Compile Data Set for Download or QSAR
Report error Found 174 of affinity data for UniProtKB/TrEMBL: P00730
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50365328(CHEMBL1955927)
Affinity DataIC50: 250nMAssay Description:Inhibition of bovine pancreas carboxypeptidase A using N-(4-methoxyphenylazoformyl)-phenylalanine as substrate after 5 mins by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283501(CHEMBL4167456)
Affinity DataIC50: 260nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283541(CHEMBL4176703)
Affinity DataIC50: 470nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283502(CHEMBL4168849)
Affinity DataIC50: 510nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283507(CHEMBL4163047)
Affinity DataIC50: 570nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50277985(CHEMBL4166112)
Affinity DataIC50: 750nMAssay Description:Inhibition of bovine pancreas carboxypeptidase A using N-4-(methoxyphenylazoformyl)-Phe-OH as substrate measured after 5 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283499(CHEMBL4173339)
Affinity DataIC50: 960nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283496(CHEMBL4169911)
Affinity DataIC50: 970nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283497(CHEMBL4165424)
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283505(CHEMBL4159372)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283508(CHEMBL4161983)
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283500(CHEMBL4166484)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283500(CHEMBL4166484)
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50277995(CHEMBL4159803)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of bovine pancreas carboxypeptidase A using N-4-(methoxyphenylazoformyl)-Phe-OH as substrate measured after 5 mins by colorimetric methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/4/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50478892(Anabaenopeptin T)
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of carboxypeptidase A in bovine pancreas assessed as reduction in hydrolysis of hippuryl-L-phenylalanine using hippuryl-L-phenylalanine as...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/27/2022
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50236983(2-hydroxycyclohepta-2,4,6-trienone | tropolone | 2...)
Affinity DataIC50: 2.73E+3nMAssay Description:Inhibition of Bos taurus (bovine) pancrease carboxypeptidase A after 15 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50330794(2-Hydroxy-4-isopropyl-cyclohepta-2,4,6-trienone | ...)
Affinity DataIC50: 2.76E+3nMAssay Description:Inhibition of Bos taurus (bovine) pancrease carboxypeptidase A after 15 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21478((2S)-2-{[(1S)-2-(1-benzyl-1H-imidazol-5-yl)-1-carb...)
Affinity DataIC50: 2.80E+3nMpH: 7.5 T: 2°CAssay Description:Assay for the inhibition of carboxypeptidase A (CPDA) was conducted in 96-well microplates format. Activity was monitored by measuring decrease in ab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50365329(CHEMBL1955931)
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of bovine pancreas carboxypeptidase A using N-(4-methoxyphenylazoformyl)-phenylalanine as substrate after 5 mins by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/23/2012
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283494(CHEMBL4175727)
Affinity DataIC50: 8.25E+3nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21482((2S)-2-{[(1S)-1-carboxy-2-{1-[(4-chlorophenyl)meth...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Assay for the inhibition of carboxypeptidase A (CPDA) was conducted in 96-well microplates format. Activity was monitored by measuring decrease in ab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21484((2S)-2-{[(1S)-1-carboxy-2-{1-[(4-methylphenyl)meth...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Assay for the inhibition of carboxypeptidase A (CPDA) was conducted in 96-well microplates format. Activity was monitored by measuring decrease in ab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21486((2S)-2-{[(1S)-1-carboxy-2-{1-[(3-methylphenyl)meth...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Assay for the inhibition of carboxypeptidase A (CPDA) was conducted in 96-well microplates format. Activity was monitored by measuring decrease in ab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21487((2S)-2-{[(1S)-1-carboxy-2-{1-[(3,4-dimethylphenyl)...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Assay for the inhibition of carboxypeptidase A (CPDA) was conducted in 96-well microplates format. Activity was monitored by measuring decrease in ab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21488((2S)-2-{[(1S)-1-carboxy-2-{1-[(3,5-dimethylphenyl)...)
Affinity DataIC50: 1.00E+4nMpH: 7.5 T: 2°CAssay Description:Assay for the inhibition of carboxypeptidase A (CPDA) was conducted in 96-well microplates format. Activity was monitored by measuring decrease in ab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283506(CHEMBL4177108)
Affinity DataIC50: 1.12E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21491((2S)-2-{[(1S)-1-carboxy-2-[1-(2-cyclohexylpropan-2...)
Affinity DataIC50: 1.20E+4nMpH: 7.5 T: 2°CAssay Description:Assay for the inhibition of carboxypeptidase A (CPDA) was conducted in 96-well microplates format. Activity was monitored by measuring decrease in ab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283501(CHEMBL4167456)
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283538(CHEMBL4165531)
Affinity DataIC50: 1.64E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283541(CHEMBL4176703)
Affinity DataIC50: 1.87E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283502(CHEMBL4168849)
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21489(MLN4760 | (2S)-2-{[(1S)-1-carboxy-2-{1-[(3,5-dichl...)
Affinity DataIC50: 2.70E+4nMpH: 7.5 T: 2°CAssay Description:Assay for the inhibition of carboxypeptidase A (CPDA) was conducted in 96-well microplates format. Activity was monitored by measuring decrease in ab...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50289561(4-tert-Butyl-benzoic acid [1-(2-hydroxy-naphthalen...)
Affinity DataIC50: 2.90E+4nMAssay Description:Inhibitory concentration required to inhibit carboxypeptidase A (CPA, bovine, Type I) was evaluatedMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/21/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283495(CHEMBL4172319)
Affinity DataIC50: 3.18E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283495(CHEMBL4172319)
Affinity DataIC50: 3.19E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283504(CHEMBL4159548)
Affinity DataIC50: 3.19E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283503(CHEMBL4173750)
Affinity DataIC50: 3.31E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 3 hrs followed by susbtrate addition ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283499(CHEMBL4173339)
Affinity DataIC50: 4.63E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283497(CHEMBL4165424)
Affinity DataIC50: 4.83E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283508(CHEMBL4161983)
Affinity DataIC50: 5.79E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283496(CHEMBL4169911)
Affinity DataIC50: 6.00E+4nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283505(CHEMBL4159372)
Affinity DataIC50: 1.15E+5nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50283506(CHEMBL4177108)
Affinity DataIC50: 2.76E+5nMAssay Description:Inhibition of bovine carboxypeptidase A using N-(4-methoxyphenylazoformyl)-Phe-OH as substrate preincubated for 2 mins followed by susbtrate addition...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/5/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50092158(CHEMBL415879 | cid_1318 | 1,10-phenanthroline | US...)
Affinity DataIC50: 4.22E+5nMAssay Description:Inhibition of Bos taurus (bovine) pancrease carboxypeptidase A after 15 minMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/31/2020
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21471(2-benzyl-3-{[1-(2-acetamido-4-methylpentanamido)-2...)
Affinity DataKi:  0.300nMAssay Description:Continuous assays were performed by recording the fluorescence increase at 405 nm (excitation@ 320 nm) induced by the cleavage of fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM21464(The second fraction of the HPLC chromatogram. | 2-...)
Affinity DataKi:  0.5nMAssay Description:Continuous assays were performed by recording the fluorescence increase at 405 nm (excitation@ 320 nm) induced by the cleavage of fluorogenic substra...More data for this Ligand-Target Pair
In Depth
Date in BDB:
4/18/2008
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50109593(SQ-14603 | 2-Mercaptomethyl-3-phenyl-propionic aci...)
Affinity DataKi:  10nMAssay Description:Inhibition of bovine carboxypeptidase A (CPA) using hippuryl-L-phenylalanine (Hipp-L-Phe) as a substrate.More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50109593(SQ-14603 | 2-Mercaptomethyl-3-phenyl-propionic aci...)
Affinity DataKi:  11nMAssay Description:Inhibition of bovine pancreatic carboxypeptidase AMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/11/2009
Entry Details Article
PubMed
TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50109593(SQ-14603 | 2-Mercaptomethyl-3-phenyl-propionic aci...)
Affinity DataKi:  11nMAssay Description:Binding affinity against carboxypeptidase A using hippurylphenylalanine as substrateMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

TargetCarboxypeptidase A1(Bovine)
National Institute of Diabetes and Digestive and Kidney Diseases

Curated by ChEMBL
LigandPNGBDBM50109593(SQ-14603 | 2-Mercaptomethyl-3-phenyl-propionic aci...)
Affinity DataKi:  11nMAssay Description:Compound was evaluated for binding affinity against carboxypeptidase A (CPA), expressed as inhibitory constant (Ki)More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2010
Entry Details Article

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