Compile Data Set for Download or QSAR
Report error Found 236 of affinity data for UniProtKB/TrEMBL: P02829
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM20732(geldanomycin | GM-BODIPY | Geldanamycin | CHEMBL27...)
Affinity DataKd:  1.20E+3nMAssay Description:Binding affinity to N-terminal ATP/ADP-binding domain of yeast Hsp90More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50347503(RADICICOL)
Affinity DataKd:  19nMAssay Description:Binding affinity to N-terminal ATP/ADP-binding domain of yeast Hsp90More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/22/2012
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM15361(CHEMBL414883 | Monorden | (4R,6R,8R,9Z,11E)-16-chl...)
Affinity DataIC50: 30nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM15361(CHEMBL414883 | Monorden | (4R,6R,8R,9Z,11E)-16-chl...)
Affinity DataIC50: 47nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68248(Microlactone, 15a)
Affinity DataIC50: 100nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68256(Microlactone, 15c)
Affinity DataIC50: 100nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68263(Microlactone, 15h)
Affinity DataIC50: 100nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68248(Microlactone, 15a)
Affinity DataIC50: 120nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68250(Microlactone, 15b)
Affinity DataIC50: 160nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68263(Microlactone, 15h)
Affinity DataIC50: 160nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68264(Microlactone, 15i)
Affinity DataIC50: 160nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68249(Microlactone, 16a)
Affinity DataIC50: 190nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM15361(CHEMBL414883 | Monorden | (4R,6R,8R,9Z,11E)-16-chl...)
Affinity DataIC50: 200nMpH: 7.4 T: 2°CAssay Description:The HSP90 ATPase activity was determined by following the procedure of malachite green assay. The assay is based on quantitation of the green complex...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/4/2007
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM15361(CHEMBL414883 | Monorden | (4R,6R,8R,9Z,11E)-16-chl...)
Affinity DataIC50: 200nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68264(Microlactone, 15i)
Affinity DataIC50: 220nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68266(Microlactone, 15j)
Affinity DataIC50: 240nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68251(Microlactone, 16b)
Affinity DataIC50: 250nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68249(Microlactone, 16a)
Affinity DataIC50: 310nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68250(Microlactone, 15b)
Affinity DataIC50: 310nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68251(Microlactone, 16b)
Affinity DataIC50: 310nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68255(Microlactone, 14c)
Affinity DataIC50: 500nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68260(Microlactone, 15f cis)
Affinity DataIC50: 500nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68255(Microlactone, 14c)
Affinity DataIC50: 540nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68261(Microlactone, 15f trans)
Affinity DataIC50: 590nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68263(Microlactone, 15h)
Affinity DataIC50: 760nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68260(Microlactone, 15f cis)
Affinity DataIC50: 850nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68266(Microlactone, 15j)
Affinity DataIC50: 870nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68248(Microlactone, 15a)
Affinity DataIC50: 1.00E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68250(Microlactone, 15b)
Affinity DataIC50: 1.00E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68256(Microlactone, 15c)
Affinity DataIC50: 1.00E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68256(Microlactone, 15c)
Affinity DataIC50: 1.00E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68261(Microlactone, 15f trans)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68265(Microlactone, 18)
Affinity DataIC50: 1.10E+3nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68252(Microlactone, 17)
Affinity DataIC50: 1.29E+3nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68248(Microlactone, 15a)
Affinity DataIC50: 1.30E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68250(Microlactone, 15b)
Affinity DataIC50: 1.50E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50409989(CHEMBL361941)
Affinity DataIC50: 1.55E+3nMAssay Description:Inhibition of yeast Hsp90 ATPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50409996(CHEMBL191228)
Affinity DataIC50: 1.60E+3nMAssay Description:Inhibition of yeast Hsp90 ATPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50409992(CHEMBL364882)
Affinity DataIC50: 1.65E+3nMAssay Description:Inhibition of yeast Hsp90 ATPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68251(Microlactone, 16b)
Affinity DataIC50: 1.90E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68259(Microlactone, 15e)
Affinity DataIC50: 1.90E+3nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68249(Microlactone, 16a)
Affinity DataIC50: 2.10E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68258(Microlactone, 19)
Affinity DataIC50: 2.10E+3nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM20732(geldanomycin | GM-BODIPY | Geldanamycin | CHEMBL27...)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of yeast Hsp90 ATPase activity by ATPase assay using malachite green colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/27/2010
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68260(Microlactone, 15f cis)
Affinity DataIC50: 2.40E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50409990(CHEMBL190249)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of yeast Hsp90 ATPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM50409994(CHEMBL188495)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of yeast Hsp90 ATPase activityMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/20/2013
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68249(Microlactone, 16a)
Affinity DataIC50: 2.50E+3nMAssay Description:A colorimetric assay for the release of inorganic phosphate upon hydrolysis of ATP was used to determine the potency of Hsp 90 inhibitor against enzy...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68265(Microlactone, 18)
Affinity DataIC50: 2.63E+3nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
TargetATP-dependent molecular chaperone HSP82(Baker's yeast)
Memorial Sloan-Kettering Cancer Center

Curated by ChEMBL
LigandPNGBDBM68258(Microlactone, 19)
Affinity DataIC50: 2.90E+3nMAssay Description:Binding competition assay with a fluorescent probe.More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/15/2011
Entry Details Article
PubMed
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