966(CHEMBL1916224)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356968(CHEMBL1916225)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356969(CHEMBL1916226)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356970(CHEMBL1916227)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356971(CHEMBL1916228)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356974(CHEMBL1916229)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356975(CHEMBL1916230)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356976(CHEMBL1916231)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356977(CHEMBL1916232)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356978(CHEMBL1916233)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356972(CHEMBL1916234)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356973(CHEMBL1916235)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at rat muscarinic M5 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM43822(ethyl 4-[2-[(2-methylbenzoyl)amino]ethylamino]pipe...)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant muscarinic M5 receptor by HTS cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50356966(CHEMBL1916224)
Affinity DataEC50: >3.00E+4nMAssay Description:Agonist activity at rat recombinant muscarinic M5 receptor by HTS cell based assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/21/2012
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423967(CHEMBL2057417)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50423968(CHEMBL2313377)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as acetylcholine responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50433574(CHEMBL2381694)
Affinity DataEC50:  0.224nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50433574(CHEMBL2381694)
Affinity DataEC50:  0.225nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  0.263nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  0.263nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptor assessed as effect on acetylcholine-induced responseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50433574(CHEMBL2381694)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50433574(CHEMBL2381694)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50258656(VU0238429 | CHEMBL466253 | cid_42633508 | 1-(4-met...)
Affinity DataEC50:  4.60nMAssay Description:Positive allosteric modulation of rat muscarinic M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50207463(CHEMBL3963788)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M5 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2018
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50207516(CHEMBL3942511)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M5 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2018
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50207517(CHEMBL3915634)
Affinity DataEC50: >3.00E+4nMAssay Description:Binding affinity to rat M5 receptor by radio-ligand binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/29/2018
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50249403(CHEMBL4091821)
Affinity DataEC50: >3.00E+4nMAssay Description:Activity at rat M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2019
Entry Details Article
PubMed
TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50546065(CHEMBL4795177)
Affinity DataEC50: >3.00E+4nMAssay Description:Positive allosteric modulation of rat M5 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2022
Entry Details Article
PubMed
LigandPNGBDBM50213281(CHEMBL351561)
Affinity DataIC50: 0.0200nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50213074(CHEMBL156050)
Affinity DataIC50: 0.0300nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50213283(CHEMBL350223)
Affinity DataIC50: 0.100nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50213207(CHEMBL160582)
Affinity DataIC50: 0.150nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50280565(5-(1-Aza-bicyclo[2.2.1]hept-3-yl)-[1,2,4]oxadiazol...)
Affinity DataIC50: 0.300nMAssay Description:Compound was evaluated for inhibition of [3H]cis-methyldioxolane binding to label agonist sites (RCMD) in rat neocortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetMuscarinic acetylcholine receptor M5(Rat)
Vanderbilt University Medical Center

Curated by ChEMBL
LigandPNGBDBM50426242(CHEMBL2312346)
Affinity DataIC50: 0.450nMAssay Description:Orthosteric antagonist activity at M5 muscarinic receptor in rat striatal slices assessed as inhibition of 100 uM oxotremorine-evoked [3H]DA releaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
LigandPNGBDBM50213070(CHEMBL405426)
Affinity DataIC50: 0.450nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50213278(CHEMBL156445)
Affinity DataIC50: 0.520nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50213077(CHEMBL348412)
Affinity DataIC50: 0.570nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50070692(CHEMBL99240)
Affinity DataIC50: 0.730nMAssay Description:Binding affinity against muscarinic receptor in rat brain membranes using oxotremorine-M as ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50291551(Trimethyl-[4-(3-oxo-isoxazolidin-2-yl)-but-2-ynyl]...)
Affinity DataIC50: 0.800nMAssay Description:Compound was assessed for the binding affinity against muscarinic receptor subtypes in rat brain using [3H]OXO-M radioligand as a muscarinic receptor...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2010
Entry Details Article

LigandPNGBDBM50072214((R)-3-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]thiadiaz...)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity against muscarinic receptor in rat brain membranes using oxotremorine-M as ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50213286(CHEMBL346580)
Affinity DataIC50: 0.800nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50065207(1-Aza-bicyclo[2.2.1]heptan-3-one O-((Z)-3-methyl-p...)
Affinity DataIC50: 1nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50049757((2R,4S)-2-(6-Iodo-pyridin-3-yl)-7-aza-bicyclo[2.2....)
Affinity DataIC50: 1nMAssay Description:In vitro displacement of [3H]oxotremorine-M from muscarinic acetylcholine receptor in rat brain cortexMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2020
Entry Details Article
PubMed
LigandPNGBDBM50213279(CHEMBL345415)
Affinity DataIC50: 1.10nMAssay Description:Binding affinity against muscarinic receptor using radioligand [3H]cis-methyldioxolane (CMD) binding assay in membrane preparations of rat neocortex.More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2018
Entry Details

LigandPNGBDBM50072227((1R,5R,6R)-6-[4-(3-Phenyl-prop-2-ynyloxy)-[1,2,5]t...)
Affinity DataIC50: 1.20nMAssay Description:Binding affinity against muscarinic receptor in rat brain membranes using oxotremorine-M as ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50070735(CHEMBL317324)
Affinity DataIC50: 1.20nMAssay Description:Binding affinity against muscarinic receptor in rat brain membranes using oxotremorine-M as ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
LigandPNGBDBM50070647(CHEMBL329924)
Affinity DataIC50: 1.30nMAssay Description:Binding affinity against muscarinic receptor in rat brain membranes using oxotremorine-M as ligandMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/29/2012
Entry Details Article
PubMed
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