Compile Data Set for Download or QSAR
Report error Found 590 for UniProtKB: P04054
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50236230(ursodeoxy cholic acid | 2-((R)-4-((3R,5S,7S,8R,9S,...)
Affinity DataKd:  1.00E+4nMAssay Description:Binding affinity to human pancreatic recombinant 1B PLA2 expressed in Escherichia coli by resonance energy transfer assay in presence of trimethyl-am...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM21680(Cholic Acid | (R)-4-((3R,5S,7R,8R,10S,12S,13R,14S,...)
Affinity DataKd: >1.50E+5nMAssay Description:Binding affinity to human pancreatic recombinant 1B PLA2 expressed in Escherichia coli by resonance energy transfer assay in presence of trimethyl-am...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053109([1-Aminooxalyl-3-(2-benzyl-benzyl)-2-ethyl-indoliz...)
Affinity DataIC50: 1.30nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053136((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methyl-indo...)
Affinity DataIC50: 1.40nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053106([1-Aminooxalyl-2-ethyl-3-(3-trifluoromethyl-benzyl...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053108((1-Aminooxalyl-3-benzyl-2-methyl-indolizin-8-yloxy...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053102([1-Aminooxalyl-3-(3-chloro-benzyl)-2-ethyl-indoliz...)
Affinity DataIC50: 3nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053114((1-Aminooxalyl-3-biphenyl-3-ylmethyl-2-ethyl-indol...)
Affinity DataIC50: 4.20nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053133((1-Aminooxalyl-3-benzyl-2-ethyl-indolizin-8-yloxy)...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053096([1-Aminooxalyl-3-(4-butyl-benzyl)-2-ethyl-indolizi...)
Affinity DataIC50: 5nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053123((1-Aminooxalyl-2-ethyl-3-naphthalen-1-ylmethyl-ind...)
Affinity DataIC50: 5nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053102([1-Aminooxalyl-3-(3-chloro-benzyl)-2-ethyl-indoliz...)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053137((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053109([1-Aminooxalyl-3-(2-benzyl-benzyl)-2-ethyl-indoliz...)
Affinity DataIC50: 6nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053147((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-cyclopropyl...)
Affinity DataIC50: 6nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053095((1-Aminooxalyl-2-ethyl-3-naphthalen-2-ylmethyl-ind...)
Affinity DataIC50: 7.30nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053108((1-Aminooxalyl-3-benzyl-2-methyl-indolizin-8-yloxy...)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053136((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methyl-indo...)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053133((1-Aminooxalyl-3-benzyl-2-ethyl-indolizin-8-yloxy)...)
Affinity DataIC50: 8nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053147((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-cyclopropyl...)
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053106([1-Aminooxalyl-2-ethyl-3-(3-trifluoromethyl-benzyl...)
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053114((1-Aminooxalyl-3-biphenyl-3-ylmethyl-2-ethyl-indol...)
Affinity DataIC50: 9nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053140((1-Aminooxalyl-3-[2,2']bithiophenyl-4-ylmethyl-2-e...)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053116((1-Aminooxalyl-3-cyclohexylmethyl-2-methyl-indoliz...)
Affinity DataIC50: 10nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053112((1-Aminooxalyl-2-ethyl-3-thiophen-2-ylmethyl-indol...)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053096([1-Aminooxalyl-3-(4-butyl-benzyl)-2-ethyl-indolizi...)
Affinity DataIC50: 11nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053140((1-Aminooxalyl-3-[2,2']bithiophenyl-4-ylmethyl-2-e...)
Affinity DataIC50: 11nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053104((3-Benzyl-1-carbamoylmethyl-2-ethyl-indolizin-8-yl...)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053112((1-Aminooxalyl-2-ethyl-3-thiophen-2-ylmethyl-indol...)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053139((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methoxy-ind...)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053113((3-Biphenyl-2-ylmethyl-1-carbamoylmethyl-2-cyclopr...)
Affinity DataIC50: 13nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053155((1-Aminooxalyl-3-biphenyl-4-ylmethyl-2-ethyl-indol...)
Affinity DataIC50: 13nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053125((3-Biphenyl-2-ylmethyl-1-carbamoylmethyl-2-ethyl-i...)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053141((1-Aminooxalyl-3-cyclopentylmethyl-2-methyl-indoli...)
Affinity DataIC50: 14nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053125((3-Biphenyl-2-ylmethyl-1-carbamoylmethyl-2-ethyl-i...)
Affinity DataIC50: 14nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053139((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methoxy-ind...)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053116((1-Aminooxalyl-3-cyclohexylmethyl-2-methyl-indoliz...)
Affinity DataIC50: 15nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053154([1-Carbamoylmethyl-3-(3-chloro-benzyl)-2-ethyl-ind...)
Affinity DataIC50: 15nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053110((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-methylsulfa...)
Affinity DataIC50: 16nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053095((1-Aminooxalyl-2-ethyl-3-naphthalen-2-ylmethyl-ind...)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053120((1-Aminooxalyl-3-biphenyl-2-ylmethyl-2-ethyl-indol...)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053143([1-Aminooxalyl-2-ethyl-3-(2-methyl-pentyl)-indoliz...)
Affinity DataIC50: 17nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053155((1-Aminooxalyl-3-biphenyl-4-ylmethyl-2-ethyl-indol...)
Affinity DataIC50: 18nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM82341(hnpsPLA2-IIa Inhibitor, 2l)
Affinity DataIC50: 19nMAssay Description:Compounds 2a-q were evaluated as inhibitors by using an in vitro colorimetric enzyme assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/23/2011
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053132((1-Aminooxalyl-3-cyclopentylmethyl-2-ethyl-indoliz...)
Affinity DataIC50: 19nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053132((1-Aminooxalyl-3-cyclopentylmethyl-2-ethyl-indoliz...)
Affinity DataIC50: 19nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053146([1-Aminooxalyl-2-ethyl-3-((S)-3-pentyl-cyclohexylm...)
Affinity DataIC50: 20nMAssay Description:Inhibitory activity against recombinant human secretory phospholipase A2 (s-PLA2) by phosphatidylcholine/deoxycholate assay (PC/DOC).More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053098((1-Aminooxalyl-3-cyclohexylmethyl-2-ethyl-indolizi...)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetPhospholipase A2(Human)
University of Delaware

Curated by ChEMBL
LigandPNGBDBM50053153([1-Aminooxalyl-2-ethyl-3-(3-methoxy-benzyl)-indoli...)
Affinity DataIC50: 21nMAssay Description:Inhibition of recombinant human secretory phospholipase A2 (sPLA2), chromogenic screening assay.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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