Compile Data Set for Download or QSAR
Report error Found 772 of affinity data for UniProtKB/TrEMBL: P03468
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50360450(CHEMBL1934618)
Affinity DataEC50:  1.35E+6nMAssay Description:Inhibition of Human influenza virus A/PR/8/34 (H1N1) neuraminidase using 4-MU-Neu5Ac as substrate after 30 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50360451(CHEMBL1934619)
Affinity DataEC50:  2.48E+6nMAssay Description:Inhibition of Human influenza virus A/PR/8/34 (H1N1) neuraminidase using 4-MU-Neu5Ac as substrate after 30 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50360452(CHEMBL1934620)
Affinity DataEC50:  7.43E+5nMAssay Description:Inhibition of Human influenza virus A/PR/8/34 (H1N1) neuraminidase using 4-MU-Neu5Ac as substrate after 30 mins by fluorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/22/2012
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM5003((3R,4R,5S)-5-amino-4-acetamido-3-{[(3S)-1-phenylpe...)
Affinity DataIC50: 0.300nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50097655((4S,5R,6R)-4-Amino-6-dipropylcarbamoyl-5-(2,2,2-tr...)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory activity against influenza A sialidase (Aichi)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM5011((3R,4R,5S)-3-[(2R)-butan-2-yloxy]-5-carbamimidamid...)
Affinity DataIC50: 0.5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM5012((3R,4R,5S)-4-Acetamido-5-guanidinyl-3-(1(S)-methyl...)
Affinity DataIC50: 0.5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM5013((3R,4R,5S)-4-Acetamido-5-guanidinyl-3-(1-ethylprop...)
Affinity DataIC50: 0.5nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 0.5nMAssay Description:Inhibitory activity was determined against Neuraminidase A from influenza virus A/Tokyo/3/67More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50598994(CHEMBL5192262)
Affinity DataIC50: 0.5nMAssay Description:Inhibition of Influenza A virus A/PR/8/1934 (H1N1) neuraminidase using MUNANA as substrate preincubated for 10 mins followed by substrate addition an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 0.524nMAssay Description:Inhibition of Influenza A virus A/PR/8/34(H1N1) sialidase preincubated for 15 mins followed by MUNA substrate addition measured after 15 mins by fluo...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 0.648nMAssay Description:Inhibition of Influenza A virus (H1N1) neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/12/2021
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50097648((4S,5R,6R)-4-Amino-6-(phenethyl-propyl-carbamoyl)-...)
Affinity DataIC50: 0.700nMAssay Description:Inhibitory activity against influenza A sialidase (Aichi)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50601844(CHEMBL5181864)
Affinity DataIC50: 0.730nMAssay Description:Inhibition of Influenza A virus A/PR/8/1934 (H1N1) neuraminidase using 2(4-methylurnbellifery1)-a-u-acetyl neuraminic acid sodium salt hydrate (4-MUN...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50165355((2R,4S)-3-(acetylamino)-4-{[(E)-amino(imino)methyl...)
Affinity DataIC50: 0.770nMAssay Description:Inhibitory concentration against neuraminidase of influenza A/Mem/Bel/71 (H3N1) virus starin; (n=5)More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50598999(CHEMBL5197351)
Affinity DataIC50: 0.950nMAssay Description:Inhibition of Influenza A virus A/PR/8/1934 (H1N1) neuraminidase using MUNANA as substrate preincubated for 10 mins followed by substrate addition an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 1nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4995((3R,4R,5S)-4-Acetamido-5-amino-3-[[(1S)-1-ethylbut...)
Affinity DataIC50: 1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4997((3R,4R,5S)-5-amino-3-[(3S)-decan-3-yloxy]-4-acetam...)
Affinity DataIC50: 1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM5000((3R,4R,5S)-4-Acetamido-5-amino-3-(1(S)-(2-cyclohex...)
Affinity DataIC50: 1nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 1nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/27/2005
Entry Details Article

TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 1nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/27/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 1nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/28/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4942((2R,3R,4S)-4-carbamimidamido-2-(diethylcarbamoyl)-...)
Affinity DataIC50: 1nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50028503(Guanidino-Oseltamivir Carboxylicacid | CHEMBL81717)
Affinity DataIC50: 1nMAssay Description:Inhibition of influenza A virus (A/WSN/1933(H1N1)) neuraminidase using MUNANA as fluorogenic substrate preincubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50028503(Guanidino-Oseltamivir Carboxylicacid | CHEMBL81717)
Affinity DataIC50: 1nMAssay Description:Inhibition of influenza A virus (A/WSN/1933(H1N1)) neuraminidase using MUNANA as fluorogenic substrate preincubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 1.17nMAssay Description:Inhibition of Influenza A PR/8/34 H1N1 virus neuraminidase activity by MUN-ANA substrate based fluorimetric assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50365361(CHEMBL4161935)
Affinity DataIC50: 1.20nMAssay Description:Inhibition of Influenza A virus (A/PuertoRico/8/1934(H1N1)) neuraminidase activity using 4-MUNANA as substrate preincubated for 10 mins followed by s...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/14/2020
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of influenza A viral enzyme neuraminidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/30/2012
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50529805(CHEMBL4562671)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of influenza A virus (A/WSN/1933(H1N1)) neuraminidase using MUNANA as fluorogenic substrate preincubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50529805(CHEMBL4562671)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of influenza A virus (A/WSN/1933(H1N1)) neuraminidase using MUNANA as fluorogenic substrate preincubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM5024((-)-(1S,2S,3R,4R)-3-[(1S)-1-(Acetylamino)-2-ethylb...)
Affinity DataIC50: 1.40nMAssay Description:inhibitory concentration required to inhibit neuraminidase enzyme from different strains of influenza A virusMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/15/2012
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 1.56nMAssay Description:Inhibition of human Influenza A virus A/PR/8/34(H1N1) neuraminidase by fluorometric method using 4MU-NeuAc substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/3/2013
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50219990(CHEMBL293938)
Affinity DataIC50: 1.78nMAssay Description:Inhibition of sialidase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/2/2018
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM5009(carbocyclic analogue 18 | (3R,4R,5S)-5-carbamimida...)
Affinity DataIC50: 1.80nMpH: 6.5 T: 2°CAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/27/2005
Entry Details Article

TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50289699((3R,4R,5S)-4-Acetylamino-5-guanidino-3-propoxy-cyc...)
Affinity DataIC50: 1.80nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/27/2005
Entry Details Article

TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50529806(CHEMBL4440605)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of influenza A virus (A/WSN/1933(H1N1)) neuraminidase using MUNANA as fluorogenic substrate preincubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of influenza A virus (A/WSN/1933(H1N1)) neuraminidase using MUNANA as fluorogenic substrate preincubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4994(CHEMBL674 | (3R,4R,5S)-5-amino-4-acetamido-3-(pent...)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of influenza A virus (A/WSN/1933(H1N1)) neuraminidase using MUNANA as fluorogenic substrate preincubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50529806(CHEMBL4440605)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of influenza A virus (A/WSN/1933(H1N1)) neuraminidase using MUNANA as fluorogenic substrate preincubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/26/2021
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50599004(CHEMBL5196029)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of Influenza A virus A/PR/8/1934 (H1N1) neuraminidase using MUNANA as substrate preincubated for 10 mins followed by substrate addition an...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/23/2023
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50469488(CHEMBL4287425)
Affinity DataIC50: 1.90nMAssay Description:Inhibition of Influenza A virus A/PR/8/1934 (H1N1) neuraminidase using 2(4-methylurnbellifery1)-a-u-acetyl neuraminic acid sodium salt hydrate (4-MUN...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/24/2023
Entry Details
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM5009(carbocyclic analogue 18 | (3R,4R,5S)-5-carbamimida...)
Affinity DataIC50: 2nMAssay Description:A standard fluorimetric assay was used to measure influenza virus neuraminidase activity. The substrate 2 -(4-methylumbelliferyl)-alpha-D-acetylneura...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2005
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4940((2R,3R,4S)-4-carbamimidamido-2-(dipropylcarbamoyl)...)
Affinity DataIC50: 2nMAssay Description:Inhibition of influenza sialidase was determined by measuring the ability to inhibit the hydrolysis of MUN by A/Aichi virus grown in hen eggsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/26/2012
Entry Details Article

TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4940((2R,3R,4S)-4-carbamimidamido-2-(dipropylcarbamoyl)...)
Affinity DataIC50: 2nMAssay Description:Inhibition of influenza A sialidase (neuraminidase)More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against influenza A virus sialidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4945((2R,3R,4S)-4-amino-3-acetamido-2-[(2-phenylethyl)(...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against influenza A virus sialidaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/27/2012
Entry Details Article

TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM50330326((4S,5R,6R)-5-Acetylamino-4-guanidino-6-((1R,3R)-1,...)
Affinity DataIC50: 2nMAssay Description:Inhibitory activity against influenza A sialidase (Aichi)More data for this Ligand-Target Pair
In Depth
Date in BDB:
10/4/2012
Entry Details Article
PubMed
TargetNeuraminidase(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)
Saitama University

Curated by ChEMBL
LigandPNGBDBM4945((2R,3R,4S)-4-amino-3-acetamido-2-[(2-phenylethyl)(...)
Affinity DataIC50: 2nMAssay Description:Compound was tested for inhibitory concentration against Influenza sialidase type AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2012
Entry Details Article
PubMed
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