Compile Data Set for Download or QSAR
Report error Found 799 of affinity data for UniProtKB/TrEMBL: P00489
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM23210((1S,2R,4aS,6aS,6bR,8R,9R,10R,11R,12aR,12bR,14bS)-8...)
Affinity DatapH: 7.2 T: 2°CAssay Description:The activity of the compounds is determined by measuring the inhibitory effect of the compounds in the direction of glycogen synthesis, the conversio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM23211((2S,3R,4S,5S,6R)-6-({[(2R,3R,4R,5S,6R)-3,4-dihydro...)
Affinity DatapH: 7.2 T: 2°CAssay Description:The activity of the compounds is determined by measuring the inhibitory effect of the compounds in the direction of glycogen synthesis, the conversio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM23212((2S,3R,4S,5S,6R)-6-({[(2R,3R,4R,5S,6R)-3,4-dihydro...)
Affinity DatapH: 7.2 T: 2°CAssay Description:The activity of the compounds is determined by measuring the inhibitory effect of the compounds in the direction of glycogen synthesis, the conversio...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/29/2008
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM35332(2-oxo-1,2-dihydropyridin-3-yl amide derivative, 7u)
Affinity DatapH: 7.2 T: 2°CAssay Description:RMGPa (Rabbit Muscle Glycogen Phosphorylase a) activity was measured in the direction of glycogen synthesis by the formation of inorganic phosphate f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50277972([5-(6-Amino-9-phenethyl-9H-purin-8-yl)-furan-2-yl]...)
Affinity DataEC50: >2.50E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50277565({5-[6-Amino-9-(2,2-dimethyl-propyl)-9H-purin-8-yl]...)
Affinity DataEC50: >1.00E+5nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
1/11/2010
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50133435(4-(2-Chloro-phenyl)-1-ethyl-6-methyl-1,4-dihydro-p...)
Affinity DataIC50: 1.60nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50497973(CHEMBL3323454)
Affinity DataIC50: 7nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase a assessed as inhibition of release of phosphate from glucose-1-phosphate after 30 mins by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50382964(CHEMBL2030481)
Affinity DataIC50: 24nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50497969(CHEMBL3323453)
Affinity DataIC50: 45nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase a assessed as inhibition of release of phosphate from glucose-1-phosphate after 30 mins by spectro...More data for this Ligand-Target Pair
In Depth
Date in BDB:
9/3/2020
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50196903(CHEMBL3916767)
Affinity DataIC50: 178nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase b using 10 mM of glucose-1-phosphate as substrate preincubated for 60 mins followed by substrate a...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/13/2018
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50334099(2-((4R,5R,8R,9R,10R,13S,14R,15R)-4-(carboxymethyl)...)
Affinity DataIC50: 210nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50194701((2R,3R,4R)-2-Hydroxymethylpyrrolidin-3,4-diol hydr...)
Affinity DataIC50: 330nMAssay Description:Inhibition of phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50194701((2R,3R,4R)-2-Hydroxymethylpyrrolidin-3,4-diol hydr...)
Affinity DataIC50: 390nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM34110(glucopyranosylidene-spiro-isoxazoline, 4e)
Affinity DataIC50: 630nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50182801(CHEMBL206468 | AFEGOSTAT TARTRATE | D-Isofagomine ...)
Affinity DataIC50: 760nMAssay Description:Inhibition of phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50194702((3R,4R,5R)-5-(HYDROXYMETHYL)-1-(3-PHENYLPROPYL)PIP...)
Affinity DataIC50: 840nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50382963(CHEMBL2030480)
Affinity DataIC50: 900nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346702(CHEMBL574993)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346702(CHEMBL574993)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase a assessed as glycogen synthesisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/25/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346677(CHEMBL1796866)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50310522(2alpha-Hydroxyurs-12-en-28-oic acid | CHEMBL107884...)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase assessed as release of phosphate from glucose-1-phosphate after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM5655(2-(2-chlorophenyl)-5,7-dihydroxy-8-[(3S,4R)-3-hydr...)
Affinity DataIC50: 1.20E+3nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50182801(CHEMBL206468 | AFEGOSTAT TARTRATE | D-Isofagomine ...)
Affinity DataIC50: 1.21E+3nMAssay Description:Inhibition of non-phosphorylated form of rabbit muscle glycogen phosphorylaseMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346595(CHEMBL1797018)
Affinity DataIC50: 1.25E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346692(CHEMBL1797010)
Affinity DataIC50: 1.51E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50146082(CHEMBL3763876)
Affinity DataIC50: 1.54E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase bMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/16/2017
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50150651(CHEMBL3769527)
Affinity DataIC50: 1.92E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase-a assessed as formation of inorganic phosphate from glucose-1-phosphate by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50150650(CHEMBL3769814)
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase-a assessed as formation of inorganic phosphate from glucose-1-phosphate by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346683(CHEMBL1796873)
Affinity DataIC50: 2.13E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346688(CHEMBL1796878)
Affinity DataIC50: 2.23E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50150653(CHEMBL3770692)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase-a assessed as formation of inorganic phosphate from glucose-1-phosphate by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346694(CHEMBL1797012)
Affinity DataIC50: 2.59E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM34072(benzamide derivative, 12)
Affinity DataIC50: 2.68E+3nMpH: 7.2 T: 2°CAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50382965(CHEMBL2030483)
Affinity DataIC50: 2.70E+3nMAssay Description:Binding affinity to rabbit muscular GPa by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50334100(methyl 2-((4R,5R,8R,9R,10R,13S,14R,15R)-4-(2-metho...)
Affinity DataIC50: 2.87E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase aMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/22/2011
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50350687(CHEMBL1814684)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346598(CHEMBL1797021)
Affinity DataIC50: 3.07E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50263768(BETA-D-GLUCOPYRANOSE SPIROHYDANTOIN | (5S,7R,8S,9S...)
Affinity DataIC50: 3.10E+3nMAssay Description:Binding affinity to rabbit muscular GPb by NMR binding assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50310509((4aS,6aS,6bR,8aS,12aS,12bR,14bS)-benzyl 2,2,6a,6b,...)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase assessed as release of phosphate from glucose-1-phosphate after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50350688(CHEMBL1814498)
Affinity DataIC50: 3.20E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase 1a assessed as release of phosphate from glucose-1- phosphate after 20 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50310509((4aS,6aS,6bR,8aS,12aS,12bR,14bS)-benzyl 2,2,6a,6b,...)
Affinity DataIC50: 3.24E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346689(CHEMBL1796879)
Affinity DataIC50: 3.25E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346670(CHEMBL238219)
Affinity DataIC50: 3.26E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50346608(CHEMBL1797139)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 mins by microplate reader bas...More data for this Ligand-Target Pair
In Depth
Date in BDB:
3/23/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50184615((4aS,6aS,6bR,10S,12aR,14bS,E)-10-(3-(4-chloropheny...)
Affinity DataIC50: 3.30E+3nMAssay Description:Inhibition of rabbit muscle GPaMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/7/2012
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50150645(CHEMBL3771019)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase-a assessed as formation of inorganic phosphate from glucose-1-phosphate by colorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
6/27/2017
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM34074(benzamide derivative, 13b)
Affinity DataIC50: 3.50E+3nMpH: 7.2 T: 2°CAssay Description:The enzymatic inhibition of phosphorylase activity was monitored using microplate reader (Bio-Rad). In brief, GPa activity was measured in the direct...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/9/2009
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50310507(2-isooleanolic acid | CHEMBL1080965)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase assessed as release of phosphate from glucose-1-phosphate after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/17/2010
Entry Details Article
PubMed
TargetGlycogen phosphorylase, muscle form(Rabbit)
China Pharmaceutical University

LigandPNGBDBM50303206(((1R,3aS,5aR,5bR,7aR,8R,9S,11aR,11bR,13bR)-9-aceto...)
Affinity DataIC50: 3.50E+3nMAssay Description:Inhibition of rabbit muscle glycogen phosphorylase A assessed as release of phosphate from glucose-1-phosphate after 25 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/27/2012
Entry Details Article
PubMed
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