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Report error Found 6 of affinity data for UniProtKB/TrEMBL: O54698
TargetEquilibrative nucleoside transporter 1(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM23617(NBTI | Nitrobenzylthioinosine | CHEMBL418509 | (2R...)
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration against human Adenosine A3 receptor expressed in HEK293 cells using 0.1 nM [3H]AB-MECAMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/5/2012
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50241166(N6-benzylado | CHEMBL388757 | (2R,3R,4S,5R)-2-(6-(...)
Affinity DataKi:  203nMAssay Description:Inhibition of [3H]S-(4-Nitrobenzyl)-6-thioinosine binding to adenosine uptake sites in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50367298(Cardene | NICARDIPINE)
Affinity DataKi:  5.36E+3nMAssay Description:Ability to displace radioligand from Na+ independent Adenosine transporter in ratMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/1/2012
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM21221(2-Cl-IB-MECA | CHEMBL431733 | C-IBzA-MU | 2-chloro...)
Affinity DataKi:  1.52E+4nMAssay Description:Inhibition of [3H]S-(4-Nitrobenzyl)-6-thioinosine binding to adenosine uptake sites in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50118812(CHEMBL119709 | (3S,4R,5R)-3,4-Dihydroxy-5-[6-(3-io...)
Affinity DataKi:  2.82E+4nMAssay Description:Inhibition of [3H]S-(4-Nitrobenzyl)-6-thioinosine binding to adenosine uptake sites in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed
TargetEquilibrative nucleoside transporter 1(Rat)
University of Urbino

Curated by ChEMBL
LigandPNGBDBM50407234(CHEMBL2113557)
Affinity DataKi:  4.95E+4nMAssay Description:Inhibition of [3H]S-(4-Nitrobenzyl)-6-thioinosine binding to adenosine uptake sites in rat brain membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
10/28/2012
Entry Details Article
PubMed