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TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50423921(CHEMBL2312756)
Affinity DataKd:  2.80E+3nMAssay Description:Binding affinity to human c-Myc bHLH-ZIP domain (353 to 437 amino acid residues) expressed in Escherichia coli BL21 (DE3) by fluorescence polarizatio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50148027(CHEMBL3765705 | US20240287089, Compound LMP517)
Affinity DataKd:  109nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694224(US20240287089, Compound LMP776)
Affinity DataKd:  69nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50237809(CHEMBL126159 | US20240287089, Compound LMP744)
Affinity DataKd:  11nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694222(US20240287089, Compound LMP400)
Affinity DataKd:  301nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694221(US20240287089, Compound G108)
Affinity DataKd:  14nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694220(US20240287089, Compound G107)
Affinity DataKd:  59nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694219(US20240287089, Compound G106)
Affinity DataKd:  55nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694218(US20240287089, Compound G105)
Affinity DataKd:  97nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694217(US20240287089, Compound G104)
Affinity DataKd:  55nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694216(US20240287089, Compound G103)
Affinity DataKd:  77nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694215(US20240287089, Compound G102)
Affinity DataKd:  147nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM694214(US20240287089, Compound G101)
Affinity DataKd:  249nMAssay Description:MycG4 Stabilization Measured by FRET Melting. A F rster Resonance Energy Transfer (FRET)-melting assay was conducted in order to determine whether th...More data for this Ligand-Target Pair
Ligand InfoSimilars
In Depth
Date in BDB:
12/12/2024
Entry Details
Go to US Patent

TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50498222(CHEMBL3427045)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to human recombinant 15N labeled c-Myc-Max(S) heterodimer assessed as chemical shift up to 100 uM by NMR spectroscopyMore data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463126(CHEMBL4238599)
Affinity DataKd:  6.5nMAssay Description:Binding affinity to His-tagged Myc (unknown origin) expressed in Escherichia coli BL21 by Bio-FET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463128(CHEMBL4249055)
Affinity DataKd:  13nMAssay Description:Binding affinity to His-tagged Myc (unknown origin) expressed in Escherichia coli BL21 by Bio-FET analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM445524(US10683290, Example 16 | 2-{7-[4-(2H3)Methyl-1-met...)
Affinity DataIC50: 0.200nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM445528(US10683290, Example 20 | 2-[7-(Dimethyl-1H-1,2,3-t...)
Affinity DataIC50: 0.600nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM296947(US10112941, Example 54 | 2-[3-(Dimethyl-1H-1,2,3-t...)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50579853(CHEMBL5075294)
Affinity DataIC50: 0.700nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM445527(US10683290, Example 19 | 2-[7-(Dimethyl-1H-1,2,3-t...)
Affinity DataIC50: 0.800nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM445527(US10683290, Example 19 | 2-[7-(Dimethyl-1H-1,2,3-t...)
Affinity DataIC50: 1nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50579851(CHEMBL5084198)
Affinity DataIC50: 1.30nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50579852(CHEMBL5090513)
Affinity DataIC50: 2.40nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM445515(US10683290, Example 11 | 2-[7-(Dimethyl-1H-1,2,3-t...)
Affinity DataIC50: 3.40nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM331520(US9725449, Example 364 | BDBM331524 | 2-{11-[4-(2H...)
Affinity DataIC50: 6.90nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM445584(US10683290, Example 77)
Affinity DataIC50: 42nMAssay Description:Inhibition of c-MYC (unknown origin)More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/4/2023
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463126(CHEMBL4238599)
Affinity DataIC50: 1.00E+3nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463135(CHEMBL4243878)
Affinity DataIC50: 2.00E+3nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463127(CHEMBL4237402)
Affinity DataIC50: 2.50E+3nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463138(CHEMBL4240401)
Affinity DataIC50: 3.00E+3nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463140(CHEMBL4240109)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463128(CHEMBL4249055)
Affinity DataIC50: 5.00E+3nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50498221(CHEMBL3427016)
Affinity DataIC50: 5.60E+3nMAssay Description:Disruption of human recombinant c-Myc-Max/DNA (unknown origin) binding assessed as complex level by electrophoretic mobility shift assay relative to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463131(CHEMBL4248559)
Affinity DataIC50: 7.00E+3nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50520737(CHEMBL4467662)
Affinity DataIC50: 8.90E+3nMAssay Description:Inhibition of Myc-Max (unknown origin) expressed in human LNCAP cells assessed as reduction in transcriptional activity after 1 day by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463139(CHEMBL4243533)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463134(CHEMBL4246868)
Affinity DataIC50: 1.00E+4nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50498222(CHEMBL3427045)
Affinity DataIC50: 1.16E+4nMAssay Description:Disruption of human recombinant c-Myc-Max/DNA (unknown origin) binding assessed as complex level by electrophoretic mobility shift assay relative to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50498221(CHEMBL3427016)
Affinity DataIC50: 1.25E+4nMAssay Description:Disruption of human recombinant Myc(L)-Max(L)/DNA (unknown origin) binding assessed as complex level by electrophoretic mobility shift assay relative...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50498222(CHEMBL3427045)
Affinity DataIC50: 2.00E+4nMAssay Description:Disruption of human recombinant Myc(L)-Max(L)/DNA (unknown origin) binding assessed as complex level by electrophoretic mobility shift assay relative...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50498219(CHEMBL3427047)
Affinity DataIC50: 2.02E+4nMAssay Description:Disruption of human recombinant c-Myc-Max/DNA (unknown origin) binding assessed as complex level by electrophoretic mobility shift assay relative to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50520738(CHEMBL224118)
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of Myc-Max (unknown origin) expressed in human LNCAP cells assessed as reduction in transcriptional activity after 1 day by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50498217(CHEMBL3427021)
Affinity DataIC50: 2.38E+4nMAssay Description:Disruption of human recombinant c-Myc-Max/DNA (unknown origin) binding assessed as complex level by electrophoretic mobility shift assay relative to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50520739(CHEMBL443375)
Affinity DataIC50: 2.89E+4nMAssay Description:Inhibition of Myc-Max (unknown origin) expressed in human LNCAP cells assessed as reduction in transcriptional activity after 1 day by luciferase rep...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463130(CHEMBL4247460)
Affinity DataIC50: 3.00E+4nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM93880(4-(7-Nitro-benzo[1,2,5]oxadiazol-4-ylamino)-benzoi...)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of recombinant His6-tagged c-Myc bHLH-ZIP domain (353 to 437 amino acid residues) (unknown origin) assessed as disruption of Myc-Max dimer...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/24/2013
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463129(CHEMBL4245253)
Affinity DataIC50: 4.00E+4nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50463141(CHEMBL4244986)
Affinity DataIC50: 4.00E+4nMAssay Description:Binding affinity to ATG-Myc (unknown origin) expressed in CEF cells assessed as inhibition of microtumor formationMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetMyc proto-oncogene protein/Protein max(Human)
University of Maryland

Curated by ChEMBL
LigandPNGBDBM50498218(CHEMBL3427054)
Affinity DataIC50: 4.30E+4nMAssay Description:Disruption of human recombinant c-Myc-Max/DNA (unknown origin) binding assessed as complex level by electrophoretic mobility shift assay relative to ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
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