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Report error Found 6 of affinity data for UniProtKB/TrEMBL: P04180
TargetPhosphatidylcholine-sterol acyltransferase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM303816((+)-4,5-Dihydroxy-4-(trifluoromethyl)-3-{1-[5-(tri...)
Affinity DataEC50:  4nMAssay Description:A fraction composed of HDL3 (1.125More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
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TargetPhosphatidylcholine-sterol acyltransferase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM303817((+)-cis-5-Hydroxy-4-(trifluoromethyl)-3-{1-[2-(tri...)
Affinity DataEC50:  18nMAssay Description:A fraction composed of HDL3 (1.125More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/29/2019
Entry Details
Go to US Patent

TargetPhosphatidylcholine-sterol acyltransferase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM92615(Difluoroketone phospholipid analogue, 3)
Affinity DataIC50: 28nMpH: 7.5 T: 2°CAssay Description:The phospholipase A2 activity of LCAT was assayed using lecithin and apoA-I containing [9,10-3H] dipalmitoylphosphatidylcholine (DPPC) and measuremen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details

TargetPhosphatidylcholine-sterol acyltransferase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM92614(Difluoroketone phospholipid analogue, 2)
Affinity DataIC50: 60nMpH: 7.5 T: 2°CAssay Description:The phospholipase A2 activity of LCAT was assayed using lecithin and apoA-I containing [9,10-3H] dipalmitoylphosphatidylcholine (DPPC) and measuremen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details

TargetPhosphatidylcholine-sterol acyltransferase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM92616(Difluoroketone phospholipid analogue, 4)
Affinity DataIC50: 60nMpH: 7.5 T: 2°CAssay Description:The phospholipase A2 activity of LCAT was assayed using lecithin and apoA-I containing [9,10-3H] dipalmitoylphosphatidylcholine (DPPC) and measuremen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details

TargetPhosphatidylcholine-sterol acyltransferase(Human)
Daiichi Sankyo

US Patent
LigandPNGBDBM92613(Difluoroketone phospholipid analogue, 1)
Affinity DataIC50: 500nMpH: 7.5 T: 2°CAssay Description:The phospholipase A2 activity of LCAT was assayed using lecithin and apoA-I containing [9,10-3H] dipalmitoylphosphatidylcholine (DPPC) and measuremen...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2012
Entry Details