Compile Data Set for Download or QSAR
Report error Found 7 of affinity data for UniProtKB/TrEMBL: P00546
TargetCyclin-dependent kinase 1(Baker's yeast)
University of California

Curated by ChEMBL
LigandPNGBDBM27216((2R)-2-({6-[(3-chlorophenyl)amino]-9-(propan-2-yl)...)
Affinity DataIC50: 80nMAssay Description:Inhibition of Saccharomyces cerevisiae cdc28More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Baker's yeast)
University of California

Curated by ChEMBL
LigandPNGBDBM7478(CHEMBL23254 | 2-chloro-4-[(2-{[(2R)-1-hydroxy-3-me...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of Saccharomyces cerevisiae cdc28More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Baker's yeast)
University of California

Curated by ChEMBL
LigandPNGBDBM7377(CHEMBL75680 | aloisine A | 7-n-Butyl-6-(4-hydroxyp...)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of hemagglutininin-tagged Saccharomyces cerevisiae MNY629 Cdc28/Clb2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Baker's yeast)
University of California

Curated by ChEMBL
LigandPNGBDBM50113707(2,6,9-Trisubstitute purine, 2 | CHEMBL311228 | 2-[...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of yeast W303 cdc28 phosphorylation assessed as [32P] incorporation in histone H1 from [gamma32P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Baker's yeast)
University of California

Curated by ChEMBL
LigandPNGBDBM50129555(CHEMBL70590 | cid_310900 | 2-((1S,8R,9S,11R,13S,15...)
Affinity DataIC50: 2.40E+4nMAssay Description:Inhibition of cyclin-dependent kinase activity of Cdc28p/CDK2p in Saccharomyces cerevisiaeMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Baker's yeast)
University of California

Curated by ChEMBL
LigandPNGBDBM50295351(N-methyl-aloisine A | CHEMBL560452)
Affinity DataIC50: 3.30E+4nMAssay Description:Inhibition of hemagglutininin-tagged Saccharomyces cerevisiae MNY629 Cdc28/Clb2More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/26/2010
Entry Details Article
PubMed
TargetCyclin-dependent kinase 1(Baker's yeast)
University of California

Curated by ChEMBL
LigandPNGBDBM50267719(2-(6-((3-chlorophenyl)(methyl)amino)-9-isopropyl-9...)
Affinity DataIC50: 5.00E+5nMAssay Description:Inhibition of yeast W303 cdc28 phosphorylation assessed as [32P] incorporation in histone H1 from [gamma32P]ATP by scintillation countingMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/21/2012
Entry Details Article
PubMed